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Home > Imidazoles > 59939-16-1
CAS No: 59939-16-1 Catalog No: AG00E9LS MDL No:
Title | Journal |
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The effects of the co-administration of the α₁-adrenoreceptor antagonist prazosin on the anxiolytic effect of citalopram in conditioned fear stress in the rat. | Progress in neuro-psychopharmacology & biological psychiatry 20121001 |
The contribution of d-tubocurarine-sensitive and apamin-sensitive K-channels to EDHF-mediated relaxation of mesenteric arteries from eNOS-/- mice. | Journal of cardiovascular pharmacology 20120501 |
Mutual independence of 5-HT(2) and α1 noradrenergic receptors in mediating deficits in sensorimotor gating. | Psychopharmacology 20120401 |
α- and β-Adrenergic receptors differentially modulate the emission of spontaneous and amphetamine-induced 50-kHz ultrasonic vocalizations in adult rats. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20120201 |
Clonidine improved laboratory-measured decision-making performance in abstinent heroin addicts. | PloS one 20120101 |
Reducing the harm of stress: medications to rescue the prefrontal cortex and overcome bad habits: the science of stress: focus on the brain, breaking bad habits, and chronic disease. | The Yale journal of biology and medicine 20111201 |
Corticotropin-releasing factor and noradrenergic signalling exert reciprocal control over startle reactivity. | The international journal of neuropsychopharmacology 20111001 |
Long-term α1A-adrenergic receptor stimulation improves synaptic plasticity, cognitive function, mood, and longevity. | Molecular pharmacology 20111001 |
Quantification of functional selectivity at the human α(1A)-adrenoceptor. | Molecular pharmacology 20110201 |
[Alteration of brown adipocyte Ca2+ responses in culture by adrenergic activation]. | Tsitologiia 20110101 |
Protection of protease-activated receptor 2 mediated vasodilatation against angiotensin II-induced vascular dysfunction in mice. | BMC pharmacology 20110101 |
The involvement of noradrenaline in rapid eye movement sleep mentation. | Frontiers in neurology 20110101 |
Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis. | Bioorganic & medicinal chemistry letters 20101101 |
Modulation of N-type calcium currents by presynaptic imidazoline receptor activation in rat superior cervical ganglion neurons. | Experimental physiology 20101001 |
Attenuation of store-operated Ca2+ entry and enhanced expression of TRPC channels in caudal artery smooth muscle from Type 2 diabetic Goto-Kakizaki rats. | Clinical and experimental pharmacology & physiology 20100701 |
Alpha1-adrenoceptors modulate citalopram-induced serotonin release. | Neuropharmacology 20100601 |
Impairment of α1-adrenoceptor-mediated contractile activity in caudal arterial smooth muscle from type 2 diabetic Goto-Kakizaki rats. | Clinical and experimental pharmacology & physiology 20100301 |
The selective alpha1 adrenoceptor antagonist HEAT reduces L-DOPA-induced dyskinesia in a rat model of Parkinson's disease. | Synapse (New York, N.Y.) 20100201 |
Might adrenergic alpha2C-agonists/alpha2A-antagonists become novel therapeutic tools for pain treatment with morphine? | Journal of medicinal chemistry 20091126 |
Acute dilation to alpha(2)-adrenoceptor antagonists uncovers dual constriction and dilation mediated by arterial alpha(2)-adrenoceptors. | British journal of pharmacology 20091101 |
Human and mouse trace amine-associated receptor 1 have distinct pharmacology towards endogenous monoamines and imidazoline receptor ligands. | The Biochemical journal 20091023 |
alpha(1A)- and alpha(1B)-adrenergic receptors differentially modulate antidepressant-like behavior in the mouse. | Brain research 20090818 |
alpha1-Adrenergic receptors regulate neurogenesis and gliogenesis. | Molecular pharmacology 20090801 |
Dual regulation of heat-activated K+ channel in rat DRG neurons via alpha(1) and beta adrenergic receptors. | Life sciences 20090717 |
Catecholaminergic automatic activity in the rat pulmonary vein: electrophysiological differences between cardiac muscle in the left atrium and pulmonary vein. | American journal of physiology. Heart and circulatory physiology 20090701 |
Effects of a Western diet versus high glucose on endothelium-dependent relaxation in murine micro- and macro-vasculature. | European journal of pharmacology 20081228 |
Evidence that some imidazoline derivatives inhibit peripherally the vasopressor sympathetic outflow in pithed rats. | Autonomic neuroscience : basic & clinical 20081205 |
Enhanced alpha1 adrenergic sensitivity in sensorimotor gating deficits in neonatal ventral hippocampus-lesioned rats. | The international journal of neuropsychopharmacology 20081201 |
Signal transduction and gene expression in cultured accessory olfactory bulb neurons. | Neuroscience 20081119 |
The adrenergic receptor subtypes present in frog (Rana esculenta) skin. | Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20080801 |
QSAR study of imidazoline antihypertensive drugs. | Bioorganic & medicinal chemistry 20080801 |
Different response of ANP secretion to adrenoceptor stimulation in renal hypertensive rat atria. | Peptides 20080701 |
The effects of Cirazoline, an alpha-1 adrenoreceptor agonist, on the firing rates of thermally classified anterior hypothalamic neurons in rat brain slices. | Brain research 20080208 |
Antihypertensive drug guanabenz is active in vivo against both yeast and mammalian prions. | PloS one 20080101 |
Alpha 1-adrenoceptor agonists protect against stress-induced death of neural progenitor cells. | European journal of pharmacology 20071114 |
Mechanisms of modafinil: A review of current research. | Neuropsychiatric disease and treatment 20070601 |
Presynaptic alpha-adrenoceptors in median preoptic nucleus modulate inhibitory neurotransmission from subfornical organ and organum vasculosum lamina terminalis. | American journal of physiology. Regulatory, integrative and comparative physiology 20070501 |
Medial prefrontal cortical alpha1 adrenoreceptor modulation of the nucleus accumbens dopamine response to stress in Long-Evans rats. | Psychopharmacology 20070401 |
Beta(2)-Adrenergic activation increases glycogen synthesis in L6 skeletal muscle cells through a signalling pathway independent of cyclic AMP. | Diabetologia 20070101 |
Increased Rho activation and PKC-mediated smooth muscle contractility in the absence of caveolin-1. | American journal of physiology. Cell physiology 20061201 |
Disruption of prepulse inhibition after stimulation of central but not peripheral alpha-1 adrenergic receptors. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20061001 |
Iloperidone reduces sensorimotor gating deficits in pharmacological models, but not a developmental model, of disrupted prepulse inhibition in rats. | Neuropharmacology 20060901 |
Discriminative stimulus properties of the selective and highly potent alpha2-adrenoceptor agonist, S18616, in rats: mediation by the alpha2A subtype, and blockade by the atypical antidepressants, mirtazapine and mianserin. | Neuropharmacology 20060901 |
Separable noradrenergic and dopaminergic regulation of prepulse inhibition in rats: implications for predictive validity and Tourette Syndrome. | Psychopharmacology 20060601 |
Presynaptic alpha1 adrenergic receptors differentially regulate synaptic glutamate and GABA release to hypothalamic presympathetic neurons. | The Journal of pharmacology and experimental therapeutics 20060201 |
Pharmacological characterization of alpha1- and beta-adrenergic synergism of 5'DII activity in rat brown adipocytes. | Archives of physiology and biochemistry 20060201 |
Imidazoline receptors in relaxation of acetylcholine-constricted isolated rat jejunum. | Pharmacological reports : PR 20060101 |
Augmentation of alpha1-adrenoceptor-mediated contraction by warming without increased phosphorylation of myosin in rat caudal arterial smooth muscle. | Journal of pharmacological sciences 20050901 |
Yohimbine disrupts prepulse inhibition in rats via action at 5-HT1A receptors, not alpha2-adrenoceptors. | Psychopharmacology 20050701 |
Effects of chloride substitution in isolated mesenteric blood vessels from Dahl normotensive and hypertensive rats. | Journal of cardiovascular pharmacology 20050701 |
Impact of nitric oxide synthase inhibitor and chloride channel antagonist on mesenteric vascular conductance in anesthetized Dahl normotensive and hypertensive rats. | Journal of cardiovascular pharmacology 20050601 |
Impaired alpha1-adrenergic responses in aged rat hearts. | Fundamental & clinical pharmacology 20050601 |
Addition of a signal peptide sequence to the alpha1D-adrenoceptor gene increases the density of receptors, as determined by [3H]-prazosin binding in the membranes. | British journal of pharmacology 20050301 |
alpha1A-adrenoceptors activate glucose uptake in L6 muscle cells through a phospholipase C-, phosphatidylinositol-3 kinase-, and atypical protein kinase C-dependent pathway. | Endocrinology 20050201 |
Protein kinase C overactivity impairs prefrontal cortical regulation of working memory. | Science (New York, N.Y.) 20041029 |
Allosteric modulation of semicarbazide-sensitive amine oxidase activities in vitro by imidazoline receptor ligands. | British journal of pharmacology 20041001 |
Neurotensin agonists block the prepulse inhibition deficits produced by a 5-HT2A and an alpha1 agonist. | Psychopharmacology 20040901 |
Noradrenergic inputs mediate state dependence of auditory responses in the avian song system. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20040901 |
Cold adaptation modulates Ca2+ signaling in brown preadipocytes. | Bulletin of experimental biology and medicine 20040701 |
Preoptic alpha 1- and alpha 2-noradrenergic agonists induce, respectively, PGE2-independent and PGE2-dependent hyperthermic responses in guinea pigs. | American journal of physiology. Regulatory, integrative and comparative physiology 20040601 |
Effects of chloride substitution on electromechanical responses in the pulmonary artery of Dahl normotensive and hypertensive rats. | British journal of pharmacology 20040301 |
Noradrenaline inhibits autonomous activity in the isolated guinea pig bladder. | BJU international 20040201 |
Identification and pharmacological characterization of a specific agmatine transport system in human tumor cell lines. | Annals of the New York Academy of Sciences 20031201 |
Atypical [(3)H]clonidine binding sites in human caudate and platelets on cryostat-cut sections. | Annals of the New York Academy of Sciences 20031201 |
Tempol, an antioxidant, restores endothelium-derived hyperpolarizing factor-mediated vasodilation during hypertension. | European journal of pharmacology 20031114 |
Stimulation of alpha1-adrenoceptors in the rat medial prefrontal cortex increases the local in vivo 5-hydroxytryptamine release: reversal by antipsychotic drugs. | Journal of neurochemistry 20031101 |
Regulation of the release of serotonin in the dorsal raphe nucleus by alpha1 and alpha2 adrenoceptors. | Synapse (New York, N.Y.) 20031001 |
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives. | Journal of medicinal chemistry 20030508 |
Alpha 1-adrenoceptor-activated cation currents in neurones acutely isolated from rat cardiac parasympathetic ganglia. | The Journal of physiology 20030401 |
Identification and characterization of the imidazoline I2b-binding sites in the hamster brown adipose tissue as a study model for imidazoline receptors. | Archives of physiology and biochemistry 20030401 |
A photosensitive vascular smooth muscle store of nitric oxide in mouse aorta: no dependence on expression of endothelial nitric oxide synthase. | British journal of pharmacology 20030301 |
Contractile actions of imidazoline alpha-adrenoceptor agonists and effects of noncompetitive alpha1-adrenoceptor antagonists in human vas deferens. | European journal of pharmacology 20030221 |
Opposite effects of alpha 1- and beta-adrenoceptor stimulation on both glutamate- and gamma-aminobutyric acid-mediated spontaneous transmission in cultured rat hippocampal neurons. | Journal of neuroscience research 20030215 |
Alpha(1)-adrenoceptor activation: a comparison of 4-(anilinomethyl)imidazoles and 4-(phenoxymethyl)imidazoles to related 2-imidazolines. | Bioorganic & medicinal chemistry letters 20021202 |
Cholesterol depletion disrupts caveolae and differentially impairs agonist-induced arterial contraction. | Arteriosclerosis, thrombosis, and vascular biology 20020801 |
A comparative study of the effects of Cl(-) channel blockers on mesenteric vascular conductance in anaesthetized rat. | European journal of pharmacology 20020712 |
A novel pathway for adrenergic stimulation of cAMP-response-element-binding protein (CREB) phosphorylation: mediation via alpha1-adrenoceptors and protein kinase C activation. | The Biochemical journal 20020515 |
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
Effect of nitric oxide synthase inhibitor N(omega) nitro-L-arginine methyl ester on relaxant responses to calcium channel antagonists in isolated aortic rings from Dahl normotensive and hypertensive rats. | Journal of cardiovascular pharmacology 20020301 |
2-(anilinomethyl)imidazolines as alpha1A adrenergic receptor agonists: 2'-heteroaryl and 2'-oxime ether series. | Bioorganic & medicinal chemistry letters 20020225 |
alpha(1)-Adrenoceptor agonists: the identification of novel alpha(1A )subtype selective 2'-heteroaryl-2-(phenoxymethyl)imidazolines. | Bioorganic & medicinal chemistry letters 20020211 |
Noradrenaline release-inhibiting receptors on PC12 cells devoid of alpha(2(-)) and CB(1) receptors: similarities to presynaptic imidazoline and edg receptors. | Neurochemistry international 20020201 |
Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole. | Journal of medicinal chemistry 20020103 |
[Excitatory effect of noradrenaline on rat airway parasympathetic ganglion neurons]. | Fukuoka igaku zasshi = Hukuoka acta medica 20011101 |
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists. | The Journal of biological chemistry 20010706 |
The release of noradrenaline in the locus coeruleus and prefrontal cortex studied with dual-probe microdialysis. | Brain research 20010706 |
Agmatine and putrescine uptake in the human glioma cell line SK-MG-1. | Naunyn-Schmiedeberg's archives of pharmacology 20010601 |
Use of trifluoroperazine isolates a [(3)H]Ifenprodil binding site in rat brain membranes with the pharmacology of the voltage-independent ifenprodil site on N-methyl-D-aspartate receptors containing NR2B subunits. | The Journal of pharmacology and experimental therapeutics 20010101 |
Adrenergic stimulation of lipoprotein lipase gene expression in rat brown adipocytes differentiated in culture: mediation via beta3- and alpha1-adrenergic receptors. | The Biochemical journal 19970201 |
Selectivity of the imidazoline alpha-adrenoceptor agonists (oxymetazoline and cirazoline) for human cloned alpha 1-adrenoceptor subtypes. | British journal of pharmacology 19950901 |
Selectivity of agonists for cloned alpha 1-adrenergic receptor subtypes. | Molecular pharmacology 19941101 |
Single and repeated doses of the vasodilator/beta-adrenergic antagonist, carvedilol, block cirazoline- and isoproterenol-mediated hemodynamic responses in the conscious rat. | Cardiovascular drugs and therapy 19921001 |
Orthostatic hypotension occurs following alpha 2-adrenoceptor blockade in chronic prazosin-pretreated conscious spontaneously hypertensive rats. | Journal of autonomic pharmacology 19920801 |
Effects on ingestive behavior in rats of the alpha 1-adrenoceptor agonist cirazoline. | European journal of pharmacology 19920107 |
Effects of staurosporine on the pressor responses to alpha-adrenoceptor agonists in pithed rats: a comparison with nifedipine. | Pharmacology 19910101 |
Receptor interactions of imidazolines. IX. Cirazoline is an alpha-1 adrenergic agonist and an alpha-2 adrenergic antagonist. | The Journal of pharmacology and experimental therapeutics 19820701 |
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