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Home > Other Heterocycles > 21102-94-3
CAS No: 21102-94-3 Catalog No: AG002L57 MDL No:
Title | Journal |
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Blockade of voltage-gated calcium channel Cav1.2 and α1-adrenoceptors increases vertebral artery blood flow induced by the antivertigo agent difenidol. | European journal of pharmacology 20120815 |
Yohimbine antagonises α1A- and α1D-adrenoceptor mediated components in addition to the α2A-adrenoceptor component to pressor responses in the pithed rat. | European journal of pharmacology 20120315 |
Synthesis, biological evaluation, and docking studies of tetrahydrofuran- cyclopentanone- and cyclopentanol-based ligands acting at adrenergic α₁- and serotonine 5-HT1A receptors. | Journal of medicinal chemistry 20120112 |
Molecular and pharmacological characteristics of the gerbil α(1a)-adrenergic receptor. | Hearing research 20120101 |
Effect of inter-renal aortic coarctation-induced hypertension on function and expression of vascular α(1A)- and α(1D)-adrenoceptors. | Canadian journal of physiology and pharmacology 20120101 |
[Medical expulsive therapy facilitated by alpha 1 adrenoceptor antagonist]. | Clinical calcium 20111001 |
Discovery of LASSBio-772, a 1,3-benzodioxole N-phenylpiperazine derivative with potent alpha 1A/D-adrenergic receptor blocking properties. | European journal of medicinal chemistry 20110701 |
Interaction of alpha1D-adrenergic and P2X(7) receptors in the rat lacrimal gland and the effect on intracellular [Ca2+] and protein secretion. | Investigative ophthalmology & visual science 20110701 |
Vasopressor nerve responses in the pithed rat, previously identified as α2-adrenoceptor mediated, may be α1D-adrenoceptor mediated. | European journal of pharmacology 20110511 |
Characterization of α1-adrenoceptor subtypes mediating contraction in human isolated ureters. | Urology 20110301 |
α(1D)-Adrenoceptor regulates the vasopressor action of α(1A)-adrenoceptor in mesenteric vascular bed of α(1D)-adrenoceptor knockout mice. | Autonomic & autacoid pharmacology 20110101 |
1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: structure-affinity/activity relationship at alpha1-adrenoceptor subtypes and at 5-HT1A receptors. | European journal of medicinal chemistry 20100901 |
alpha(1)-Adrenergic receptor subtype function in fetal and adult cerebral arteries. | American journal of physiology. Heart and circulatory physiology 20100601 |
Discovery of a new series of 5-HT1A receptor agonists. | Bioorganic & medicinal chemistry letters 20100315 |
Gene expressions and mechanical functions of α1-adrenoceptor subtypes in mouse ureter. | World journal of urology 20091201 |
Epinephrine, phenylephrine, and methoxamine induce infiltrative anesthesia via alpha1-adrenoceptors in rats. | Acta pharmacologica Sinica 20090901 |
Mechanical function and gene expression of alpha(1)-adrenoceptor subtypes in dog intravesical ureter. | Urology 20090801 |
Adventitia removal does not modify the alphaID-adrenoceptors response in aorta during hypertension and ageing. | Autonomic & autacoid pharmacology 20090701 |
Inhibitory effect of fentanyl on phenylephrine-induced contraction of the rat aorta. | Yonsei medical journal 20090630 |
Phenylephrine contracts porcine pulmonary veins via alpha(1B)-, alpha(1D)-, and alpha(2)-adrenoceptors. | European journal of pharmacology 20090624 |
Serotonin1A-mediated amplification of light-induced phase advances of circadian rhythms in the Syrian hamster: post-light effects. | Brain research 20090123 |
Influence of high dietary sodium intake on the functional subtypes of alpha-adrenoceptors in the renal cortical vasculature of Wistar-Kyoto rats. | Autonomic & autacoid pharmacology 20090101 |
Increased alpha1D adrenergic receptor activity and protein expression in the urinary bladder of aged rats. | World journal of urology 20081201 |
Structure-activity relationships in 1,4-benzodioxan-related compounds. 9. From 1,4-benzodioxane to 1,4-dioxane ring as a promising template of novel alpha1D-adrenoreceptor antagonists, 5-HT1A full agonists, and cytotoxic agents. | Journal of medicinal chemistry 20081023 |
Smooth muscle alpha1D-adrenoceptors mediate phenylephrine-induced vasoconstriction and increases in endothelial cell Ca2+ in hamster cremaster arterioles. | British journal of pharmacology 20081001 |
The alpha1D-adrenergic receptor induces vascular smooth muscle apoptosis via a p53-dependent mechanism. | Molecular pharmacology 20081001 |
Functional subtypes of renal alpha1-adrenoceptor in diabetic and non-diabetic 2K1C Goldblatt renovascular hypertension. | Acta pharmacologica Sinica 20080501 |
Different affinities of native alpha1B-adrenoceptors for ketanserin between intact tissue segments and membrane preparations. | European journal of pharmacology 20080428 |
Role of alpha1-adrenoceptor subtypes in the effects of methylenedioxy methamphetamine (MDMA) on body temperature in the mouse. | British journal of pharmacology 20080201 |
Noradrenergic vasoconstriction of pig prostatic small arteries. | Naunyn-Schmiedeberg's archives of pharmacology 20080201 |
Characteristics of contractile activity in the renal artery of ovariectomized rats. | Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi 20080201 |
Alpha1A- and alpha1D-adrenoceptors are the major functional subtypes of renal alpha1-adrenoceptors in streptozotocin-induced diabetic and normal Sprague-Dawley rats. | Autonomic & autacoid pharmacology 20080101 |
Evidence of alpha1-adrenoceptor functional changes in omental arteries of patients with end-stage renal disease. | Autonomic & autacoid pharmacology 20080101 |
Vascular alpha-1D-adrenoceptors are overexpressed in aorta of the aryl hydrocarbon receptor null mouse: role of increased angiotensin II. | Autonomic & autacoid pharmacology 20080101 |
Alpha(1D)-adrenoceptors mediate nerve and agonist-evoked contractions in mouse vas deferens: evidence obtained from knockout technology. | Autonomic & autacoid pharmacology 20080101 |
Ma huang and alpha subtype adrenoceptors in the cat pulmonary vascular bed. | Journal of dietary supplements 20080101 |
Expressions and mechanical functions of alpha1-adrenoceptor subtypes in hamster ureter. | European journal of pharmacology 20071114 |
Trophic effects induced by alpha1D-adrenoceptors on endothelial cells are potentiated by hypoxia. | American journal of physiology. Heart and circulatory physiology 20071001 |
alpha1-Adrenoceptors in proximal segments of tail arteries from control and reserpinised rats. | Naunyn-Schmiedeberg's archives of pharmacology 20071001 |
Influence of cisplatin-induced renal failure on the alpha(1)-adrenoceptor subtype causing vasoconstriction in the kidney of the rat. | European journal of pharmacology 20070813 |
Alpha1A-adrenoceptors predominate in the control of blood pressure in mouse mesenteric vascular bed. | Autonomic & autacoid pharmacology 20070701 |
Alpha1A-adrenergic receptors are functionally expressed by a subpopulation of cornu ammonis 1 interneurons in rat hippocampus. | The Journal of pharmacology and experimental therapeutics 20070601 |
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes. | Cardiovascular research 20070601 |
Identification of alpha-1L and alpha-1A adrenoceptors in human prostate by tissue segment binding. | The Journal of urology 20070101 |
Vascular alpha1-adrenoceptors in isolated perfused rat kidney: influence of ageing. | Autonomic & autacoid pharmacology 20070101 |
Effect of alpha-adrenoceptor subtype-selective inverse agonists on non-pregnant and late-pregnant cervical resistance in vitro in the rat. | Clinical and experimental pharmacology & physiology 20070101 |
Effects of alpha1D-adrenergic receptors on shedding of biologically active EGF in freshly isolated lacrimal gland epithelial cells. | American journal of physiology. Cell physiology 20061101 |
Alpha(1A/L)-adrenoceptors mediate contraction of the circular smooth muscle of the pig urethra. | Autonomic & autacoid pharmacology 20061001 |
Selective agonists reveal alpha(1A)- and alpha(1B)-adrenoceptor subtypes in caudal artery of the young rat. | Autonomic & autacoid pharmacology 20061001 |
Potentiation of the resetting effects of light on circadian rhythms of hamsters using serotonin and neuropeptide Y receptor antagonists. | Neuroscience 20060901 |
Sympathetic neurotransmission in the rat testicular capsule: functional characterization and identification of mRNA encoding alpha1-adrenoceptor subtypes. | European journal of pharmacology 20060814 |
Alpha1D-adrenoceptor-induced relaxation on rat carotid artery is impaired during the endothelial dysfunction evoked in the early stages of hyperhomocysteinemia. | European journal of pharmacology 20060814 |
Evidence against alpha-adrenoceptors mediating relaxation in rat thoracic aortae: alpha-agonists relaxation depends on interaction with alpha-adrenoceptors. | Fundamental & clinical pharmacology 20060801 |
Heterodimers of alpha1B- and alpha1D-adrenergic receptors form a single functional entity. | Molecular pharmacology 20060101 |
Captopril therapy decreases both expression and function of alpha-adrenoceptors in pre- hypertensive rat aorta. | Autonomic & autacoid pharmacology 20060101 |
A two model receptor system of the alpha1D adrenergic receptor to describe interactions with epinephrine and BMY7378. | Journal of chemical information and modeling 20060101 |
Nandrolone treatment decreases the alpha1B-adrenoceptor mRNA level in rat kidney, but not the density of alpha1B-adrenoceptors in cultured MDCK-D1 kidney cells. | European journal of pharmacology 20051219 |
Correlation between mRNA levels and functional role of alpha1-adrenoceptor subtypes in arteries: evidence of alpha1L as a functional isoform of the alpha1A-adrenoceptor. | American journal of physiology. Heart and circulatory physiology 20051101 |
Correlation between vasoconstrictor roles and mRNA expression of alpha1-adrenoceptor subtypes in blood vessels of genetically engineered mice. | British journal of pharmacology 20051001 |
The alpha (1D)-adrenoceptor antagonist BMY 7378 is also an alpha (2C)-adrenoceptor antagonist. | Autonomic & autacoid pharmacology 20051001 |
Chloroethylclonidine reveals that alpha (1 A)-adrenoceptors mediate contraction in aorta of alpha (1 D)-adrenoceptor knockout mice. | Autonomic & autacoid pharmacology 20051001 |
Differential distribution of functional alph}1-adrenergic receptor subtypes along the rat tail artery. | The Journal of pharmacology and experimental therapeutics 20050801 |
Nitric oxide and cGMP mediate alpha1D-adrenergic receptor-Stimulated protein secretion and p42/p44 MAPK activation in rat lacrimal gland. | Investigative ophthalmology & visual science 20050801 |
Fentanyl attenuates alpha1B-adrenoceptor-mediated pulmonary artery contraction. | Anesthesiology 20050801 |
Postjunctional alpha1-adrenoceptors in the vasculature of the pithed mouse are of the alpha1A-subtype. | Autonomic & autacoid pharmacology 20050701 |
Synthesis and structure-activity relationship of fluoro analogues of 8-{2-[4-(4-methoxyphenyl)piperazin-1yl]ethyl}-8-azaspiro[4.5]decane-7,9-dione as selective alpha(1d)-adrenergic receptor antagonists. | Journal of medicinal chemistry 20050421 |
1,2,4-Benzothiadiazine derivatives as alpha1 and 5-HT1A receptor ligands. | Bioorganic & medicinal chemistry letters 20050215 |
Differential antagonism by conotoxin rho-TIA of contractions mediated by distinct alpha1-adrenoceptor subtypes in rat vas deferens, spleen and aorta. | European journal of pharmacology 20050131 |
Sympathectomy reveals alpha 1A- and alpha 1D-adrenoceptor components to contractions to noradrenaline in rat vas deferens. | British journal of pharmacology 20041101 |
Effects of norepinephrine on alpha-subtype receptors in the feline pulmonary vascular bed. | Critical care medicine 20041101 |
Pharmacological characterization of alpha1-adrenoceptors in mouse isolated femoral small arteries. | European journal of pharmacology 20041025 |
Cloned human 5-HT1A receptor pharmacology determined using agonist binding and measurement of cAMP accumulation. | The Journal of pharmacy and pharmacology 20041001 |
Different roles of alpha1-adrenoceptor subtypes in mediating cardiomyocyte protein synthesis in neonatal rats. | Clinical and experimental pharmacology & physiology 20040901 |
Effects of androgen manipulation on alpha1-adrenoceptor subtypes in the rat seminal vesicle. | Life sciences 20040806 |
Chromatography studies on bio-affinity of nine ligands of alpha1-adrenoceptor to alpha1D subtypes overexpressed in cell membrane. | Science in China. Series C, Life sciences 20040801 |
Alpha1-adrenoceptor subtype substitution in knockout mice. | British journal of pharmacology 20040701 |
Hepatocytes from alpha1B-adrenoceptor knockout mice reveal compensatory adrenoceptor subtype substitution. | British journal of pharmacology 20040701 |
Alpha-1D adrenoceptors are involved in reserpine-induced supersensitivity of rat tail artery. | British journal of pharmacology 20040601 |
The contribution of adrenoceptor subtype(s) in the renal vasculature of diabetic spontaneously hypertensive rats. | British journal of pharmacology 20040601 |
Human alpha1D-adrenoceptor phosphorylation and desensitization. | Biochemical pharmacology 20040515 |
Synthesis, screening, and molecular modeling of new potent and selective antagonists at the alpha 1d adrenergic receptor. | Journal of medicinal chemistry 20040408 |
Evidence that alpha(1B)-adrenoceptors are involved in noradrenaline-induced contractions of rat tail artery. | European journal of pharmacology 20040319 |
Alpha1-adrenoceptor subtypes involved in vasoconstrictor responses to exogenous and neurally released noradrenaline in rat femoral resistance arteries. | British journal of pharmacology 20040301 |
alpha1A-adrenergic receptor mediated pressor response to phenylephrine in anesthetized rat. | Science in China. Series C, Life sciences 20040201 |
The hypotensive effect of BMY 7378 involves central 5-HT1A receptor stimulation in the adult but not in the young rat. | Archives of medical research 20040101 |
Alpha 1-adrenoceptor subtypes mediating noradrenaline-induced contraction of pulmonary artery from pulmonary hypertensive rats. | European journal of pharmacology 20031215 |
Excitatory alpha1-adrenergic receptors predominate over inhibitory beta-receptors in rabbit dorsal detrusor. | The Journal of urology 20031201 |
New pyrimido[5,4-b]indoles as ligands for alpha(1)-adrenoceptor subtypes. | Journal of medicinal chemistry 20030703 |
Effects of intravenous and infravesical administration of suramin, terazosin and BMY 7378 on bladder instability in conscious rats with bladder outlet obstruction. | BJU international 20030701 |
Functional characterization of alpha-adrenoceptors mediating pupillary dilation in rats. | European journal of pharmacology 20030620 |
Effects of castration and of testosterone replacement on alpha(1)-adrenoceptor subtypes in the rat vas deferens. | European journal of pharmacology 20030620 |
Cytosolic Ca2+ and phosphoinositide hydrolysis linked to constitutively active alpha 1D-adrenoceptors in vascular smooth muscle. | The Journal of pharmacology and experimental therapeutics 20030601 |
Interaction between neuropeptide Y Y1 receptors and alpha1B-adrenoceptors in the neurovascular junction of canine splenic arteries. | European journal of pharmacology 20030418 |
Alpha 1-adrenergic receptor responses in alpha 1AB-AR knockout mouse hearts suggest the presence of alpha 1D-AR. | American journal of physiology. Heart and circulatory physiology 20030401 |
Functional alpha1-adrenergic receptor subtypes in human right gastroepiploic artery. | Acta pharmacologica Sinica 20030401 |
Investigation of postjunctional alpha1- and alpha2-adrenoceptor subtypes in vas deferens from wild-type and alpha(2A/D)-adrenoceptor knockout mice. | British journal of pharmacology 20030301 |
Evidence for the role of alpha1D- and alpha1A-adrenoceptors in contraction of the rat mesenteric artery. | Vascular pharmacology 20030201 |
Serotonergic serotonin (1A) mixed agonists/antagonists elicit large-magnitude phase shifts in hamster circadian wheel-running rhythms. | Neuroscience 20030101 |
Pharmacological characterization of alpha1-adrenoceptor in mouse iliac artery. | European journal of pharmacology 20021205 |
5-HT1A receptor-mediated regulation of mitogen-activated protein kinase phosphorylation in rat brain. | European journal of pharmacology 20021004 |
Alpha(1)-adrenoceptor stimulation directly induces growth of vascular wall in vivo. | American journal of physiology. Heart and circulatory physiology 20021001 |
Pharmacological characterization of alpha1-adrenoceptor subtypes in the bovine tail artery. | Journal of veterinary pharmacology and therapeutics 20021001 |
Noradrenaline-induced contraction of human saphenous vein and human internal mammary artery: involvement of different alpha-adrenoceptor subtypes. | Naunyn-Schmiedeberg's archives of pharmacology 20020801 |
(+/-)-Domesticine, a novel and selective alpha1D-adrenoceptor antagonist in animal tissues and human alpha 1-adrenoceptors. | European journal of pharmacology 20020607 |
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes. | Journal of medicinal chemistry 20020411 |
Adrenergic activation of cardiac phospholipase D: role of alpha(1)-adrenoceptor subtypes. | Cardiovascular research 20020401 |
The alpha(1D)-adrenergic receptor directly regulates arterial blood pressure via vasoconstriction. | The Journal of clinical investigation 20020315 |
Modulatory role of a constitutively active population of alpha(1D)-adrenoceptors in conductance arteries. | American journal of physiology. Heart and circulatory physiology 20020201 |
alpha(1A)-adrenoceptors mediate sympathetically evoked pupillary dilation in rats. | The Journal of pharmacology and experimental therapeutics 20020201 |
Changes in alpha(1)-adrenergic vascular reactivity in monocrotaline-treated rats. | Naunyn-Schmiedeberg's archives of pharmacology 20020201 |
Existence of functional alpha1A- and alpha1D- but no alpha1B-adrenoceptor subtypes in rat common carotid arteries. | Japanese journal of pharmacology 20020201 |
Pathological role of a constitutively active population of alpha(1D)-adrenoceptors in arteries of spontaneously hypertensive rats. | British journal of pharmacology 20020101 |
The functional alpha-adrenoceptor in dog caudal vesical arteries is mainly an alpha1A subtype. | Autonomic & autacoid pharmacology 20020101 |
The role of alpha1D-adrenoceptors in prostatic contraction examined using protection studies. | Autonomic & autacoid pharmacology 20020101 |
A-315456: a selective alpha(1D)-adrenoceptor antagonist with minimal dopamine D(2) and 5-HT(1A) receptor affinity. | European journal of pharmacology 20011214 |
Different subtypes of alpha1-adrenoceptor modulate different K+ currents via different signaling pathways in canine ventricular myocytes. | The Journal of biological chemistry 20011102 |
Functional characterization of alpha1-adrenoceptor subtypes in human subcutaneous resistance arteries. | The Journal of pharmacology and experimental therapeutics 20011101 |
alpha(1)-Adrenoceptor subtypes in the mouse mesenteric artery and abdominal aorta. | British journal of pharmacology 20011101 |
Existence of alpha(1A)- and alpha(1B)-adrenoceptor subtypes in canine mandibular alveolar arteries. | Clinical and experimental pharmacology & physiology 20010901 |
Molecular cloning and functional expression of the guinea pig alpha(1a)-adrenoceptor. | European journal of pharmacology 20010831 |
alpha(1D)-Adrenoceptors do not contribute to phosphoinositide hydrolysis in adult rat cardiac myocytes. | Archives of biochemistry and biophysics 20010801 |
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta. | European journal of pharmacology 20010720 |
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists. | The Journal of biological chemistry 20010706 |
Alpha1-adrenoceptor subtypes on rat afferent arterioles assessed by radioligand binding and RT-PCR. | American journal of physiology. Renal physiology 20010701 |
Functional characterization of alpha(1)-adrenoceptor subtypes in human skeletal muscle resistance arteries. | British journal of pharmacology 20010701 |
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries. | European journal of pharmacology 20010622 |
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes. | Japanese journal of pharmacology 20010601 |
Two novel and potent 3-[(o-methoxyphenyl)piperazinylethyl]-5-phenylthien. | Bioorganic & medicinal chemistry letters 20010507 |
Role of spinal alpha1-adrenoceptor subtypes in the bladder reflex in anesthetized rats. | American journal of physiology. Regulatory, integrative and comparative physiology 20010501 |
Use of antisense oligonucleotides to verify the role of the alpha(1A)-adrenergic receptor in the contractility of the rat uterus post partum. | Molecular pharmacology 20010501 |
The role of several alpha(1)- and alpha(2)-adrenoceptor subtypes mediating vasoconstriction in the canine external carotid circulation. | British journal of pharmacology 20010301 |
Failure of AH11110A to functionally discriminate between alpha(1)-adrenoceptor subtypes A, B and D or between alpha(1)- and alpha(2)-adrenoceptors. | European journal of pharmacology 20010301 |
Inositolphosphate formation in thoracic and abdominal rat aorta following Gq/11-coupled receptor stimulation. | Naunyn-Schmiedeberg's archives of pharmacology 20010301 |
Alpha1-adrenoceptor subtypes mediating vasoconstriction in the carotid circulation of anaesthetized pigs: possible avenues for antimigraine drug development. | Cephalalgia : an international journal of headache 20010301 |
The hypotensive effect of BMY 7378 is antagonized by a silent 5-HT(1A) receptor antagonist: comparison with 8-hydroxy-dipropylamino tetralin. | Archives of medical research 20010101 |
Characterization of alpha1-adrenoceptor subtypes mediating noradrenaline-induced contraction of rat epididymal vas deferens in calcium-free medium. | Life sciences 19990101 |
4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]-piperazinyl]-6, 7-dimethoxyquinazoline (L-765,314): a potent and selective alpha1b adrenergic receptor antagonist. | Journal of medicinal chemistry 19980409 |
Pharmacological characterization of recombinant human 5-hydroxytryptamine1A receptors using a novel antagonist radioligand, [3H]WAY-100635. | Life sciences 19970101 |
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