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Home > Indoles and Oxindole > 496-15-1
496-15-1 | Indoline
CAS No: 496-15-1 Catalog No: AG00I8V1 MDL No:MFCD00005705
Product Description
Catalog Number:
AG00I8V1
Chemical Name:
Indoline
CAS Number:
496-15-1
MDL Number:
MFCD00005705
IUPAC Name:
2,3-dihydro-1H-indole
InChI:
InChI=1S/C8H9N/c1-2-4-8-7(3-1)5-6-9-8/h1-4,9H,5-6H2
InChI Key:
LPAGFVYQRIESJQ-UHFFFAOYSA-N
EC Number:
207-816-8
UNII:
6DPT9AB2NK
Properties
Complexity:
101
Compound Is Canonicalized:
Yes
Covalently-Bonded Unit Count:
1
Defined Atom Stereocenter Count:
0
Defined Bond Stereocenter Count:
0
Exact Mass:
119.073g/mol
Formal Charge:
0
Heavy Atom Count:
9
Hydrogen Bond Acceptor Count:
1
Hydrogen Bond Donor Count:
1
Isotope Atom Count:
0
Molecular Weight:
119.167g/mol
Monoisotopic Mass:
119.073g/mol
Rotatable Bond Count:
0
Topological Polar Surface Area:
12A^2
Undefined Atom Stereocenter Count:
0
Undefined Bond Stereocenter Count:
0
XLogP3:
1.9
Literature
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| 2-[(2,3-dihydro-1H-indol-1-yl)methyl]melatonin analogues: a novel class of MT2-selective melatonin receptor antagonists. | Journal of medicinal chemistry 20090212 |
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| Novel indoline-based acyl-CoA:cholesterol acyltransferase inhibitor with antiperoxidative activity: improvement of physicochemical properties and biological activities by introduction of carboxylic acid. | Journal of medicinal chemistry 20080814 |
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| CYP2D6-Mediated metabolism of a novel acyl coenzyme A:cholesterol acyltransferase inhibitor, pactimibe, and its unique plasma metabolite, R-125528. | Drug metabolism and disposition: the biological fate of chemicals 20080301 |
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| Synthesis and properties of novel porphyrin spin probes containing isoindoline nitroxides. | Free radical biology & medicine 20070701 |
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| Studies in sigmatropic rearrangements of N-prenylindole derivatives--a formal enantiomerically pure synthesis of tryprostatin B. | Organic & biomolecular chemistry 20061107 |
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| A metal-free approach to the synthesis of indoline derivatives by a phenyliodine(III) bis(trifluoroacetate)-mediated amidohydroxylation reaction. | The Journal of organic chemistry 20061013 |
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| Efficient synthesis of achiral seco-cyclopropylbenz[2,3-e]indoline analogues: [4-amino-2-(5,6,7-trimethoxyindole-2-carboxamido)naphthalen-1-yl]ethyl chloride and [4-hydroxy-2-(5,6,7-trimethoxyindole-2-carboxamido)naphthalen-1-yl]ethyl chloride. | The Journal of organic chemistry 20060609 |
| Preparation of 7-Halo-indoles by Thallation of N-formylindoline and their attempted use for synthesis of the right-hand segment of chloropeptin. | Chemical & pharmaceutical bulletin 20060601 |
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| The design and enzyme-bound crystal structure of indoline based peptidomimetic inhibitors of hepatitis C virus NS3 protease. | Journal of medicinal chemistry 20041216 |
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| Indoline derivatives as 5-HT(2C) receptor agonists. | Bioorganic & medicinal chemistry letters 20040503 |
| Synthesis and evaluation of some new spiro indoline-based heterocycles as potentially active antimicrobial agents. | Bioorganic & medicinal chemistry 20040501 |
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| Novel non-peptidic neuropeptide Y Y2 receptor antagonists. | Bioorganic & medicinal chemistry letters 20040308 |
| Spirobipyridopyrans, spirobinaphthopyrans, indolinospiropyridopyrans, indolinospironaphthopyrans and indolinospironaphtho-1,4-oxazines: synthesis, study of X-ray crystal structure, antitumoral and antiviral evaluation. | Bioorganic & medicinal chemistry 20040301 |
| Unexpected syntheses of seco-cyclopropyltetrahydroquinolines - from a radical 5-exo-trig cyclization reaction: analogs of CC-1065 and the duocarmycins. | Molecules (Basel, Switzerland) 20040227 |
| Highly-efficient metal-free organic dyes for dye-sensitized solar cells. | Chemical communications (Cambridge, England) 20031221 |
| Aptamers switch on fluorescence of triphenylmethane dyes. | Journal of the American Chemical Society 20031203 |
| The effect of remote chirality on the antibacterial activity of indolinyl, tetrahydroquinolyl and dihydrobenzoxazinyl oxazolidinones. | Bioorganic & medicinal chemistry letters 20031201 |
| A convergent synthetic approach to the nucleoside-type liposidomycin antibiotics. | Organic letters 20031016 |
| Stereospecific construction of contiguous quaternary and tertiary stereocenters by rearrangement from indoline-2-methanol to 2,2,3-trisubstituted tetrahydroquinoline: application to an efficient total synthesis of natural virantmycin. | Angewandte Chemie (International ed. in English) 20030606 |
| Total synthesis of the duocarmycins. | Journal of the American Chemical Society 20030604 |
| Preparation and pharmacological profile of 7-(alpha-azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitors. | Bioorganic & medicinal chemistry letters 20030505 |
| Cardioselective anti-ischemic ATP-sensitive potassium channel (KATP) openers: benzopyranyl indoline and indole analogues. | European journal of medicinal chemistry 20030501 |
| Synthesis of 6H-pyrrolo[3',4':2,3][1,4]diazepino[6,7,1-hi]indole-8,10(7H,9H)-diones using 3-bromo-4-(indol-1-yl)maleimide scaffold. | Organic & biomolecular chemistry 20030307 |
| Sulfur ylide-initiated thio-claisen rearrangements. The synthesis of highly substituted indolines. | The Journal of organic chemistry 20030207 |
| Novel strategies for the solid phase synthesis of substituted indolines and indoles. | Bioorganic & medicinal chemistry 20030206 |
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| Free radical-mediated aryl amination and its use in a convergent [3 + 2] strategy for enantioselective indoline alpha-amino acid synthesis. | Journal of the American Chemical Society 20030108 |
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| Indoline and piperazine containing derivatives as a novel class of mixed D(2)/D(4) receptor antagonists. Part 2: asymmetric synthesis and biological evaluation. | Bioorganic & medicinal chemistry letters 20021104 |
| Novel furano analogues of duocarmycin C1 and C2: design, synthesis, and biological evaluation of seco-iso-cyclopropylfurano[2,3-e]indoline (seco-iso-CFI) and seco-cyclopropyltetrahydrofurano[2,3-f]quinoline (seco-CFQ) analogues. | Bioorganic & medicinal chemistry 20020901 |
| A convergent approach to 3-substituted-5-methoxyindoles. Application to the synthesis of melatonin [correction]. | Chemical communications (Cambridge, England) 20020821 |
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| A new strychnobrasiline base of Strychnos mattogrossensis. | Natural product letters 20020801 |
| Nature of non-radiative processes involved in the excited state of 9-cyanoanthracene in presence of 2-methylindole/2-methylindoline quenchers. A laser flash photolysis study to reveal the medium effects. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20020601 |
| Antimicrobial activities of a new schizozygane indoline alkaloid from Schizozygia coffaeoides and the revised structure of isoschizogaline. | Journal of natural products 20020401 |
| Erythropoietin mimetics derived from solution phase combinatorial libraries. | Journal of the American Chemical Society 20020130 |
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| Design, synthesis, and biological activity of diiminoisoindolines as complement component 3a antagonists. | Bioorganic & medicinal chemistry letters 20011105 |
| Multiple mutations at the active site of naphthalene dioxygenase affect regioselectivity and enantioselectivity. | Journal of industrial microbiology & biotechnology 20010801 |
| The discovery of linezolid, the first oxazolidinone antibacterial agent. | Current drug targets. Infectious disorders 20010801 |
| Asymmetric synthesis of novel isoindolines: azasaccharide mimics as potential enzyme inhibitors. | The Journal of pharmacy and pharmacology 20010701 |
| Beta D305A mutant of tryptophan synthase shows strongly perturbed allosteric regulation and substrate specificity. | Biochemistry 20010626 |
| A new and general synthetic pathway to strychnos indole alkaloids: total syntheses of (-)-dehydrotubifoline and (-)-tubifoline by palladium-catalyzed asymmetric allylic substitution. | Organic letters 20010614 |
| A novel series of thromboxane A2 synthetase inhibitors with free radical scavenging and anti-peroxidative activities. | Chemical & pharmaceutical bulletin 20010501 |
| N-Aminoindoline derivatives as inhibitors of 5-lipoxygenase. | Bioorganic & medicinal chemistry letters 20010326 |
| 1-Nitroindoline. | Acta crystallographica. Section C, Crystal structure communications 20010301 |
| Human beta3 adrenergic receptor agonists containing cyanoguanidine and nitroethylenediamine moieties. | Bioorganic & medicinal chemistry letters 20010212 |
| Trapping of the putative cationic intermediate in the Morin rearrangement with carbon nucleophiles. | The Journal of organic chemistry 20010209 |
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