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CAS No: 18426-20-5 Catalog No: AG0075PR MDL No:
Title | Journal |
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Imaging of dopamine D2/3 agonist binding in cocaine dependence: a [11C]NPA positron emission tomography study. | Synapse (New York, N.Y.) 20111201 |
CODA-RET reveals functional selectivity as a result of GPCR heteromerization. | Nature chemical biology 20110901 |
Effect of risperidone on high-affinity state of dopamine D2 receptors: a PET study with agonist ligand [11C](R)-2-CH3O-N-n-propylnorapomorphine. | The international journal of neuropsychopharmacology 20110201 |
Effects of unilateral 6-OHDA lesions on [3H]-N-propylnorapomorphine binding in striatum ex vivo and vulnerability to amphetamine-evoked dopamine release in rat. | Neurochemistry international 20110201 |
Dopamine beta-hydroxylase-deficient mice have normal densities of D(2) dopamine receptors in the high-affinity state based on in vivo PET imaging and in vitro radioligand binding. | Synapse (New York, N.Y.) 20100901 |
D2 receptor occupancy in conscious rat brain is not significantly distinguished with [3H]-MNPA, [3H]-(+)-PHNO, and [3H]-raclopride. | Synapse (New York, N.Y.) 20100801 |
A comparative evaluation of the dopamine D(2/3) agonist radiotracer [11C](-)-N-propyl-norapomorphine and antagonist [11C]raclopride to measure amphetamine-induced dopamine release in the human striatum. | The Journal of pharmacology and experimental therapeutics 20100501 |
Co-operativity in agonist binding at the D2 dopamine receptor: evidence from agonist dissociation kinetics. | Journal of neurochemistry 20100301 |
Measurement error analysis for the determination of dopamine D(2) receptor occupancy using the agonist radioligand [(11)C]MNPA. | Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20100101 |
Agonist binding fraction of dopamine D2/3 receptors in rat brain: a quantitative autoradiographic study. | Neurochemistry international 20100101 |
Advancement in PET quantification using 3D-OP-OSEM point spread function reconstruction with the HRRT. | European journal of nuclear medicine and molecular imaging 20091001 |
Dopamine D(2/3) receptor occupancy of apomorphine in the nonhuman primate brain--a comparative PET study with [11C]raclopride and [11C]MNPA. | Synapse (New York, N.Y.) 20090501 |
Quantitative PET analysis of the dopamine D2 receptor agonist radioligand 11C-(R)-2-CH3O-N-n-propylnorapomorphine in the human brain. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20090501 |
Human biodistribution and dosimetry of the D2/3 agonist 11C-N-propylnorapomorphine (11C-NPA) determined from PET. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20090501 |
The A(2B)-D(2) receptor interaction that controls carotid body catecholamines release locates between the last two steps of hypoxic transduction cascade. | Advances in experimental medicine and biology 20090101 |
Effects of dorsal striatal infusions of R(-)-propylnorapomorphine on kappa-opioid-mediated locomotor activity in the young rat: possible role of the indirect pathway. | Neuroscience 20080826 |
Synthesis and evaluation of novel pyridine based PLG tripeptidomimetics. | Organic & biomolecular chemistry 20080507 |
Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors. | Archives of pharmacal research 20080401 |
Synthesis and dopamine receptor affinities of N-alkyl-11-hydroxy-2-methoxynoraporphines: N-alkyl substituents determine D1 versus D2 receptor selectivity. | Journal of medicinal chemistry 20080227 |
Modulation of heroin and cocaine self-administration by dopamine D1- and D2-like receptor agonists in rhesus monkeys. | The Journal of pharmacology and experimental therapeutics 20070601 |
Amphetamine-induced dopamine release: duration of action as assessed with the D2/3 receptor agonist radiotracer (-)-N-[(11)C]propyl-norapomorphine ([11C]NPA) in an anesthetized nonhuman primate. | Synapse (New York, N.Y.) 20070201 |
Advances in development of dopaminergic aporphinoids. | Journal of medicinal chemistry 20070125 |
Subchronic intermittent caffeine administration to unilaterally 6-hydroxydopamine-lesioned rats sensitizes turning behaviour in response to dopamine D(1) but not D(2) receptor agonists. | Behavioural pharmacology 20051201 |
Measurement of the proportion of D2 receptors configured in state of high affinity for agonists in vivo: a positron emission tomography study using [11C]N-propyl-norapomorphine and [11C]raclopride in baboons. | The Journal of pharmacology and experimental therapeutics 20051001 |
Mechanisms of inverse agonist action at D2 dopamine receptors. | British journal of pharmacology 20050501 |
A preliminary PET evaluation of the new dopamine D2 receptor agonist [11C]MNPA in cynomolgus monkey. | Nuclear medicine and biology 20050501 |
Effects of dopamine, SKF-38393 and R(-)-NPA on ATP-activated currents in rat DRG neurons. | Canadian journal of physiology and pharmacology 20050301 |
Effects of the intravitreal administration of dopaminergic ligands on the b-wave amplitude of the rabbit electroretinogram. | Vision research 20050101 |
Design, synthesis and evaluation of a PLG tripeptidomimetic based on a pyridine scaffold. | Journal of medicinal chemistry 20041216 |
In vivo vulnerability to competition by endogenous dopamine: comparison of the D2 receptor agonist radiotracer (-)-N-[11C]propyl-norapomorphine ([11C]NPA) with the D2 receptor antagonist radiotracer [11C]-raclopride. | Synapse (New York, N.Y.) 20040601 |
Investigation of the mechanism of agonist and inverse agonist action at D2 dopamine receptors. | Biochemical pharmacology 20040501 |
Quantitative analysis of (-)-N-(11)C-propyl-norapomorphine in vivo binding in nonhuman primates. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20040201 |
Constitutive oligomerization of human D2 dopamine receptors expressed in Spodoptera frugiperda 9 (Sf9) and in HEK293 cells. Analysis using co-immunoprecipitation and time-resolved fluorescence resonance energy transfer. | European journal of biochemistry 20031001 |
Iso-lactam and reduced amide analogues of the peptidomimetic dopamine receptor modulator 3(R)-[(2(S)-pyrrolidinylcarbonyl)amino]-2-oxo-1-pyrrolidineacetamide. | Bioorganic & medicinal chemistry 20030901 |
Endogenous RGS proteins facilitate dopamine D(2S) receptor coupling to G(alphao) proteins and Ca2+ responses in CHO-K1 cells. | FEBS letters 20030102 |
Reversible and irreversible components of [(3)H]-N-propylnorapomorphine interaction with rat striatal membranes. | Neuroscience letters 20020607 |
Specific binding of [(11)C]raclopride and N-[(3)H]propyl-norapomorphine to dopamine receptors in living mouse striatum: occupancy by endogenous dopamine and guanosine triphosphate-free G protein. | Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20020501 |
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
Partial dopamine agonists in the treatment of psychosis. | Journal of neural transmission (Vienna, Austria : 1996) 20020301 |
Agonist-independent and -dependent oligomerization of dopamine D(2) receptors by fusion to fluorescent proteins. | FEBS letters 20011019 |
Receptor crosstalk protein, calcyon, regulates affinity state of dopamine D1 receptors. | European journal of pharmacology 20010921 |
D2 dopamine receptors in striatal medium spiny neurons reduce L-type Ca2+ currents and excitability via a novel PLC[beta]1-IP3-calcineurin-signaling cascade. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20001215 |
Dopamine D1- and D2-like receptor mechanisms in relapse to cocaine-seeking behavior: effects of selective antagonists and agonists. | The Journal of pharmacology and experimental therapeutics 20000801 |
Dopaminergic mechanisms in relapse to cocaine-seeking behavior. Implications for medications development. | Annals of the New York Academy of Sciences 20000101 |
Enhanced striatal dopamine D(2) receptor-induced [35S]GTPgammaS binding after haloperidol treatment. | European journal of pharmacology 19991008 |
Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist. | Nature 19990722 |
Bromocriptine transcriptionally activates the multidrug resistance gene (pgp2/mdr1b) by a novel pathway. | The Journal of biological chemistry 19970425 |
Nafadotride, a potent preferential dopamine D3 receptor antagonist, activates locomotion in rodents. | The Journal of pharmacology and experimental therapeutics 19951201 |
A functional test identifies dopamine agonists selective for D3 versus D2 receptors. | Neuroreport 19950126 |
Expression and pharmacological characterization of the human D3 dopamine receptor. | The Journal of pharmacology and experimental therapeutics 19940101 |
Dopamine D4 versus D2 receptor selectivity of dopamine receptor antagonists: possible therapeutic implications. | European journal of pharmacology 19930604 |
Behavioural pharmacology of imidazole, a potential antidepressant agent. | Archives internationales de pharmacodynamie et de therapie 19851001 |
Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain. | European journal of pharmacology 19840720 |
Neurotensin affects hyperactivity but not stereotypy induced by pre and post synaptic dopaminergic stimulation. | Neuroscience and biobehavioral reviews 19830101 |
Influence of lisuride on morphine withdrawal signs in the rat: a dopamine-mimetic effect. | Psychopharmacology 19820101 |
Penile erection induced by apomorphine and N-n-propyl-norapomorphine in rats. | Archives internationales de pharmacodynamie et de therapie 19791201 |
Treatment of Parkinson's disease with aporphines. Possible role of growth hormone. | The New England journal of medicine 19760311 |
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