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CAS No: 7773-06-0 Catalog No: AG0013OX MDL No:MFCD00011429
Title | Journal |
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Betulinyl Sulfamates as Anticancer Agents and Radiosensitizers in Human Breast Cancer Cells. | International journal of molecular sciences 20151101 |
Ethylenediammonium dication: H-bonded complexes with terephthalate, chloroacetate, phosphite, selenite and sulfamate anions. Detailed vibrational spectroscopic and theoretical studies of ethylenediammonium terephthalate. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20121201 |
Efficacious N-protection of O-aryl sulfamates with 2,4-dimethoxybenzyl groups. | Organic & biomolecular chemistry 20121007 |
A modular synthesis of dithiocarbamate pendant unnatural α-amino acids. | Chemical communications (Cambridge, England) 20120914 |
Measurement of nitrosamine and nitramine formation from NOx reactions with amines during amine-based carbon dioxide capture for postcombustion carbon sequestration. | Environmental science & technology 20120904 |
Sulfamate proton solvent exchange in heparin oligosaccharides: evidence for a persistent hydrogen bond in the antithrombin-binding pentasaccharide Arixtra. | Glycobiology 20120901 |
Acyl-sulfamates target the essential glycerol-phosphate acyltransferase (PlsY) in Gram-positive bacteria. | Bioorganic & medicinal chemistry 20120815 |
Comparison of arylboron-based nucleophiles in Ni-catalyzed Suzuki-Miyaura cross-coupling with aryl mesylates and sulfamates. | The Journal of organic chemistry 20120720 |
Ureido-substituted sulfamates show potent carbonic anhydrase IX inhibitory and antiproliferative activities against breast cancer cell lines. | Bioorganic & medicinal chemistry letters 20120715 |
Modular functionalization of allenes to aminated stereotriads. | Journal of the American Chemical Society 20120704 |
Palladium-catalysed aminosulfonylation of aryl-, alkenyl- and heteroaryl halides: scope of the three-component synthesis of N-aminosulfonamides. | Organic & biomolecular chemistry 20120528 |
Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors. | The Journal of organic chemistry 20120504 |
Hydrolysis of N-alkyl sulfamates and the catalytic efficiency of an S-N cleaving sulfamidase. | The Journal of organic chemistry 20120316 |
Total synthesis of (-)-kaitocephalin based on a Rh-catalyzed C-H amination. | Organic letters 20120316 |
Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana. | Bioorganic & medicinal chemistry 20120215 |
Mechanistic studies of substrate-assisted inhibition of ubiquitin-activating enzyme by adenosine sulfamate analogues. | The Journal of biological chemistry 20111125 |
Promiscuity of carbonic anhydrase II. Unexpected ester hydrolysis of carbohydrate-based sulfamate inhibitors. | Journal of the American Chemical Society 20111116 |
Detection of the 1H and 15N NMR resonances of sulfamate groups in aqueous solution: a new tool for heparin and heparan sulfate characterization. | Analytical chemistry 20111015 |
Aziridines from intramolecular alkene aziridination of sulfamates: reactivity toward carbon nucleophiles. application to the synthesis of spisulosine and its fluoro analogue. | The Journal of organic chemistry 20110916 |
Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates. | Bioorganic & medicinal chemistry 20110815 |
Aromatase and dual aromatase-steroid sulfatase inhibitors from the letrozole and vorozole templates. | ChemMedChem 20110801 |
Structure-activity relationships of C-17-substituted estratriene-3-O-sulfamates as anticancer agents. | Journal of medicinal chemistry 20110714 |
Development of steroid sulfatase inhibitors. | Molecular and cellular endocrinology 20110704 |
Rapid nickel-catalyzed Suzuki-Miyaura cross-couplings of aryl carbamates and sulfamates utilizing microwave heating. | The Journal of organic chemistry 20110304 |
Nickel-catalyzed amination of aryl sulfamates. | Angewandte Chemie (International ed. in English) 20110225 |
A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth. | Bioorganic & medicinal chemistry 20110201 |
Mechanisms of hydrolysis of phenyl- and benzyl 4-nitrophenyl-sulfamate esters. | Organic & biomolecular chemistry 20110121 |
Characterization and anions inhibition studies of an α-carbonic anhydrase from the teleost fish Dicentrarchus labrax. | Bioorganic & medicinal chemistry 20110115 |
Design and synthesis of cyclic sulfonamides and sulfamates as new calcium sensing receptor agonists. | Bioorganic & medicinal chemistry letters 20101215 |
Sulfamic acid catalyzed solvent-free synthesis of 10-aryl-7,7-dimethyl-6,7,8,10-tetrahydro-9H-[1,3]-dioxolo [4,5- b]xanthen-9-ones and 12-aryl-9,9-dimethyl-8,9,10,12-tetrahydro-11H-benzo[a]xanthen-11-ones. | Molecular diversity 20101101 |
The effect of aminosulfonate buffers on the light responses and intracellular pH of goldfish retinal horizontal cells. | Journal of neurochemistry 20101001 |
Bicyclic derivatives of the potent dual aromatase-steroid sulfatase inhibitor 2-bromo-4-{[(4-cyanophenyl)(4h-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: synthesis, SAR, crystal structure, and in vitro and in vivo activities. | ChemMedChem 20100903 |
Inhibition of the R1 fragment of the cadmium-containing zeta-class carbonic anhydrase from the diatom Thalassiosira weissflogii with anions. | Bioorganic & medicinal chemistry letters 20100815 |
Affinity of sulfamates and sulfamides to carbonic anhydrase II isoform: experimental and molecular modeling approaches. | Journal of chemical information and modeling 20100628 |
Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. | Bioorganic & medicinal chemistry letters 20100615 |
Brucella carbonic anhydrases: new targets for designing anti-infective agents. | Current pharmaceutical design 20100101 |
Suzuki-Miyaura coupling of aryl carbamates, carbonates, and sulfamates. | Journal of the American Chemical Society 20091216 |
Design and synthesis of carbon-11-labeled dual aromatase-steroid sulfatase inhibitors as new potential PET agents for imaging of aromatase and steroid sulfatase expression in breast cancer. | Steroids 20091101 |
Carbonic anhydrase inhibitors. Comparison of aliphatic sulfamate/bis-sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors. | Journal of medicinal chemistry 20091008 |
Carbonic anhydrase inhibitors; fluorinated phenyl sulfamates show strong inhibitory activity and selectivity for the inhibition of the tumor-associated isozymes IX and XII over the cytosolic ones I and II. | Bioorganic & medicinal chemistry letters 20090901 |
Which carbonic anhydrases are targeted by the antiepileptic sulfonamides and sulfamates? | Chemical biology & drug design 20090901 |
One-pot three-component Mannich-type reactions using sulfamic acid catalyst under ultrasound irradiation. | Ultrasonics sonochemistry 20090801 |
Identification of new 2-amino-3-methylimidazo[4,5-f]quinoline urinary metabolites from beta-naphthoflavone-treated mice. | Drug metabolism and disposition: the biological fate of chemicals 20090801 |
Development of structure-taste relationships for thiazolyl-, benzothiazolyl-, and thiadiazolylsulfamates. | Journal of agricultural and food chemistry 20090624 |
Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis. | Journal of medicinal chemistry 20090514 |
Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate. | Journal of medicinal chemistry 20090423 |
Copper(II) sulfamate: an efficient catalyst for the one-pot synthesis of 3,4-dihydropyrimidine-2(1H)-ones and thiones. | Molecules (Basel, Switzerland) 20090213 |
Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates. | Bioorganic & medicinal chemistry 20090201 |
Structure and inhibition of the CO2-sensing carbonic anhydrase Can2 from the pathogenic fungus Cryptococcus neoformans. | Journal of molecular biology 20090130 |
N,N-Dichloroaminosulfonic acids as novel topical antimicrobial agents. | Bioorganic & medicinal chemistry letters 20090101 |
A stereoselective synthesis of the bromopyrrole natural product (-)-agelastatin A. | Angewandte Chemie (International ed. in English) 20090101 |
Synthesis of aryl sulfamate and phenol small peptide derivatives using a multidetachable sulfamate linker strategy. | Advances in experimental medicine and biology 20090101 |
Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: synthesis, in vitro evaluation and computational modelling. | Organic & biomolecular chemistry 20081121 |
Mouse Ae1 E699Q mediates SO42-i/anion-o exchange with [SO42-]i-dependent reversal of wild-type pHo sensitivity. | American journal of physiology. Cell physiology 20080801 |
A chiral rhodium carboxamidate catalyst for enantioselective C-H amination. | Journal of the American Chemical Society 20080723 |
Poly(amidosulfonic acid) modified glassy carbon electrode for determination of isoniazid in pharmaceuticals. | Bioelectrochemistry (Amsterdam, Netherlands) 20080601 |
Enantioselective silica-based monoliths modified with a novel aminosulfonic acid-derived strong cation exchanger for electrically driven and pressure-driven capillary chromatography. | Electrophoresis 20080401 |
Carboxylic acid bioisosteres acylsulfonamides, acylsulfamides, and sulfonylureas as novel antagonists of the CXCR2 receptor. | Bioorganic & medicinal chemistry letters 20080315 |
Direct evidence for ArO-S bond cleavage upon inactivation of Pseudomonas aeruginosa arylsulfatase by aryl sulfamates. | Chembiochem : a European journal of chemical biology 20080303 |
Catalytic enantioselective addition of organometallic reagents to N-formylimines using monodentate phosphoramidite ligands. | The Journal of organic chemistry 20080201 |
Anticonvulsant sulfonamides/sulfamates/sulfamides with carbonic anhydrase inhibitory activity: drug design and mechanism of action. | Current pharmaceutical design 20080101 |
Three-component one-pot synthesis of 4,6-diarylpyrimidin- 2(1H)-ones under solvent-free conditions in the presence of sulfamic acid as a green and reusable catalyst. | Molecular diversity 20080101 |
Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides. | Bioorganic & medicinal chemistry 20071201 |
Aminosulfonate modulated pH-induced conformational changes in connexin26 hemichannels. | The Journal of biological chemistry 20070323 |
Stereospecific construction of substituted piperidines. Synthesis of (-)-paroxetine and (+)-laccarin. | Chemical communications (Cambridge, England) 20070221 |
Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors. | Journal of medicinal chemistry 20070125 |
Antitubercular nucleosides that inhibit siderophore biosynthesis: SAR of the glycosyl domain. | Journal of medicinal chemistry 20061228 |
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity. | Journal of medicinal chemistry 20061228 |
Synthesis and evaluation of general mechanism-based inhibitors of sulfatases based on (difluoro)methyl phenyl sulfate and cyclic phenyl sulfamate motifs. | Bioorganic & medicinal chemistry 20061215 |
Inhibitory effects of sulfamic acid on three thiosulfate-oxidizing chemolithotrophs. | FEMS microbiology letters 20061101 |
New zinc binding motifs in the design of selective carbonic anhydrase inhibitors. | Mini reviews in medicinal chemistry 20060801 |
Examination of two independent kinetic assays for determining the inhibition of carbonic anhydrases I and II: structure-activity comparison of sulfamates and sulfamides. | Chemical biology & drug design 20060801 |
Reactivity of cyclic sulfamidates towards sulfur-stabilised enolates. Stereocontrolled synthesis of functionalised lactams. | Organic & biomolecular chemistry 20060521 |
Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs. | Journal of medicinal chemistry 20060323 |
1,2,3,4-Tetrahydroisoquinolinyl sulfamic acids as phosphatase PTP1B inhibitors. | Bioorganic & medicinal chemistry letters 20060315 |
Synthesis and biological properties of new phosmidosine analogs having an N-acylsulfamate linkage. | Nucleosides, nucleotides & nucleic acids 20060101 |
Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors. | Journal of medicinal chemistry 20051201 |
Inhibition of MDA-MB-231 cell cycle progression and cell proliferation by C-2-substituted oestradiol mono- and bis-3-O-sulphamates. | International journal of cancer 20051020 |
Exploring new uses for C-H amination: Ni-catalyzed cross-coupling of cyclic sulfamates. | Organic letters 20051013 |
Cyclic sulfamide gamma-secretase inhibitors. | Bioorganic & medicinal chemistry letters 20051001 |
Synthesis of an N-acyl sulfamate analog of luciferyl-AMP: a stable and potent inhibitor of firefly luciferase. | Bioorganic & medicinal chemistry letters 20050901 |
A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents. | Journal of medicinal chemistry 20050811 |
Inhibition of laccase activity from Trametes versicolor by heavy metals and organic compounds. | Chemosphere 20050801 |
Carbonic anhydrase inhibitors. Synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with boron-containing sulfonamides, sulfamides, and sulfamates: toward agents for boron neutron capture therapy of hypoxic tumors. | Bioorganic & medicinal chemistry letters 20050701 |
Comparison of sulfamate and sulfamide groups for the inhibition of carbonic anhydrase-II by using topiramate as a structural platform. | Journal of medicinal chemistry 20050324 |
Sulfamates and their therapeutic potential. | Medicinal research reviews 20050301 |
Catabolism of sulfamate by Mycobacterium sp. CF1. | Environmental microbiology 20050301 |
Tethered aminohydroxylation using acyclic homo-allylic sulfamate esters and sulfonamides as substrates. | Organic & biomolecular chemistry 20050221 |
Identification of nonpeptidic small-molecule inhibitors of interleukin-2. | Bioorganic & medicinal chemistry letters 20050215 |
Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides. | Bioorganic & medicinal chemistry letters 20050215 |
Cyclic sulfamide HIV-1 protease inhibitors, with sidechains spanning from P2/P2' to P1/P1'. | Bioorganic & medicinal chemistry 20050201 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with bis-sulfamates. | Bioorganic & medicinal chemistry letters 20050201 |
The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates. | Biochemical and biophysical research communications 20040910 |
Carbonic anhydrase inhibitors: aliphatic N-phosphorylated sulfamates--a novel zinc-anchoring group leading to nanomolar inhibitors. | Journal of enzyme inhibition and medicinal chemistry 20040601 |
Sulfamide derivatives as transition state analogue inhibitors for carboxypeptidase A. | Bioorganic & medicinal chemistry 20040501 |
Inhibition of in vitro angiogenesis by 2-methoxy- and 2-ethyl-estrogen sulfamates. | International journal of cancer 20040420 |
2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells. | The Journal of steroid biochemistry and molecular biology 20040401 |
Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acid. | Bioorganic & medicinal chemistry letters 20040209 |
Carbonic anhydrase inhibitors: inhibition of transmembrane, tumor-associated isozyme IX, and cytosolic isozymes I and II with aliphatic sulfamates. | Journal of medicinal chemistry 20031204 |
Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates. | The Journal of steroid biochemistry and molecular biology 20031101 |
Measurement of physiological S-nitrosothiols: a problem child and a challenge. | Nitric oxide : biology and chemistry 20030801 |
The effects of 2-methoxy oestrogens and their sulphamoylated derivatives in conjunction with TNF-alpha on endothelial and fibroblast cell growth, morphology and apoptosis. | The Journal of steroid biochemistry and molecular biology 20030801 |
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors. | Journal of medicinal chemistry 20030522 |
Is the negative charge on RNHSO3-M+ an essential requirement for sulfamate sweetness? | Journal of agricultural and food chemistry 20030507 |
Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV. | Bioorganic & medicinal chemistry letters 20030310 |
Structure-activity relationship determination within a group of substituted phenyl sulfamate based compounds against the enzyme oestrone sulfatase. | The Journal of pharmacy and pharmacology 20030201 |
Growth inhibition of multi-drug-resistant breast cancer cells by 2-methoxyoestradiol-bis-sulphamate and 2-ethyloestradiol-bis-sulphamate. | The Journal of steroid biochemistry and molecular biology 20030201 |
3Beta-sulfamate derivatives of C19 and C21 steroids bearing a t-butylbenzyl or a benzyl group: synthesis and evaluation as non-estrogenic and non-androgenic steroid sulfatase inhibitors. | Journal of enzyme inhibition and medicinal chemistry 20030201 |
Solid-phase parallel synthesis of 17alpha-substituted estradiol sulfamate and phenol libraries using the multidetachable sulfamate linker. | Journal of combinatorial chemistry 20030101 |
Sulfamoyloxy-substituted 2-phenylindoles: antiestrogen-based inhibitors of the steroid sulfatase in human breast cancer cells. | Bioorganic & medicinal chemistry 20021201 |
A multidetachable sulfamate linker successfully used in a solid-phase strategy to generate libraries of sulfamate and phenol derivatives. | Bioorganic & medicinal chemistry letters 20021021 |
Application of the U and gamma' models in binary sweet taste mixtures. | Chemical senses 20020701 |
The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds. | Bioorganic & medicinal chemistry letters 20020506 |
Evidence for the mechanism of the irreversible inhibition of oestrone sulphatase (ES) by aminosulphonate based compounds. | The Journal of steroid biochemistry and molecular biology 20020401 |
Nonsteroidal compounds designed to mimic potent steroid sulfatase inhibitors. | The Journal of steroid biochemistry and molecular biology 20020301 |
Crystal structure of human carbonic anhydrase II complexed with an anti-convulsant sugar sulphamate. | The Biochemical journal 20020201 |
Carbonic anhydrase activity modulators: synthesis of inhibitors and activators incorporating 2-substituted-thiazol-4-yl-methyl scaffolds. | Journal of enzyme inhibition 20011001 |
Change in rate-determining step in an E1cB mechanism during aminolysis of sulfamate esters in acetonitrile. | The Journal of organic chemistry 20010921 |
Antitumour benzothiazoles. Part 15: The synthesis and physico-chemical properties of 2-(4-aminophenyl)benzothiazole sulfamate salt derivatives. | Bioorganic & medicinal chemistry letters 20010423 |
Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES). | Bioorganic & medicinal chemistry letters 20010409 |
Novel inhibitors of the enzyme estrone sulfatase (ES). | Bioorganic & medicinal chemistry letters 20010326 |
Sulfonylated aminothiazoles as new small molecule inhibitors of protein phosphatases. | Bioorganic & medicinal chemistry letters 20010212 |
Non-steroidal and steroidal sulfamates: new drugs for cancer therapy. | Molecular and cellular endocrinology 20010122 |
Alternative splicing of a Drosophila GABA receptor subunit gene identifies determinants of agonist potency. | Neuroscience 20010101 |
Nonpeptidic HIV protease inhibitors: 6-alkyl-5,6-dihydropyran-2-ones possessing a novel and achiral 3-(2-t-butyl-5-methyl-4-sulfamate)phenylthio moiety. | Bioorganic & medicinal chemistry letters 19990802 |
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