200,000+ products from a single source!
sales@angenechem.com
Home > Sulfanilamide > 452-35-7
CAS No: 452-35-7 Catalog No: AG00DEP4 MDL No:MFCD00057089
Title | Journal |
---|---|
Carbonic anhydrase inhibitors: synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety. | Bioorganic & medicinal chemistry 20131001 |
Single and mixed poloxamine micelles as nanocarriers for solubilization and sustained release of ethoxzolamide for topical glaucoma therapy. | Journal of the Royal Society, Interface 20120907 |
Methazolamide is a new hepatic insulin sensitizer that lowers blood glucose in vivo. | Diabetes 20120801 |
Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target. | Journal of medicinal chemistry 20120412 |
Mutation of active site residues Asn67 to Ile, Gln92 to Val and Leu204 to Ser in human carbonic anhydrase II: influences on the catalytic activity and affinity for inhibitors. | Bioorganic & medicinal chemistry 20120401 |
Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI. | European journal of medicinal chemistry 20120301 |
Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana. | Bioorganic & medicinal chemistry 20120215 |
Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives. | Bioorganic & medicinal chemistry letters 20120201 |
Dependence of avidity on linker length for a bivalent ligand-bivalent receptor model system. | Journal of the American Chemical Society 20120111 |
Topiramate and the vision: a systematic review. | Clinical ophthalmology (Auckland, N.Z.) 20120101 |
Differential scanning fluorometry signatures as indicators of enzyme inhibitor mode of action: case study of glutathione S-transferase. | PloS one 20120101 |
Thermodynamics of aryl-dihydroxyphenyl-thiadiazole binding to human Hsp90. | PloS one 20120101 |
Regulation of the cyanobacterial CO2-concentrating mechanism involves internal sensing of NADP+ and α-ketogutarate levels by transcription factor CcmR. | PloS one 20120101 |
Carbonic anhydrase activity in Arabidopsis thaliana thylakoid membrane and fragments enriched with PSI or PSII. | Photosynthesis research 20111201 |
Testing the limits of sensitivity in a solid-state structural investigation by combined X-ray powder diffraction, solid-state NMR, and molecular modelling. | Physical chemistry chemical physics : PCCP 20111028 |
Photosynthetic characteristics of a multicellular green alga Volvox carteri in response to external CO2 levels possibly regulated by CCM1/CIA5 ortholog. | Photosynthesis research 20110901 |
Evidence for the occurrence of photorespiration in synurophyte algae. | Photosynthesis research 20110901 |
Carbonic anhydrase inhibitors. Synthesis, molecular structures, and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with novel 3-pyridinesulfonamide derivatives. | European journal of medicinal chemistry 20110901 |
Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates. | Bioorganic & medicinal chemistry 20110815 |
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies. | Bioorganic & medicinal chemistry 20110515 |
Carbonate precipitates and bicarbonate secretion in the intestine of sea bass, Dicentrarchus labrax. | Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20110501 |
Extracellular β-class carbonic anhydrase of the alkaliphilic cyanobacterium Microcoleus chthonoplastes. | Journal of photochemistry and photobiology. B, Biology 20110404 |
Evaluation of the reproductive and developmental risks of caffeine. | Birth defects research. Part B, Developmental and reproductive toxicology 20110401 |
Purification and inhibition studies with anions and sulfonamides of an α-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii. | Bioorganic & medicinal chemistry 20110315 |
Bioinspired imprinted PHEMA-hydrogels for ocular delivery of carbonic anhydrase inhibitor drugs. | Biomacromolecules 20110314 |
(R)-/(S)-10-camphorsulfonyl-substituted aromatic/heterocyclic sulfonamides selectively inhibit mitochondrial over cytosolic carbonic anhydrases. | Bioorganic & medicinal chemistry letters 20110301 |
A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth. | Bioorganic & medicinal chemistry 20110201 |
Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. | Bioorganic & medicinal chemistry letters 20110115 |
A high throughput screen identifies chemical modulators of the laminin-induced clustering of dystroglycan and aquaporin-4 in primary astrocytes. | PloS one 20110101 |
Treat ankylosing spondylitis with methazolamide. | International journal of medical sciences 20110101 |
Bacterial carbonic anhydrases as drug targets: toward novel antibiotics? | Frontiers in pharmacology 20110101 |
Transport activity of the sodium bicarbonate cotransporter NBCe1 is enhanced by different isoforms of carbonic anhydrase. | PloS one 20110101 |
Sharpey-Schafer lecture: gas channels. | Experimental physiology 20101201 |
Carbonic anhydrase II regulates differentiation of ameloblasts via intracellular pH-dependent JNK signaling pathway. | Journal of cellular physiology 20101101 |
Carbonic anhydrase inhibitors. Regioselective synthesis of novel 1-substituted 1,4-dihydro-4-oxo-3-pyridinesulfonamides and their inhibition of the human cytosolic isozymes I and II and transmembrane cancer-associated isozymes IX and XII. | European journal of medicinal chemistry 20100901 |
Mutation of Phe91 to Asn in human carbonic anhydrase I unexpectedly enhanced both catalytic activity and affinity for sulfonamide inhibitors. | Bioorganic & medicinal chemistry 20100801 |
Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. | Bioorganic & medicinal chemistry letters 20100615 |
New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors. | Bioorganic & medicinal chemistry letters 20100615 |
Carbonic anhydrase inhibitors: synthesis and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with 4-substituted 3-pyridinesulfonamides. | European journal of medicinal chemistry 20100601 |
Carbonic anhydrase inhibitors. The beta-carbonic anhydrases from the fungal pathogens Cryptococcus neoformans and Candida albicans are strongly inhibited by substituted-phenyl-1H-indole-5-sulfonamides. | Bioorganic & medicinal chemistry letters 20100415 |
Nonenzymatic augmentation of lactate transport via monocarboxylate transporter isoform 4 by carbonic anhydrase II. | The Journal of membrane biology 20100401 |
Cloning, characterization, and inhibition studies of a beta-carbonic anhydrase from Brucella suis. | Journal of medicinal chemistry 20100311 |
Differences in transcription between free-living and CO2-activated third-stage larvae of Haemonchus contortus. | BMC genomics 20100101 |
Alterations in osteoclast function and phenotype induced by different inhibitors of bone resorption--implications for osteoclast quality. | BMC musculoskeletal disorders 20100101 |
Saccharomyces cerevisiae β-carbonic anhydrase: inhibition and activation studies. | Current pharmaceutical design 20100101 |
Role of carbonic anhydrase IV in the bicarbonate-mediated activation of murine and human sperm. | PloS one 20100101 |
Increased expression of carbonic anhydrase I in the synovium of patients with ankylosing spondylitis. | BMC musculoskeletal disorders 20100101 |
T tubules and surface membranes provide equally effective pathways of carbonic anhydrase-facilitated lactic acid transport in skeletal muscle. | PloS one 20100101 |
Cyclodextrins in delivery systems: Applications. | Journal of pharmacy & bioallied sciences 20100101 |
Ocular inserts - Advancement in therapy of eye diseases. | Journal of advanced pharmaceutical technology & research 20100101 |
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c. | Bioorganic & medicinal chemistry letters 20091201 |
A pea mutant (costata) expressing higher activity in thylakoid membrane-bound carbonic anhydrase alters PSII downregulation mechanisms. | Cell biology international 20090801 |
Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides. | Bioorganic & medicinal chemistry 20090715 |
Carbonic anhydrase inhibitors. Inhibition and homology modeling studies of the fungal beta-carbonic anhydrase from Candida albicans with sulfonamides. | Bioorganic & medicinal chemistry 20090701 |
Carbonic anhydrase inhibitors. Phenacetyl-, pyridylacetyl- and thienylacetyl-substituted aromatic sulfonamides act as potent and selective isoform VII inhibitors. | Bioorganic & medicinal chemistry letters 20090615 |
Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII. | Bioorganic & medicinal chemistry letters 20090601 |
Measurement of nanomolar dissociation constants by titration calorimetry and thermal shift assay - radicicol binding to Hsp90 and ethoxzolamide binding to CAII. | International journal of molecular sciences 20090601 |
Titration calorimetry standards and the precision of isothermal titration calorimetry data. | International journal of molecular sciences 20090601 |
Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis. | Journal of medicinal chemistry 20090514 |
Ligand-directed tosyl chemistry for protein labeling in vivo. | Nature chemical biology 20090501 |
Manganese-dependent carboanhydrase activity of photosystem II proteins. | Biochemistry. Biokhimiia 20090501 |
Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate. | Journal of medicinal chemistry 20090423 |
Carbonic anhydrase inhibitors. The nematode alpha-carbonic anhydrase of Caenorhabditis elegans CAH-4b is highly inhibited by 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides. | Bioorganic & medicinal chemistry 20090415 |
QSAR studies for the inhibition of the transmembrane carbonic anhydrase isozyme XIV with sulfonamides using PRECLAV software. | Journal of enzyme inhibition and medicinal chemistry 20090401 |
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases. | Bioorganic & medicinal chemistry letters 20090301 |
Design of a carbonic anhydrase IX active-site mimic to screen inhibitors for possible anticancer properties. | Biochemistry 20090217 |
Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the difference. | Bioorganic & medicinal chemistry 20090201 |
Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates. | Bioorganic & medicinal chemistry 20090201 |
Carbonic anhydrase inhibitors. Comparison of chlorthalidone and indapamide X-ray crystal structures in adducts with isozyme II: when three water molecules and the keto-enol tautomerism make the difference. | Journal of medicinal chemistry 20090122 |
Inhibition of aquaporin 4 by antiepileptic drugs. | Bioorganic & medicinal chemistry 20090101 |
Label-free determination of protein-ligand binding constants using mass spectrometry and validation using surface plasmon resonance and isothermal titration calorimetry. | Journal of molecular recognition : JMR 20090101 |
Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions. | Bioorganic & medicinal chemistry letters 20081215 |
The bicarbonate transporter is essential for Bacillus anthracis lethality. | PLoS pathogens 20081101 |
Lack of aquaporin-4 water transport inhibition by antiepileptics and arylsulfonamides. | Bioorganic & medicinal chemistry 20080801 |
Carbonic anhydrase inhibitors: design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes. | Bioorganic & medicinal chemistry letters 20080615 |
Isolation and characterization of a gene encoding carbonic anhydrase from Ostertagia ostertagi and quantitative measurement of expression during in vivo exsheathment. | Veterinary parasitology 20080614 |
Carbonic anhydrase inhibitors: bioreductive nitro-containing sulfonamides with selectivity for targeting the tumor associated isoforms IX and XII. | Journal of medicinal chemistry 20080612 |
Antagonistic effect of juvenile hormone on hemocyte-spreading behavior of Spodoptera exigua in response to an insect cytokine and its putative membrane action. | Journal of insect physiology 20080601 |
Diversity of inorganic carbon acquisition mechanisms by intact microbial mats of Microcoleus chthonoplastes (Cyanobacteriae, Oscillatoriaceae). | Physiologia plantarum 20080501 |
Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors. | Bioorganic & medicinal chemistry letters 20080415 |
Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct. | Bioorganic & medicinal chemistry letters 20080415 |
Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides. | Bioorganic & medicinal chemistry 20080401 |
Inhibition of carbonic anhydrases with glycosyltriazole benzene sulfonamides. | Journal of medicinal chemistry 20080327 |
Carbonic anhydrase inhibitors: interactions of phenols with the 12 catalytically active mammalian isoforms (CA I-XIV). | Bioorganic & medicinal chemistry letters 20080301 |
Fluid and osmolyte recovery in the common pond snail Lymnaea stagnalis following full-body withdrawal. | The Journal of experimental biology 20080201 |
Carbonic anhydrase inhibitors: copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII. | Bioorganic & medicinal chemistry letters 20080115 |
The alpha and beta classes carbonic anhydrases from Helicobacter pylori as novel drug targets. | Current pharmaceutical design 20080101 |
The development of topically acting carbonic anhydrase inhibitors as antiglaucoma agents. | Current pharmaceutical design 20080101 |
Direct non-cyclooxygenase-2 targets of celecoxib and their potential relevance for cancer therapy. | British journal of cancer 20071203 |
Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides. | Bioorganic & medicinal chemistry 20071201 |
Carbonic anhydrase inhibitors: Selective inhibition of the extracellular, tumor-associated isoforms IX and XII over isozymes I and II with glycosyl-thioureido-sulfonamides. | Bioorganic & medicinal chemistry letters 20070915 |
Carbonic anhydrase inhibitors. Interaction of the antiepileptic drug sulthiame with twelve mammalian isoforms: kinetic and X-ray crystallographic studies. | Bioorganic & medicinal chemistry letters 20070901 |
Carbonic anhydrase inhibitors: inhibition of human, bacterial, and archaeal isozymes with benzene-1,3-disulfonamides--solution and crystallographic studies. | Bioorganic & medicinal chemistry letters 20070801 |
Acclimation of wild-type cells and CO2-insensitive mutants of the green alga Chlorella ellipsoidea to elevated [CO2]. | Plant, cell & environment 20070801 |
Electrical parameters and ion species for active transport in human esophageal stratified squamous epithelium and Barrett's specialized columnar epithelium. | American journal of physiology. Gastrointestinal and liver physiology 20070701 |
Carbonic anhydrases as targets for medicinal chemistry. | Bioorganic & medicinal chemistry 20070701 |
Carbonic anhydrase inhibitors: the beta-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitors. | Bioorganic & medicinal chemistry letters 20070701 |
Carbonic anhydrase II increases the activity of the human electrogenic Na+/HCO3- cotransporter. | The Journal of biological chemistry 20070504 |
Carbonic anhydrase inhibitors: inhibition of isozymes I, II, and IX with triazole-linked O-glycosides of benzene sulfonamides. | Journal of medicinal chemistry 20070405 |
Inhibition of hypoxia-induced calcium responses in pulmonary arterial smooth muscle by acetazolamide is independent of carbonic anhydrase inhibition. | American journal of physiology. Lung cellular and molecular physiology 20070401 |
Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties. | Bioorganic & medicinal chemistry letters 20070315 |
Identification of arylsulfonamides as Aquaporin 4 inhibitors. | Bioorganic & medicinal chemistry letters 20070301 |
Carbonic anhydrase inhibition prevents and reverts cardiomyocyte hypertrophy. | The Journal of physiology 20070215 |
Inhibition of membrane-associated carbonic anhydrase isozymes IX, XII and XIV with a library of glycoconjugate benzenesulfonamides. | Bioorganic & medicinal chemistry letters 20070215 |
Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors. | Journal of medicinal chemistry 20070125 |
Pulmonary vasodilation by acetazolamide during hypoxia is unrelated to carbonic anhydrase inhibition. | American journal of physiology. Lung cellular and molecular physiology 20070101 |
Multiple sources of carbonic anhydrase activity in pea thylakoids: soluble and membrane-bound forms. | Photosynthesis research 20070101 |
The development of topically acting carbonic anhydrase inhibitors as anti-glaucoma agents. | Current topics in medicinal chemistry 20070101 |
Carbonic anhydrase inhibitors: clash with Ala65 as a means for designing inhibitors with low affinity for the ubiquitous isozyme II, exemplified by the crystal structure of the topiramate sulfamide analogue. | Journal of medicinal chemistry 20061130 |
A novel class of carbonic anhydrase inhibitors: glycoconjugate benzene sulfonamides prepared by 'click-tailing'. | Journal of medicinal chemistry 20061102 |
Carbonic anhydrase inhibitors: Hypoxia-activatable sulfonamides incorporating disulfide bonds that target the tumor-associated isoform IX. | Journal of medicinal chemistry 20060907 |
Expression, purification, kinetic, and structural characterization of an alpha-class carbonic anhydrase from Aedes aegypti (AaCA1). | Biochimica et biophysica acta 20060801 |
Effect of human carbonic anhydrase II on the activity of the human electrogenic Na/HCO3 cotransporter NBCe1-A in Xenopus oocytes. | The Journal of biological chemistry 20060714 |
Evidence for a plasmalemma-based CO2 concentrating mechanism in Laminaria saccharina. | Photosynthesis research 20060601 |
Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
Heterogeneous origin of carbonic anhydrase activity of thylakoid membranes. | Biochemistry. Biokhimiia 20060501 |
Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori. | Bioorganic & medicinal chemistry letters 20060415 |
Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs. | Journal of medicinal chemistry 20060323 |
Characterization of H+ and HCO3- transporters in CFPAC-1 human pancreatic duct cells. | World journal of gastroenterology 20060214 |
Carbonic anhydrase inhibitors ameliorate the symptoms of hypokalaemic periodic paralysis in rats by opening the muscular Ca2+-activated-K+ channels. | Neuromuscular disorders : NMD 20060101 |
Cryptococcus neoformans senses CO2 through the carbonic anhydrase Can2 and the adenylyl cyclase Cac1. | Eukaryotic cell 20060101 |
Pea leaf thylakoids contain several carbonic anhydrases. | Doklady. Biochemistry and biophysics 20060101 |
Transport activity of MCT1 expressed in Xenopus oocytes is increased by interaction with carbonic anhydrase. | The Journal of biological chemistry 20051202 |
Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors. | Journal of medicinal chemistry 20051201 |
Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides. | Bioorganic & medicinal chemistry letters 20051101 |
Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozymes IX and XII with a library of aromatic and heteroaromatic sulfonamides. | Bioorganic & medicinal chemistry letters 20051101 |
Modulation of carbonic anhydrase activity in two nitrogen fixing cyanobacteria, Nostoc calcicola and Anabaena sp. | Journal of plant physiology 20051001 |
Carbonic anhydrase inhibitors: inhibition of the transmembrane isozyme XIV with sulfonamides. | Bioorganic & medicinal chemistry letters 20050901 |
Carbonic anhydrase inhibitors: design of thioureido sulfonamides with potent isozyme II and XII inhibitory properties and intraocular pressure lowering activity in a rabbit model of glaucoma. | Bioorganic & medicinal chemistry letters 20050901 |
Carbonic anhydrase inhibitors. Inhibition of red blood cell ostrich (Struthio camelus) carbonic anhydrase with a series of aromatic and heterocyclic sulfonamides. | Journal of enzyme inhibition and medicinal chemistry 20050801 |
Carbonic anhydrase inhibitors. Design of fluorescent sulfonamides as probes of tumor-associated carbonic anhydrase IX that inhibit isozyme IX-mediated acidification of hypoxic tumors. | Journal of medicinal chemistry 20050728 |
Carbonic anhydrase inhibitors. Synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with boron-containing sulfonamides, sulfamides, and sulfamates: toward agents for boron neutron capture therapy of hypoxic tumors. | Bioorganic & medicinal chemistry letters 20050701 |
Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX. | Bioorganic & medicinal chemistry letters 20050615 |
Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes. | Bioorganic & medicinal chemistry letters 20050615 |
Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies. | Bioorganic & medicinal chemistry letters 20050502 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating thioureido-sulfanilyl scaffolds. | Bioorganic & medicinal chemistry letters 20050502 |
HCO3- secretion in the esophageal submucosal glands. | American journal of physiology. Gastrointestinal and liver physiology 20050401 |
Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs? | Bioorganic & medicinal chemistry letters 20050215 |
Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides. | Bioorganic & medicinal chemistry letters 20050215 |
Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides. | Bioorganic & medicinal chemistry letters 20050215 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with bis-sulfamates. | Bioorganic & medicinal chemistry letters 20050201 |
Carbonic anhydrase inhibitors. Novel sulfanilamide/acetazolamide derivatives obtained by the tail approach and their interaction with the cytosolic isozymes I and II, and the tumor-associated isozyme IX. | Bioorganic & medicinal chemistry letters 20050117 |
Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. | Bioorganic & medicinal chemistry letters 20041220 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide. | Bioorganic & medicinal chemistry letters 20041206 |
Photosystem II associated carbonic anhydrase activity in higher plants is situated in core complex. | FEBS letters 20041105 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties. | Bioorganic & medicinal chemistry letters 20041101 |
Theoretical study of gas-phase acidity, pKa, lipophilicity, and solubility of some biologically active sulfonamides. | Bioorganic & medicinal chemistry 20041015 |
Carbonic anhydrase inhibitors: the first on-resin screening of a 4-sulfamoylphenylthiourea library. | Journal of medicinal chemistry 20041007 |
Roles of carbonic anhydrase in photosynthesis of Skeletonema costatum. | Zhi wu sheng li yu fen zi sheng wu xue xue bao = Journal of plant physiology and molecular biology 20041001 |
pH microdomains in oligodendrocytes. | The Journal of biological chemistry 20040827 |
Carbonic anhydrase isoform expression and functional role in rodent extraocular muscle. | Pflugers Archiv : European journal of physiology 20040801 |
Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides. | Bioorganic & medicinal chemistry letters 20040621 |
Inhibition of alpha(1E) Ca(2+) channels by carbonic anhydrase inhibitors. | Journal of pharmacological sciences 20040601 |
Benzolamide is not a membrane-impermeant carbonic anhydrase inhibitor. | Journal of enzyme inhibition and medicinal chemistry 20040601 |
Carbonic anhydrase inhibitors: synthesis and topical intraocular pressure lowering effects of fluorine-containing inhibitors devoid of enhanced reactivity. | Journal of medicinal chemistry 20040520 |
Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with fluorine-containing sulfonamides. The first subnanomolar CA IX inhibitor discovered. | Bioorganic & medicinal chemistry letters 20040503 |
Inhibition of 3T3-L1 adipocyte differentiation by 6-ethoxyzolamide: repressed peroxisome proliferator-activated receptor gamma mRNA and enhanced CCAAT/enhancer binding protein beta mRNA levels. | Biochemical pharmacology 20040501 |
Carbonic anhydrase inhibitors are specific openers of skeletal muscle BK channel of K+-deficient rats. | FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20040401 |
Carbonic anhydrase inhibitors. Inhibition of mitochondrial isozyme V with aromatic and heterocyclic sulfonamides. | Journal of medicinal chemistry 20040226 |
Pdcd4 inhibits growth of tumor cells by suppression of carbonic anhydrase type II. | Molecular and cellular endocrinology 20040212 |
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase. | Bioorganic & medicinal chemistry letters 20040105 |
Sodium and chloride transport in soft water and hard water acclimated zebrafish (Danio rerio). | Biochimica et biophysica acta 20031230 |
Carbonic anhydrase inhibitors: inhibition of transmembrane, tumor-associated isozyme IX, and cytosolic isozymes I and II with aliphatic sulfamates. | Journal of medicinal chemistry 20031204 |
Inorganic carbon limitation induces transcripts encoding components of the CO(2)-concentrating mechanism in Synechococcus sp. PCC7942 through a redox-independent pathway. | Plant physiology 20031201 |
Bicarbonate-dependent depolarizing potentials in pyramidal cells and interneurons during epileptiform activity. | The European journal of neuroscience 20030901 |
Carbonic anhydrase inhibitors: topically acting antiglaucoma sulfonamides incorporating esters and amides of 3- and 4-carboxybenzolamide. | Bioorganic & medicinal chemistry letters 20030901 |
Carbonic anhydrase inhibitors. Inhibition of tumor-associated isozyme IX by halogenosulfanilamide and halogenophenylaminobenzolamide derivatives. | Journal of medicinal chemistry 20030522 |
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors. | Journal of medicinal chemistry 20030522 |
Spinal carbonic anhydrase contributes to nociceptive reflex enhancement by midazolam, pentobarbital, and propofol. | Anesthesiology 20030401 |
Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides. | Bioorganic & medicinal chemistry letters 20030324 |
Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives. | Bioorganic & medicinal chemistry letters 20030310 |
Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV. | Bioorganic & medicinal chemistry letters 20030310 |
Transepithelial sulfate transport by avian renal proximal tubule epithelium in primary culture. | American journal of physiology. Regulatory, integrative and comparative physiology 20021201 |
Inhibition of muscle carbonic anhydrase slows the Ca(2+) transient in rat skeletal muscle fibers. | American journal of physiology. Cell physiology 20021001 |
Proton pump activity is required for active uptake of chloride in isolated amphibian skin exposed to freshwater. | Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20020801 |
Carbonic anhydrase inhibitors. Preparation of potent sulfonamides inhibitors incorporating bile acid tails. | Bioorganic & medicinal chemistry letters 20020617 |
Biochemical and molecular inhibition of plastidial carbonic anhydrase reduces the incorporation of acetate into lipids in cotton embryos and tobacco cell suspensions and leaves. | Plant physiology 20020401 |
Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties. | Journal of medicinal chemistry 20020328 |
Potassium drives daily reversible thallus enlargement in the marine red alga Porphyra leucosticta (Rhodophyta). | Planta 20020301 |
Inhibition of muscle carbonic anhydrase increases rise and relaxation times of twitches in rat skeletal muscle fibres. | Pflugers Archiv : European journal of physiology 20020301 |
Role of carbon dioxide and ion transport in the formation of sub-embryonic fluid by the blastoderm of the Japanese quail. | British poultry science 20020301 |
The catalytic properties of human carbonic anhydrase IX. | Biochemical and biophysical research communications 20011102 |
Ionic mechanisms of GABA-induced long-term potentiation in the rat superior colliculus. | Experimental brain research 20011001 |
Cl(-)-dependent secretory mechanisms in isolated rat bile duct epithelial units. | American journal of physiology. Gastrointestinal and liver physiology 20010801 |
Physiological and molecular biological characterization of intracellular carbonic anhydrase from the marine diatom Phaeodactylum tricornutum. | Plant physiology 20010801 |
A new chloroplast envelope carbonic anhydrase activity is induced during acclimation to low inorganic carbon concentrations in Chlamydomonas reinhardtii. | Planta 20010601 |
Extracellular carbonic anhydrase activity facilitates lactic acid transport in rat skeletal muscle fibres. | The Journal of physiology 20010315 |
Asymmetric subcellular mRNA distribution correlates with carbonic anhydrase activity in Acetabularia acetabulum. | Plant physiology 20010201 |
Inhibition of carbonic anhydrase in the lens does not induce myopia in cynomolgus monkeys. | Upsala journal of medical sciences 20010101 |
© 2019 Angene International Limited. All rights Reserved.