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Home > Pyridines > 162760-96-5
162760-96-5 | Cyclohexanecarboxamide, N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl-
CAS No: 162760-96-5 Catalog No: AG001TEY MDL No:MFCD00916243
Product Description
Catalog Number:
AG001TEY
Chemical Name:
Cyclohexanecarboxamide, N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl-
CAS Number:
162760-96-5
Molecular Formula:
C25H34N4O2
Molecular Weight:
422.5631
MDL Number:
MFCD00916243
IUPAC Name:
N-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-N-pyridin-2-ylcyclohexanecarboxamide
InChI:
InChI=1S/C25H34N4O2/c1-31-23-12-6-5-11-22(23)28-18-15-27(16-19-28)17-20-29(24-13-7-8-14-26-24)25(30)21-9-3-2-4-10-21/h5-8,11-14,21H,2-4,9-10,15-20H2,1H3
InChI Key:
SBPRIAGPYFYCRT-UHFFFAOYSA-N
SMILES:
COc1ccccc1N1CCN(CC1)CCN(C(=O)C1CCCCC1)c1ccccn1
UNII:
71IH826FEG
Properties
Complexity:
546
Compound Is Canonicalized:
Yes
Covalently-Bonded Unit Count:
1
Defined Atom Stereocenter Count:
0
Defined Bond Stereocenter Count:
0
Exact Mass:
422.268g/mol
Formal Charge:
0
Heavy Atom Count:
31
Hydrogen Bond Acceptor Count:
5
Hydrogen Bond Donor Count:
0
Isotope Atom Count:
0
Molecular Weight:
422.573g/mol
Monoisotopic Mass:
422.268g/mol
Rotatable Bond Count:
7
Topological Polar Surface Area:
48.9A^2
Undefined Atom Stereocenter Count:
0
Undefined Bond Stereocenter Count:
0
XLogP3:
4.2
Literature
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| Gene expression in the anterior cingulate cortex and amygdala of adolescent marmoset monkeys following parental separations in infancy. | The international journal of neuropsychopharmacology 20090701 |
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| The role of the dorsal raphe nucleus in the development, expression, and treatment of L-dopa-induced dyskinesia in hemiparkinsonian rats. | Synapse (New York, N.Y.) 20090701 |
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| The selective 5-hydroxytryptamine 1A antagonist, AZD7371 [3(R)-(N,N-dicyclobutylamino)-8-fluoro-3,4-dihydro-2H-1-benzopyran-5-carboxamide (R,R)-tartrate monohydrate] (robalzotan tartrate monohydrate), inhibits visceral pain-related visceromotor, but not autonomic cardiovascular, responses to colorectal distension in rats. | The Journal of pharmacology and experimental therapeutics 20090601 |
| Imipramine counteracts corticosterone-induced alterations in the effects of the activation of 5-HT(7) receptors in rat hippocampus. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20090601 |
| Contribution of the striatum to the effects of 5-HT1A receptor stimulation in L-DOPA-treated hemiparkinsonian rats. | Journal of neuroscience research 20090515 |
| 5-HT(1A) receptor and 5-HTT binding during the menstrual cycle in healthy women examined with [(11)C] WAY100635 and [(11)C] MADAM PET. | Psychiatry research 20090430 |
| Dopamine D4 receptor involvement in the discriminative stimulus effects in rats of LSD, but not the phenethylamine hallucinogen DOI. | Psychopharmacology 20090401 |
| Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity, part 1. | European journal of medicinal chemistry 20090401 |
| Reversal of physiological deficits caused by diminished levels of peptidylglycine alpha-amidating monooxygenase by dietary copper. | Endocrinology 20090401 |
| Lateralization of the serotonin-1A receptor distribution in language areas revealed by PET. | NeuroImage 20090401 |
| Antinociceptive effect and GC/MS analysis of Rosmarinus officinalis L. essential oil from its aerial parts. | Planta medica 20090401 |
| Interactions between the serotonergic and histaminergic systems in the central cardiovascular regulation in haemorrhage-shocked rats: involvement of 5-HT(1A) receptors. | Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20090401 |
| The counteraction of opioid-induced ventilatory depression by the serotonin 1A-agonist 8-OH-DPAT does not antagonize antinociception in rats in situ and in vivo. | Anesthesia and analgesia 20090401 |
| Kaempferol from the leaves of Apocynum venetum possesses anxiolytic activities in the elevated plus maze test in mice. | Phytomedicine : international journal of phytotherapy and phytopharmacology 20090401 |
| Inhibitory effects of osemozotan, a serotonin 1A-receptor agonist, on methamphetamine-induced c-Fos expression in prefrontal cortical neurons. | Biological & pharmaceutical bulletin 20090401 |
| The involvement of serotonergic system in the antidepressant effect of zinc in the forced swim test. | Progress in neuro-psychopharmacology & biological psychiatry 20090317 |
| Unilateral lesion of the nigrostriatal pathway induces an increase of neuronal firing of the midbrain raphe nuclei 5-HT neurons and a decrease of their response to 5-HT(1A) receptor stimulation in the rat. | Neuroscience 20090317 |
| Effects of bifeprunox and aripiprazole on rat serotonin and dopamine neuronal activity and anxiolytic behaviour. | Journal of psychopharmacology (Oxford, England) 20090301 |
| Chronic reductions in serotonin transporter function prevent 5-HT1B-induced behavioral effects in mice. | Biological psychiatry 20090301 |
| Characterization of serotonin receptors in pregnant human myometrium. | The Journal of pharmacology and experimental therapeutics 20090301 |
| Decline in serotonergic firing activity and desensitization of 5-HT1A autoreceptors after chronic unpredictable stress. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20090301 |
| Antagonism of 5-HT(1A) receptors uncovers an excitatory effect of SSRIs on 5-HT neuronal activity, an action probably mediated by 5-HT(7) receptors. | Journal of neurochemistry 20090301 |
| An antihyperkinetic action by the serotonin 1A-receptor agonist osemozotan co-administered with psychostimulants or the non-stimulant atomoxetine in mice. | Journal of pharmacological sciences 20090301 |
| Serotonin 5-HT(2) and 5-HT(1A)-like receptors differentially modulate aggressive behaviors in Drosophila melanogaster. | Neuroscience 20090218 |
| Role of serotonin 5-HT1A receptors in the antidepressant-like effect and the antinociceptive effect of venlafaxine in mice. | The international journal of neuropsychopharmacology 20090201 |
| Allosteric modulation of 5-HT(1A) receptors by zinc: Binding studies. | Neuropharmacology 20090201 |
| Antinociceptive activity of Tilia americana var. mexicana inflorescences and quercetin in the formalin test and in an arthritic pain model in rats. | Neuropharmacology 20090201 |
| WAY 100635 produces discriminative stimulus effects in rats mediated by dopamine D(4) receptor activation. | Behavioural pharmacology 20090201 |
| Inhibition of monoamine oxidases desensitizes 5-HT1A autoreceptors and allows nicotine to induce a neurochemical and behavioral sensitization. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20090128 |
| Activation of serotonin 5-HT1-receptors decreased gripping-induced immobility episodes in taiep rats. | Neuroscience letters 20090109 |
| A fully automated one-pot synthesis of [carbonyl-11C]WAY-100635 for clinical PET applications. | Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20090101 |
| Cocaine conditioning: reversal by autoreceptor dose levels of 8-OHDPAT. | Pharmacology, biochemistry, and behavior 20090101 |
| 5-HT(1A) receptors in the frontal cortical brain areas in Cloninger type 1 and 2 alcoholics measured by whole-hemisphere autoradiography. | Alcohol and alcoholism (Oxford, Oxfordshire) 20090101 |
| 5-HT1A receptors are involved in the cannabidiol-induced attenuation of behavioural and cardiovascular responses to acute restraint stress in rats. | British journal of pharmacology 20090101 |
| [Involvement of presynaptic 5-HT1A receptors in immunomodulation under conditions of psychoemotional state]. | Zhurnal vysshei nervnoi deiatelnosti imeni I P Pavlova 20090101 |
| Bilobalide modulates serotonin-controlled behaviors in the nematode Caenorhabditis elegans. | BMC neuroscience 20090101 |
| Reduction of the number of new cells reaching olfactory bulbs impairs olfactory perception in the adult opossum. | Acta neurobiologiae experimentalis 20090101 |
| Bidirectional modulation of classical fear conditioning in mice by 5-HT(1A) receptor ligands with contrasting intrinsic activities. | Neuropharmacology 20090101 |
| The effects of the 5-HT(6) receptor agonist EMD and the 5-HT(7) receptor agonist AS19 on memory formation. | Behavioural brain research 20081216 |
| Ex vivo study of 5-HT(1A) and 5-HT(7) receptor agonists and antagonists on cAMP accumulation during memory formation and amnesia. | Behavioural brain research 20081216 |
| The serotonin-1A receptor distribution in healthy men and women measured by PET and [carbonyl-11C]WAY-100635. | European journal of nuclear medicine and molecular imaging 20081201 |
| Social instigation and aggressive behavior in mice: role of 5-HT1A and 5-HT1B receptors in the prefrontal cortex. | Psychopharmacology 20081201 |
| Neurochemical, behavioral, and physiological effects of pharmacologically enhanced serotonin levels in serotonin transporter (SERT)-deficient mice. | Psychopharmacology 20081201 |
| WAY100635 prevents the changes induced by fluoxetine upon the 5-HT1A receptor functionality. | Neuropharmacology 20081201 |
| Striatal 5-HT1A receptor stimulation reduces D1 receptor-induced dyskinesia and improves movement in the hemiparkinsonian rat. | Neuropharmacology 20081201 |
| Anxiolytic activity of a phytochemically characterized Passiflora incarnata extract is mediated via the GABAergic system. | Planta medica 20081201 |
| 5-HT(1A) and 5-HT(1B) receptors in the ventrolateral striatum differentially modulate apomorphine-induced jaw movements in rats. | Journal of oral science 20081201 |
| Involvement of median raphe nucleus 5-HT1A receptors in the regulation of generalized anxiety-related defensive behaviours in rats. | Neuroscience letters 20081121 |
| Asenapine increases dopamine, norepinephrine, and acetylcholine efflux in the rat medial prefrontal cortex and hippocampus. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20081101 |
| Modification of the effects of 5-methoxy-N,N-dimethyltryptamine on exploratory behavior in rats by monoamine oxidase inhibitors. | Psychopharmacology 20081101 |
| Involvement of glutamate neurotransmission and N-methyl-d-aspartate receptor in the activation of midbrain dopamine neurons by 5-HT1A receptor agonists: an electrophysiological study in the rat. | Neuroscience 20081028 |
| Cholesterol reduction attenuates 5-HT1A receptor-mediated signaling in human primary neuronal cultures. | Naunyn-Schmiedeberg's archives of pharmacology 20081001 |
| Aripiprazole inhibits marble-burying behavior via 5-hydroxytryptamine (5-HT)1A receptor-independent mechanisms. | European journal of pharmacology 20080911 |
| Evidence for serotonin synthesis-dependent regulation of in vitro neuronal firing rates in the midbrain raphe complex. | European journal of pharmacology 20080820 |
| Stress-induced hyperthermia and basal body temperature are mediated by different 5-HT(1A) receptor populations: a study in SERT knockout rats. | European journal of pharmacology 20080820 |
| Improvement of phencyclidine-induced social behaviour deficits in rats: involvement of 5-HT1A receptors. | Behavioural brain research 20080805 |
| Involvement of 5HT1A receptors in the anxiolytic-like effects of cannabidiol injected into the dorsolateral periaqueductal gray of rats. | Psychopharmacology 20080801 |
| Fluoxetine-induced proliferation and differentiation of neural progenitor cells isolated from rat postnatal cerebellum. | Biochemical pharmacology 20080801 |
| Diphenyl diselenide exerts anxiolytic-like effect in Wistar rats: putative roles of GABAA and 5HT receptors. | Progress in neuro-psychopharmacology & biological psychiatry 20080801 |
| Delta(9)-tetrahydrocannabinol prolongs the immobility time in the mouse forced swim test: involvement of cannabinoid CB(1) receptor and serotonergic system. | European journal of pharmacology 20080728 |
| Studies toward the discovery of the next generation of antidepressants. Part 6: Dual 5-HT1A receptor and serotonin transporter affinity within a class of arylpiperazinyl-cyclohexyl indole derivatives. | Bioorganic & medicinal chemistry 20080715 |
| Serotonin inhibits GABA synaptic transmission in presympathetic paraventricular nucleus neurons. | Neuroscience letters 20080711 |
| Sporadic autonomic dysregulation and death associated with excessive serotonin autoinhibition. | Science (New York, N.Y.) 20080704 |
| Behavior selectively elicited by novel stimuli: modulation by the 5-HT1A agonist 8-OHDPAT and antagonist WAY-100635. | Behavioural pharmacology 20080701 |
| [Impact of serotonin 1A receptors in the kappa-opioid immunosuppression]. | Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20080701 |
| Alpha-Ca2+/calmodulin-dependent protein kinase II contributes to the developmental programming of anxiety in serotonin receptor 1A knock-out mice. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20080611 |
| Phencyclidine-induced cognitive deficits in mice are improved by subsequent subchronic administration of the antipsychotic drug perospirone: role of serotonin 5-HT1A receptors. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20080601 |
| Further evidence for an antidepressant potential of the selective sigma1 agonist SA 4503: electrophysiological, morphological and behavioural studies. | The international journal of neuropsychopharmacology 20080601 |
| Role of spinal 5-HT receptors in cutaneous hypersensitivity induced by REM sleep deprivation. | Pharmacological research 20080601 |
| Effect of co-administration of the selective 5-HT1A receptor antagonist WAY 100,635 and selective 5-HT1B/1D receptor antagonist GR 127,935 on anxiolytic effect of citalopram in conditioned fear stress in the rat. | European journal of pharmacology 20080531 |
| Discovery of potent, orally bioavailable, selective 5-HT1A/B/D receptor antagonists. | Journal of medicinal chemistry 20080522 |
| Reduced sensitivity to MDMA-induced facilitation of social behaviour in MDMA pre-exposed rats. | Progress in neuro-psychopharmacology & biological psychiatry 20080515 |
| 5-HT1A receptors of the lateral septum regulate inhibitory avoidance but not escape behavior in rats. | Pharmacology, biochemistry, and behavior 20080501 |
| Nicotine-activated descending facilitation on spinal NMDA-dependent reflex potentiation from pontine tegmentum in rats. | American journal of physiology. Renal physiology 20080501 |
| Serotonin decreases HIV-1 replication in primary cultures of human macrophages through 5-HT(1A) receptors. | British journal of pharmacology 20080501 |
| Role of serotonergic input to the ventrolateral medulla in expression of the 10-Hz sympathetic nerve rhythm. | American journal of physiology. Regulatory, integrative and comparative physiology 20080501 |
| Behavioral characterization of serotonergic activation in the flatworm Planaria. | Behavioural pharmacology 20080501 |
| Evidence for topographically organized endogenous 5-HT-1A receptor-dependent feedback inhibition of the ascending serotonin system. | The European journal of neuroscience 20080501 |
| 5-HT1A receptors in the dorsal hippocampus mediate the anxiogenic effect induced by the stimulation of 5-HT neurons in the median raphe nucleus. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20080401 |
| Serotonin activates presynaptic and postsynaptic receptors in rat globus pallidus. | Journal of neurophysiology 20080401 |
| Modeling considerations for 11C-CUMI-101, an agonist radiotracer for imaging serotonin 1A receptor in vivo with PET. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20080401 |
| Fish on Prozac: effect of serotonin reuptake inhibitors on cognition in goldfish. | Behavioral neuroscience 20080401 |
| Serotonin 1A receptor reductions in postpartum depression: a positron emission tomography study. | Fertility and sterility 20080301 |
| Regulation of conditioned and unconditioned fear in rats by 5-HT1A receptors in the dorsal periaqueductal gray. | Pharmacology, biochemistry, and behavior 20080301 |
| Serotonergic neurotransmission mediates hypothermia induced by the N-phenylpiperazine antipsychotic prototypes LASSBio-579 and LASSBio-581. | Pharmacology, biochemistry, and behavior 20080301 |
| Phrenic nerve activity is enhanced by 5-HT1A receptor agonist 8-OH-DPAT in spontaneously breathing anesthetized rats. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20080301 |
| Antipsychotics differ in their ability to internalise human dopamine D2S and human serotonin 5-HT1A receptors in HEK293 cells. | European journal of pharmacology 20080226 |
| Do selective serotonin reuptake inhibitors acutely increase frontal cortex levels of serotonin? | European journal of pharmacology 20080212 |
| 5-HT2 receptor activation in the midbrain periaqueductal grey (PAG) reduces anxiety-like behaviour in mice. | Behavioural brain research 20080211 |
| Sex differences in the serotonin 1A receptor and serotonin transporter binding in the human brain measured by PET. | NeuroImage 20080201 |
| Perinatal exposure to 5-methoxytryptamine, behavioural-stress reactivity and functional response of 5-HT1A receptors in the adolescent rat. | Behavioural brain research 20080110 |
| A positron emission tomography study to assess binding of lecozotan, a novel 5-hydroxytryptamine-1A silent antagonist, to brain 5-HT1A receptors in healthy young and elderly subjects, and in patients with Alzheimer's disease. | Clinical pharmacology and therapeutics 20080101 |
| In vivo/ex vivo and behavioural study on central effects of 5-HT1B/1D and 5-HT1A antagonists in guinea pigs. | Pharmacology, biochemistry, and behavior 20080101 |
| Hallucinogen-like effects of N,N-dipropyltryptamine (DPT): possible mediation by serotonin 5-HT1A and 5-HT2A receptors in rodents. | Pharmacology, biochemistry, and behavior 20080101 |
| Activation of septal 5-HT1A receptors alters spatial memory encoding, interferes with consolidation, but does not affect retrieval in rats subjected to a water-maze task. | Hippocampus 20080101 |
| The stimulus effects of 8-OH-DPAT: evidence for a 5-HT2A receptor-mediated component. | Pharmacology, biochemistry, and behavior 20080101 |
| Activation of 5-HT(1A) receptors attenuates tachycardia induced by restraint stress in rats. | American journal of physiology. Regulatory, integrative and comparative physiology 20080101 |
| Effects of 5-HT drugs in prefrontal cortex during memory formation and the ketamine amnesia-model. | Hippocampus 20080101 |
| 5-HT1A receptors mediate (+)8-OH-DPAT-stimulation of extracellular signal-regulated kinase (MAP kinase) in vivo in rat hypothalamus: time dependence and regional differences. | Brain research 20071205 |
| A PET study on regional coexpression of 5-HT1A receptors and 5-HTT in the human brain. | Psychopharmacology 20071201 |
| Substance P neurokinin 1 receptor activation within the dorsal raphe nucleus controls serotonin release in the mouse frontal cortex. | Molecular pharmacology 20071201 |
| WAY-100635 has high selectivity for serotonin 5-HT(1A) versus dopamine D(4) receptors. | European journal of pharmacology 20071121 |
| The influence of modifications in imide fragment structure on 5-HT(1A) and 5-HT(7) receptor affinity and in vivo pharmacological properties of some new 1-(m-trifluoromethylphenyl)piperazines. | Bioorganic & medicinal chemistry 20071115 |
| 3,4-Methylenedioxymethamphetamine- and 8-hydroxy-2-di-n-propylamino-tetralin-induced hypothermia: role and location of 5-hydroxytryptamine 1A receptors. | The Journal of pharmacology and experimental therapeutics 20071101 |
| Characterization of 4-(2-hydroxyphenyl)-1-[2'-[N-(2''-pyridinyl)-p-fluorobenzamido]ethyl]piperazine (p-DMPPF) as a new potent 5-HT1A antagonist. | British journal of pharmacology 20071101 |
| Anxiolytic-like action of MTEP expressed in the conflict drinking Vogel test in rats is serotonin dependent. | Neuropharmacology 20071101 |
| Diabetes-induced changes in 5-hydroxytryptamine modulation of vagally-induced bradycardia in rat heart. | Clinical and experimental pharmacology & physiology 20071101 |
| Reciprocal effects of combined administration of serotonin, noradrenaline and dopamine reuptake inhibitors on serotonin and dopamine levels in the rat prefrontal cortex: the role of 5-HT1A receptors. | Journal of psychopharmacology (Oxford, England) 20071101 |
| The selective 5-HT1A receptor antagonist WAY-100635 inhibits neuronal activity of the ventromedial prefrontal cortex in a rodent model of Parkinson's disease. | Neuroscience bulletin 20071101 |
| Correlation of human cold pressor pain responses with 5-HT(1A) receptor binding in the brain. | Brain research 20071003 |
| Effect of early rearing conditions on alcohol drinking and 5-HT1A receptor function in C57BL/6J mice. | The international journal of neuropsychopharmacology 20071001 |
| A positron emission tomography study of 5-hydroxytryptamine-1A receptors in Alzheimer disease. | The American journal of geriatric psychiatry : official journal of the American Association for Geriatric Psychiatry 20071001 |
| Descending facilitation of spinal NMDA-dependent reflex potentiation from pontine tegmentum in rats. | American journal of physiology. Renal physiology 20071001 |
| Receptor mediation of exaggerated responses to serotonin-enhancing drugs in serotonin transporter (SERT)-deficient mice. | Neuropharmacology 20071001 |
| Serotonin-1A receptor imaging in recurrent depression: replication and literature review. | Nuclear medicine and biology 20071001 |
| [Presynaptic 5-HT1A receptors in immunomodulation]. | Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20071001 |
| Regulation of serotonin-1A receptor function in inducible brain-derived neurotrophic factor knockout mice after administration of corticosterone. | Biological psychiatry 20070901 |
| Distinct electrophysiological effects of paliperidone and risperidone on the firing activity of rat serotonin and norepinephrine neurons. | Psychopharmacology 20070901 |
| Differential effects of aripiprazole on D(2), 5-HT(2), and 5-HT(1A) receptor occupancy in patients with schizophrenia: a triple tracer PET study. | The American journal of psychiatry 20070901 |
| Hippocampal Bcl-2 expression is selectively increased following chronic but not acute treatment with antidepressants, 5-HT(1A) or 5-HT(2C/2B) receptor antagonists. | European journal of pharmacology 20070813 |
| Mechanical, thermal and formalin-induced nociception is differentially altered in 5-HT1A-/-, 5-HT1B-/-, 5-HT2A-/-, 5-HT3A-/- and 5-HTT-/- knock-out male mice. | Pain 20070801 |
| Parametric and regional maps of free serotonin 5HT1A receptor sites in human brain as function of age in healthy humans. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20070801 |
| 6-Hydroxybuspirone is a major active metabolite of buspirone: assessment of pharmacokinetics and 5-hydroxytryptamine1A receptor occupancy in rats. | Drug metabolism and disposition: the biological fate of chemicals 20070801 |
| Role of serotonin 5-HT1A and opioid receptors in the antiallodynic effect of tramadol in the chronic constriction injury model of neuropathic pain in rats. | Psychopharmacology 20070701 |
| A PET study of effects of chronic 3,4-methylenedioxymethamphetamine (MDMA, 'ecstasy') on serotonin markers in Göttingen minipig brain. | Synapse (New York, N.Y.) 20070701 |
| Antagonist-induced increase in 5-HT1A-receptor expression in adult rat hippocampus and cortex. | Synapse (New York, N.Y.) 20070701 |
| Measurement of 5-HT1A receptor binding in depressed adults before and after antidepressant drug treatment using positron emission tomography and [11C]WAY-100635. | Synapse (New York, N.Y.) 20070701 |
| Dopamine released from 5-HT terminals is the cause of L-DOPA-induced dyskinesia in parkinsonian rats. | Brain : a journal of neurology 20070701 |
| Behavioral effects of dipropyltryptamine in rats: evidence for 5-HT1A and 5-HT2A agonist activity. | Behavioural pharmacology 20070701 |
| Suppression of conditioning to ambiguous cues by pharmacogenetic inhibition of the dentate gyrus. | Nature neuroscience 20070701 |
| Role of 5-HT receptor antagonists in mediating intracavernous pressure response induced by fluvoxamine in conscious rats. | The journal of sexual medicine 20070701 |
| Anxiolytic-like effects of sinapic acid in mice. | Life sciences 20070627 |
| Antipsychotic-like effect by combined treatment with citalopram and WAY 100635: involvement of the 5-HT2C receptor. | The international journal of neuropsychopharmacology 20070601 |
| Optimal metabolite curve fitting for kinetic modeling of 11C-WAY-100635. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20070601 |
| A role for oxytocin and 5-HT(1A) receptors in the prosocial effects of 3,4 methylenedioxymethamphetamine ('ecstasy'). | Neuroscience 20070511 |
| Reduced serotonin-1A receptor binding in social anxiety disorder. | Biological psychiatry 20070501 |
| Exaggerated 5-HT1A but normal 5-HT2A receptor activity in individuals ill with anorexia nervosa. | Biological psychiatry 20070501 |
| F15063, a compound with D2/D3 antagonist, 5-HT 1A agonist and D4 partial agonist properties. II. Activity in models of positive symptoms of schizophrenia. | British journal of pharmacology 20070501 |
| Antidepressant-like effects of Albizzia julibrissin in mice: involvement of the 5-HT1A receptor system. | Pharmacology, biochemistry, and behavior 20070501 |
| Involvement of 5-HT1A and GABAA receptors in the anxiolytic-like effects of Cinnamomum cassia in mice. | Pharmacology, biochemistry, and behavior 20070501 |
| 8-Hydroxy-2-(di-n-propylamino)-tetralin inhibits food intake in fasted rats by an action at 5-HT1A receptors. | Methods and findings in experimental and clinical pharmacology 20070501 |
| 5-HT2A serotoninergic receptor in the locus coeruleus participates in the first phase of lipopolysaccharide-induced fever. | Canadian journal of physiology and pharmacology 20070501 |
| Role of peripheral 5-HT1A receptors in detrusor over activity associated with partial bladder outlet obstruction in female rats. | European journal of pharmacology 20070430 |
| Changes in the firing activity of serotonergic neurons in the dorsal raphe nucleus in a rat model of Parkinson's disease. | Sheng li xue bao : [Acta physiologica Sinica] 20070425 |
| Anti-anxiety effects of Apocynum venetum L. in the elevated plus maze test. | Journal of ethnopharmacology 20070404 |
| Serotonin receptor involvement in effects of restraint on female rat lordosis behavior. | Pharmacology, biochemistry, and behavior 20070401 |
| Role of postsynaptic serotonin1A receptors in risperidone-induced increase in acetylcholine release in rat prefrontal cortex. | European journal of pharmacology 20070322 |
| The effects of 8-hydroxy-2-(di-n-propylamino)-tetralin (8-OH-DPAT) on food intake in non-deprived C57BL6 mice. | European journal of pharmacology 20070322 |
| Serotonergic drugs and spinal cord transections indicate that different spinal circuits are involved in external urethral sphincter activity in rats. | American journal of physiology. Renal physiology 20070301 |
| Single exposure to a serotonin 1A receptor agonist, (+)8-hydroxy-2-(di-n-propylamino)-tetralin, produces a prolonged heterologous desensitization of serotonin 2A receptors in neuroendocrine neurons in vivo. | The Journal of pharmacology and experimental therapeutics 20070301 |
| Native rat hippocampal 5-HT1A receptors show constitutive activity. | Molecular pharmacology 20070301 |
| Serotonin 5-HT1A receptor stimulates c-Jun N-terminal kinase and induces apoptosis in Chinese hamster ovary fibroblasts. | Biochimica et biophysica acta 20070301 |
| Effects of the reference tissue setting on the parametric image of 11C-WAY 100635. | Nuclear medicine communications 20070301 |
| Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach. | Biological & pharmaceutical bulletin 20070301 |
| 3,4-Dihydro-2H-benzoxazinones as dual-acting 5-HT1A receptor antagonists and serotonin reuptake inhibitors. | Bioorganic & medicinal chemistry letters 20070215 |
| Screening of 5-HT1A receptor antagonists using molecularly imprinted polymers. | Journal of the American Chemical Society 20070214 |
| Acetaminophen recruits spinal p42/p44 MAPKs and GH/IGF-1 receptors to produce analgesia via the serotonergic system. | Molecular pharmacology 20070201 |
| Effects of metabotropic glutamate 2/3 receptor antagonists in the stress-induced hyperthermia test in singly housed mice. | Psychopharmacology 20070201 |
| 5-HT1A receptors are involved in the anxiolytic effect of Delta9-tetrahydrocannabinol and AM 404, the anandamide transport inhibitor, in Sprague-Dawley rats. | European journal of pharmacology 20070126 |
| 5-HT1A receptor activation counteracted the effect of acute immobilization of noradrenergic neurons in the rat locus coeruleus. | Neuroscience letters 20070122 |
| Desensitization of 5-HT(1A) autoreceptors induced by neonatal DSP-4 treatment. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20070115 |
| Cellular and behavioral effects of 5-HT1A receptor agonist 8-OH-DPAT in a rat model of levodopa-induced motor complications. | Brain research 20070105 |
| Effects of OPC-14523, a combined sigma and 5-HT1a ligand, on pre- and post-synaptic 5-HT1a receptors. | Journal of psychopharmacology (Oxford, England) 20070101 |
| Changes in central 5-HT(1A) receptor binding in mesial temporal epilepsy measured by positron emission tomography with [(11)C]WAY100635. | Epilepsy research 20070101 |
| Effects of serotonin on the intrinsic membrane properties of layer II medial entorhinal cortex neurons. | Hippocampus 20070101 |
| Neurochemical identification of stereotypic burst-firing neurons in the rat dorsal raphe nucleus using juxtacellular labelling methods. | The European journal of neuroscience 20070101 |
| Antidepressant-like effect of leptin in streptozotocin-induced diabetic mice. | Pharmacology, biochemistry, and behavior 20070101 |
| 5-HT1A receptor agonist properties of antipsychotics determined by [35S]GTPgammaS binding in rat hippocampal membranes. | Clinical and experimental pharmacology & physiology 20070101 |
| Serotonin decreases aggression via 5-HT1A receptors in the fighting fish Betta splendens. | Pharmacology, biochemistry, and behavior 20070101 |
| The partial 5-HT(1A) agonist buspirone reduces the expression and development of l-DOPA-induced dyskinesia in rats and improves l-DOPA efficacy. | Pharmacology, biochemistry, and behavior 20070101 |
| Effects of repetitive administration of tianeptine, zinc hydroaspartate and electroconvulsive shock on the reactivity of 5-HT(7) receptors in rat hippocampus. | Pharmacological reports : PR 20070101 |
| Antidepressant-like effect of combined treatment with selective sigma receptor agonists and a 5-HT1A receptor agonist in the forced swimming test in rats. | Pharmacological reports : PR 20070101 |
| Zimelidine decreases seizure susceptibility in stressed mice. | Journal of neural transmission (Vienna, Austria : 1996) 20061201 |
| Quantification of serotonin 5-HT1A receptors in monkey brain with [11C](R)-(-)-RWAY. | Synapse (New York, N.Y.) 20061201 |
| Serotonin 1A receptor availability in patients with schizophrenia and schizo-affective disorder: a positron emission tomography imaging study with [11C]WAY 100635. | Psychopharmacology 20061201 |
| In 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine-treated primates, the selective 5-hydroxytryptamine 1a agonist (R)-(+)-8-OHDPAT inhibits levodopa-induced dyskinesia but only with\ increased motor disability. | The Journal of pharmacology and experimental therapeutics 20061201 |
| In vivo evidence that 5-HT(2C) receptors inhibit 5-HT neuronal activity via a GABAergic mechanism. | British journal of pharmacology 20061201 |
| A PET study of 5-HT1A receptors at different phases of the menstrual cycle in women with premenstrual dysphoria. | Psychiatry research 20061201 |
| Anxiolytic effects of the aqueous extract of Uncaria rhynchophylla. | Journal of ethnopharmacology 20061124 |
| Involvement of 5-hydroxytryptamine1A receptors in Delta9-tetrahydrocannabinol-induced catalepsy-like immobilization in mice. | European journal of pharmacology 20061121 |
| Systemic morphine produce antinociception mediated by spinal 5-HT7, but not 5-HT1A and 5-HT2 receptors in the spinal cord. | British journal of pharmacology 20061101 |
| Capacity for 5-HT1A-mediated autoregulation predicts amygdala reactivity. | Nature neuroscience 20061101 |
| Gender-dependent regulation of G-protein-gated inwardly rectifying potassium current in dorsal raphe neurons in knock-out mice devoid of the 5-hydroxytryptamine transporter. | Journal of neurobiology 20061101 |
| Role of serotonin type 1A receptors in fluvoxamine-induced inhibition of marble-burying behavior in mice. | Behavioural pharmacology 20061101 |
| Long-term effects of nicotine on the forced swimming test in mice: an experimental model for the study of depression caused by smoke. | Neurochemistry international 20061001 |
| A comparison of recent parametric neuroreceptor mapping approaches based on measurements with the high affinity PET radioligands [11C]FLB 457 and [11C]WAY 100635. | NeuroImage 20061001 |
| WAY-100635 is a potent dopamine D4 receptor agonist. | Psychopharmacology 20061001 |
| Synthesis and biologic evaluation of a novel serotonin 5-HT1A receptor radioligand, 18F-labeled mefway, in rodents and imaging by PET in a nonhuman primate. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20061001 |
| Tandospirone, a 5-HT1A agonist, ameliorates movement disorder via non-dopaminergic systems in rats with unilateral 6-hydroxydopamine-generated lesions. | Brain research 20060927 |
| Antipsychotic-like vs cataleptogenic actions in mice of novel antipsychotics having D2 antagonist and 5-HT1A agonist properties. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060901 |
| Actions of novel antipsychotic agents on apomorphine-induced PPI disruption: influence of combined serotonin 5-HT1A receptor activation and dopamine D2 receptor blockade. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060901 |
| Differential role of 5-HT1A and 5-HT1B receptors on the antinociceptive and antidepressant effect of tramadol in mice. | Psychopharmacology 20060901 |
| Significance of initial emotional state for neuroimmunomodulation in conditions of activation and blockade of 5-HT(1A) receptors. | Neuroscience and behavioral physiology 20060901 |
| Facilitating antidepressant-like actions of estrogens are mediated by 5-HT1A and estrogen receptors in the rat forced swimming test. | Psychoneuroendocrinology 20060901 |
| SB-699551-A (3-cyclopentyl-N-[2-(dimethylamino)ethyl]-N-[(4'-{[(2-phenylethyl)amino]methyl}-4-biphenylyl)methyl]propanamide dihydrochloride), a novel 5-ht5A receptor-selective antagonist, enhances 5-HT neuronal function: Evidence for an autoreceptor role for the 5-ht5A receptor in guinea pig brain. | Neuropharmacology 20060901 |
| Attenuation by the 5-HT1A receptor agonist osemozotan of the behavioral effects of single and repeated methamphetamine in mice. | Neuropharmacology 20060901 |
| Characteristics of binding of [3H]WAY100635 to rat hippocampal membranes. | Neurochemical research 20060901 |
| Activation of lumbosacral 5-HT2C receptors induces bursts of rhythmic activity in sympathetic nerves to the vas deferens in male rats. | British journal of pharmacology 20060801 |
| Adaptive changes in serotonin neurons of the raphe nuclei in 5-HT(4) receptor knock-out mouse. | The European journal of neuroscience 20060801 |
| Alteration of 5-HIAA levels in frontal cortex and dorsal raphe nucleus in rats treated with combined administration of tryptophan and ethanol. | The Journal of toxicological sciences 20060801 |
| Anticonvulsant effect of the selective 5-HT1B receptor agonist CP 94253 in mice. | European journal of pharmacology 20060710 |
| Roles of glutamatergic and serotonergic mechanisms in reflex control of the external urethral sphincter in urethane-anesthetized female rats. | American journal of physiology. Regulatory, integrative and comparative physiology 20060701 |
| In vitro and in vivo characterization of F-97013-GD, a partial 5-HT1A agonist with antipsychotic- and antiparkinsonian-like properties. | Neuropharmacology 20060701 |
| WAY-100635 antagonist-induced plasticity of 5-HT receptors: regulatory differences between a stable cell line and an in vivo native system. | Journal of neurochemistry 20060701 |
| Suppression of bladder reflex activity in chronic spinal cord injured cats by activation of serotonin 5-HT1A receptors. | Experimental neurology 20060601 |
| Synthesis and in vivo biodistribution of F-18 labeled 3-cis-, 3-trans-, 4-cis-, and 4-trans-fluorocyclohexane derivatives of WAY 100635. | Bioorganic & medicinal chemistry 20060601 |
| Early life blockade of 5-hydroxytryptamine 1A receptors normalizes sleep and depression-like behavior in adult knock-out mice lacking the serotonin transporter. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20060517 |
| Modulation of delta opioid-evoked hypothermia in rats by WAY 100635 and fluoxetine. | Neuroscience letters 20060508 |
| Activation of pyramidal cells in rat medial prefrontal cortex projecting to ventral tegmental area by a 5-HT1A receptor agonist. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20060501 |
| Clozapine modulates aromatic L-amino acid decarboxylase activity in mouse striatum. | The Journal of pharmacology and experimental therapeutics 20060501 |
| Repeated adolescent 3,4-methylenedioxymethamphetamine (MDMA) exposure in rats attenuates the effects of a subsequent challenge with MDMA or a 5-hydroxytryptamine(1A) receptor agonist. | The Journal of pharmacology and experimental therapeutics 20060501 |
| Development of 5-HT1A receptor radioligands to determine receptor density and changes in endogenous 5-HT. | Synapse (New York, N.Y.) 20060501 |
| MDMA and fenfluramine reduce L-DOPA-induced dyskinesia via indirect 5-HT1A receptor stimulation. | The European journal of neuroscience 20060501 |
| 5-HT1A receptor activation counteracts c-Fos immunoreactivity induced in serotonin neurons of the raphe nuclei after immobilization stress in the male rat. | Neuroscience letters 20060424 |
| Dissociable contribution of 5-HT1A and 5-HT2A receptors in the medial prefrontal cortex to different aspects of executive control such as impulsivity and compulsive perseveration in rats. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060401 |
| 5-HT receptor subtypes involved in the anxiogenic-like action and associated Fos response of acute fluoxetine treatment in rats. | Psychopharmacology 20060401 |
| Augmentation by citalopram of risperidone-induced monoamine release in rat prefrontal cortex. | Psychopharmacology 20060401 |
| 5-HT(1A) receptors in endogenous regulation of neuropathic hypersensitivity in the rat. | European journal of pharmacology 20060327 |
| Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat. | European journal of pharmacology 20060327 |
| Determination of metabolic stability of positron emission tomography tracers by LC-MS/MS: an example in WAY-100635 and two analogues. | Journal of pharmaceutical and biomedical analysis 20060303 |
| Effects of 8-OH-DPAT on hippocampal NADH fluorescence in vivo in anaesthetized rats. | Journal of neuroscience research 20060301 |
| Emerging drugs for premature ejaculation. | Expert opinion on emerging drugs 20060301 |
| Activation of 5-HT1A receptors in rostral medullary raphé inhibits cutaneous vasoconstriction elicited by cold exposure in rabbits. | Brain research 20060216 |
| Participation of the 5-HT1A receptor in the antidepressant-like effect of estrogens in the forced swimming test. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060201 |
| Selective serotonin re-uptake inhibition attenuates evoked glutamate release in the dorsal horn of the anaesthetised rat in vivo. | Pharmacological research 20060201 |
| The 5-HT(1A) receptor agonist 8-OH-DPAT prevents prefrontocortical glutamate and serotonin release in response to blockade of cortical NMDA receptors. | Journal of neurochemistry 20060201 |
| Anxiolytic-like effects of Gastrodia elata and its phenolic constituents in mice. | Biological & pharmaceutical bulletin 20060201 |
| Investigation of mechanisms mediating 8-OH-DPAT-induced impairment of spatial memory: involvement of 5-HT1A receptors in the dorsal hippocampus in rats. | Brain research 20060119 |
| Altered serotonin 1A binding in major depression: a [carbonyl-C-11]WAY100635 positron emission tomography study. | Biological psychiatry 20060115 |
| Synthesis and in vivo validation of [O-methyl-11C]2-{4-[4-(7-methoxynaphthalen-1-yl)piperazin- 1-yl]butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione: a novel 5-HT1A receptor agonist positron emission tomography ligand. | Journal of medicinal chemistry 20060112 |
| Light/dark cycle manipulation influences mice behaviour in the elevated plus maze. | Behavioural brain research 20060106 |
| Serotonin1A autoreceptor activation by S 15535 enhances circadian activity rhythms in hamsters: evaluation of potential interactions with serotonin2A and serotonin2C receptors. | Neuroscience 20060101 |
| 5-HT1a receptor antagonists block perforant path-dentate LTP induced in novel, but not familiar, environments. | Learning & memory (Cold Spring Harbor, N.Y.) 20060101 |
| Hallucinogen-like actions of 5-methoxy-N,N-diisopropyltryptamine in mice and rats. | Pharmacology, biochemistry, and behavior 20060101 |
| Activation of serotonergic 5-HT(1A) receptors in the lateral parabrachial nucleus increases NaCl intake. | Brain research 20051220 |
| Stimulation of 5-HT 1A receptors increases the seizure threshold for picrotoxin in mice. | European journal of pharmacology 20051219 |
| Brain serotonin1A receptor binding in major depression is related to psychic and somatic anxiety. | Biological psychiatry 20051215 |
| Effects of novel antipsychotics with mixed D(2) antagonist/5-HT(1A) agonist properties on PCP-induced social interaction deficits in the rat. | Neuropharmacology 20051201 |
| 5-HT(1A) and 5-HT(2A) receptors in the rat dorsal periaqueductal gray mediate the antipanic-like effect induced by the stimulation of serotonergic neurons in the dorsal raphe nucleus. | Psychopharmacology 20051201 |
| Roles of extracellular signal-regulated kinase and Akt signaling in coordinating nuclear transcription factor-kappaB-dependent cell survival after serotonin 1A receptor activation. | Journal of neurochemistry 20051201 |
| Single-unit responses of serotonergic medullary raphe neurons to cardiovascular challenges in freely moving cats. | The European journal of neuroscience 20051201 |
| Anxiolytic- and antidepressant-like profiles of the galanin-3 receptor (Gal3) antagonists SNAP 37889 and SNAP 398299. | Proceedings of the National Academy of Sciences of the United States of America 20051129 |
| Repeated administration of citalopram and imipramine alters the responsiveness of rat hippocampal circuitry to the activation of 5-HT7 receptors. | European journal of pharmacology 20051107 |
| Harmane inhibits serotonergic dorsal raphe neurons in the rat. | Psychopharmacology 20051101 |
| Differential effects of simultaneous or sequential administration of paroxetine and WAY-100,635 on ejaculatory behavior. | Pharmacology, biochemistry, and behavior 20051101 |
| The novel analgesic, F 13640, produces intra- and postoperative analgesia in a rat model of surgical pain. | European journal of pharmacology 20051031 |
| Co-administration of fluoxetine and WAY100635 improves short-term memory function. | European journal of pharmacology 20051017 |
| 5-HT1A receptor-mediated G protein activation assessed by [35S]GTPgammaS binding in rat cerebral cortex. | European journal of pharmacology 20051003 |
| Differential effects of the 5-hydroxytryptamine (5-HT)1A receptor inverse agonists Rec 27/0224 and Rec 27/0074 on electrophysiological responses to 5-HT1A receptor activation in rat dorsal raphe nucleus and hippocampus in vitro. | The Journal of pharmacology and experimental therapeutics 20051001 |
| Contrasting contribution of 5-hydroxytryptamine 1A receptor activation to neurochemical profile of novel antipsychotics: frontocortical dopamine and hippocampal serotonin release in rat brain. | The Journal of pharmacology and experimental therapeutics 20051001 |
| The 5-HT1A receptor and the stimulus effects of LSD in the rat. | Psychopharmacology 20051001 |
| No interruption of lactation is needed after (11)C-WAY 100635 or (11)C-raclopride PET. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20051001 |
| Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter (SERT) and 5-HT(1A) receptor. | The Journal of pharmacy and pharmacology 20051001 |
| Antidepressant-like effect of coadministration of sulpiride and fluvoxamine in mice. | European journal of pharmacology 20050927 |
| Inhibition of serotonergic neurons in the nucleus paragigantocellularis lateralis fragments sleep and decreases rapid eye movement sleep in the piglet: implications for sudden infant death syndrome. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20050907 |
| 5-HT1A receptor expression during memory formation. | Psychopharmacology 20050901 |
| Pronociceptive role of peripheral and spinal 5-HT7 receptors in the formalin test. | Pain 20050901 |
| Altered brain serotonin 5-HT1A receptor binding after recovery from anorexia nervosa measured by positron emission tomography and [carbonyl11C]WAY-100635. | Archives of general psychiatry 20050901 |
| Effects of the potential 5-HT7 receptor agonist AS 19 in an autoshaping learning task. | Behavioural brain research 20050830 |
| Differential autoinhibition of 5-hydroxytryptamine neurons by 5-hydroxytryptamine in the dorsal raphe nucleus. | Neuroreport 20050822 |
| Novel antipsychotic agents with 5-HT(1A) agonist properties: role of 5-HT(1A) receptor activation in attenuation of catalepsy induction in rats. | Neuropharmacology 20050801 |
| Serotonin 5-HT receptor blockade enhances Ca(2+)/calmodulin-dependent protein kinase II function and membrane expression of AMPA receptor subunits in the rat hippocampus: implications for memory formation. | Journal of neurochemistry 20050801 |
| Lithium differs from anticonvulsant mood stabilizers in prefrontal cortical and accumbal dopamine release: role of 5-HT(1A) receptor agonism. | Brain research 20050712 |
| In vitro profile of the antidepressant candidate OPC-14523 at rat and human 5-HT1A receptors. | European journal of pharmacology 20050711 |
| alpha(2)-Adrenoceptor involvement in the in vitro inhibitory effect of citalopram on a subpopulation of rat locus coeruleus neurons. | European journal of pharmacology 20050704 |
| Effect of vilazodone on 5-HT efflux and re-uptake in the guinea-pig dorsal raphe nucleus. | European journal of pharmacology 20050704 |
| Effects of acute and long-term administration of escitalopram and citalopram on serotonin neurotransmission: an in vivo electrophysiological study in rat brain. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050701 |
| Yohimbine disrupts prepulse inhibition in rats via action at 5-HT1A receptors, not alpha2-adrenoceptors. | Psychopharmacology 20050701 |
| Paroxetine is effective in desensitizing 5-HT1A receptor function in adult offspring exposed prenatally to cocaine. | Psychopharmacology 20050701 |
| Prenatal stress influences 8-OH-DPAT modulated startle responding and [3H]-8-OH-DPAT binding in rats. | Pharmacology, biochemistry, and behavior 20050701 |
| Activation of 5-hydroxytryptamine 1A receptors suppresses the cardiovascular response evoked from the dorsomedial hypothalamic nucleus. | Hypertension (Dallas, Tex. : 1979) 20050701 |
| A comparison of the effects of the 5HT1A antagonists MM-77 and WAY-100635 on the mouse isolated vasa deferentia. | Autonomic & autacoid pharmacology 20050701 |
| Enhanced serotonin response in the hippocampus of Galphaz protein knock-out mice. | Neuroreport 20050621 |
| Gender-specific 5-HT1A receptor changes in BrdU nuclear labeling patterns in neonatal dentate gyrus. | Brain research. Developmental brain research 20050609 |
| Serotonergic neurons in the median raphe nucleus regulate inhibitory avoidance but not escape behavior in the rat elevated T-maze test of anxiety. | Psychopharmacology 20050601 |
| The role of 5-HT in the impairment of thermoregulation observed in rats administered MDMA ('ecstasy') when housed at high ambient temperature. | Psychopharmacology 20050601 |
| 5-Hydroxytryptamine 1A receptors in the paraventricular nucleus of the hypothalamus mediate oxytocin and adrenocorticotropin hormone release and some behavioral components of the serotonin syndrome. | The Journal of pharmacology and experimental therapeutics 20050601 |
| Serotonin (1A) receptor involvement in acute 3,4-methylenedioxymethamphetamine (MDMA) facilitation of social interaction in the rat. | Progress in neuro-psychopharmacology & biological psychiatry 20050601 |
| Dopamine and serotonin modulate the onset of metamorphosis in the ascidian Phallusia mammillata. | Developmental biology 20050601 |
| Regional reductions in serotonin 1A receptor binding in juvenile myoclonic epilepsy. | Archives of neurology 20050601 |
| Differential effects of 5-HT2C receptor ligands on place conditioning and locomotor activity in rats. | European journal of pharmacology 20050516 |
| Clozapine, ziprasidone and aripiprazole but not haloperidol protect against kainic acid-induced lesion of the striatum in mice, in vivo: role of 5-HT1A receptor activation. | Brain research 20050510 |
| In vivo effects of local activation and blockade of 5-HT1B receptors on globus pallidus neuronal spiking. | Brain research 20050510 |
| Analysis of the role of 5-HT1A receptors in spatial and aversive learning in the rat. | Neuropharmacology 20050501 |
| The 5-HT1A receptor and recognition memory. Possible modulation of its behavioral effects by the nitrergic system. | Behavioural brain research 20050430 |
| Serotonin-induced enhancement of vasopressin and oxytocin secretion in rat neurohypophyseal tissue culture. | Regulatory peptides 20050415 |
| Differential effects of intra-midbrain raphe and systemic 8-OH-DPAT on VTA self-stimulation thresholds in rats. | Psychopharmacology 20050401 |
| Interactions between serotonin and dopamine in the control of impulsive choice in rats: therapeutic implications for impulse control disorders. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050401 |
| [11C]-WAY100635 PET demonstrates marked 5-HT1A receptor changes in sporadic ALS. | Brain : a journal of neurology 20050401 |
| Spinal 5-HT1A receptors differentially influence nociceptive processing according to the nature of the noxious stimulus in rats: effect of WAY-100635 on the antinociceptive activities of paracetamol, venlafaxine and 5-HT. | Pain 20050401 |
| Biodistribution and radiation dosimetry of 11C-WAY100,635 in humans. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20050401 |
| Role of 5-HT1A and 5-HT1B receptors in the antinociceptive effect of tramadol. | European journal of pharmacology 20050321 |
| Serotonin1A-receptor antagonism blocks psychostimulant properties of diethylpropion in marmosets (Callithrix penicillata). | European journal of pharmacology 20050321 |
| Selective modulation of Ca(2+) influx pathways by 5-HT regulates synaptic long-term plasticity in the hippocampus. | Brain research 20050310 |
| A functional genetic variation of the serotonin (5-HT) transporter affects 5-HT1A receptor binding in humans. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20050309 |
| Neurochemical evaluation of the novel 5-HT1A receptor partial agonist/serotonin reuptake inhibitor, vilazodone. | European journal of pharmacology 20050307 |
| A study of the brain structures involved in the acute effects of fluoxetine on REM sleep in the rat. | The international journal of neuropsychopharmacology 20050301 |
| Dopamine uptake inhibitor-induced rotation in 6-hydroxydopamine-lesioned rats involves both D1 and D2 receptors but is modulated through 5-hydroxytryptamine and noradrenaline receptors. | The Journal of pharmacology and experimental therapeutics 20050301 |
| Role of 5-HT1A and 5-HT1B receptors in the hypophagic effect of 5-HT on the structure of feeding behavior. | Medical science monitor : international medical journal of experimental and clinical research 20050301 |
| Citalopram combined with WAY 100635 inhibits ejaculation and ejaculation-related Fos immunoreactivity. | European journal of pharmacology 20050210 |
| Evidence that the 5-HT1A autoreceptor is an important pharmacological target for the modulation of cocaine behavioral stimulant effects. | Brain research 20050209 |
| Anticataleptic properties of alpha2 adrenergic antagonists in the crossed leg position and bar tests: differential mediation by 5-HT1A receptor activation. | Psychopharmacology 20050201 |
| Partial 5-HT(1A) receptor agonist activity by the 5-HT(2C) receptor antagonist SB 206,553 is revealed in rats spinalized as neonates. | Experimental neurology 20050201 |
| N-oxide analogs of WAY-100635: new high affinity 5-HT(1A) receptor antagonists. | Bioorganic & medicinal chemistry 20050201 |
| Activation of 5-HT1A and 5-HT7 receptors in the parafascicular nucleus suppresses the affective reaction of rats to noxious stimulation. | Pain 20050201 |
| Brain 5-HT1A receptor binding in chronic fatigue syndrome measured using positron emission tomography and [11C]WAY-100635. | Biological psychiatry 20050201 |
| In-vivo effects of the 1,2,4-piperazine derivatives MM5 and MC1, putative 5-HT agonists, on dopamine and serotonin release in rat prefrontal cortex. | The Journal of pharmacy and pharmacology 20050201 |
| Somatodendritic autoreceptor regulation of serotonergic neurons: dependence on L-tryptophan and tryptophan hydroxylase-activating kinases. | The European journal of neuroscience 20050201 |
| Membrane receptors involved in modulation of responses of spinal dorsal horn interneurons evoked by feline group II muscle afferents. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20050119 |
| Effects of GABA(B), 5-HT(1A), and 5-HT(2) receptor stimulation on activation and inhibition of the rat lateral amygdala following medial geniculate nucleus stimulation in vivo. | Brain research 20050107 |
| Modulation of the activity of pyramidal neurons in rat prefrontal cortex by raphe stimulation in vivo: involvement of serotonin and GABA. | Cerebral cortex (New York, N.Y. : 1991) 20050101 |
| Sulpiride in combination with fluvoxamine increases in vivo dopamine release selectively in rat prefrontal cortex. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050101 |
| Autoradiographic characterisation of [35S]GTPgammaS binding stimulation mediated by 5-HT1B receptor in postmortem human brain. | Neuropharmacology 20050101 |
| Tandospirone activates neuroendocrine and ERK (MAP kinase) signaling pathways specifically through 5-HT1A receptor mechanisms in vivo. | Naunyn-Schmiedeberg's archives of pharmacology 20050101 |
| [Activation and blocking of 5-HT1A receptors influence on the immune response in CBA mice]. | Eksperimental'naia i klinicheskaia farmakologiia 20050101 |
| Two C-methyl derivatives of [11C]WAY-100635--effects of an amido alpha-methyl group on metabolism and brain 5-HT1A receptor radioligand behavior in monkey. | Molecular imaging and biology : MIB : the official publication of the Academy of Molecular Imaging 20050101 |
| [Significance of initial emotional state for neuroimmunomodulation under conditions of activation or blockade of 5-HT1A receptors]. | Zhurnal vysshei nervnoi deiatelnosti imeni I P Pavlova 20050101 |
| A review of the neuroprotective properties of the 5-HT1A receptor agonist repinotan HCl (BAYx3702) in ischemic stroke. | CNS drug reviews 20050101 |
| The 5HT1A receptor agonist, 8-OH-DPAT, protects neurons and reduces astroglial reaction after ischemic damage caused by cortical devascularization. | Brain research 20041231 |
| 5-HT activates ERK MAP kinase in cultured-human peripheral blood mononuclear cells via 5-HT1A receptors. | Life sciences 20041210 |
| Effects of the 5-HT7 receptor antagonists SB-269970 and DR 4004 in autoshaping Pavlovian/instrumental learning task. | Behavioural brain research 20041206 |
| Role of hippocampal CaMKII in serotonin 5-HT(1A) receptor-mediated learning deficit in rats. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20041201 |
| Serotonin 1A receptor binding and treatment response in late-life depression. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20041201 |
| Anticonvulsant action of GBR-12909 and citalopram against acute experimentally induced limbic seizures. | Neuropharmacology 20041201 |
| Acute effect of milnacipran on the relationship between the locus coeruleus noradrenergic and dorsal raphe serotonergic neuronal transmitters. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20041201 |
| 5-HT1A receptors are differentially involved in the anxiolytic- and antidepressant-like effects of 8-OH-DPAT and fluoxetine in the rat. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20041201 |
| Facilitatory effects of WAY-100635, a 5-HT1A receptor antagonist, on lordosis in female rats. | Neuroscience letters 20041123 |
| Effects of fenfluramine on free-operant timing behaviour: evidence for involvement of 5-HT2A receptors. | Psychopharmacology 20041101 |
| Endogenously released 5-hydroxytryptamine depresses the spinal monosynaptic reflex via 5-HT1D receptors. | European journal of pharmacology 20041025 |
| Combined treatment of quetiapine with haloperidol in animal models of antipsychotic effect and extrapyramidal side effects: comparison with risperidone and chlorpromazine. | Psychopharmacology 20041001 |
| Electrophysiological evidence for the tonic activation of 5-HT(1A) autoreceptors in the rat dorsal raphe nucleus. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20041001 |
| Positron emission tomographic evaluation of the putative dopamine-D3 receptor ligand, [11C]RGH-1756 in the monkey brain. | Neurochemistry international 20041001 |
| Intracerebroventricular injection of trazodone produces 5-HT receptor subtype mediated anti-nociception at the supraspinal and spinal levels. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20041001 |
| Regulators of G-protein signaling 4: modulation of 5-HT1A-mediated neurotransmitter release in vivo. | Brain research 20041001 |
| Cloned human 5-HT1A receptor pharmacology determined using agonist binding and measurement of cAMP accumulation. | The Journal of pharmacy and pharmacology 20041001 |
| Involvement of 5-HT1B receptors within the ventral tegmental area in regulation of mesolimbic dopaminergic neuronal activity via GABA mechanisms: a study with dual-probe microdialysis. | Brain research 20040917 |
| Preferential 5-HT1A autoreceptor occupancy by pindolol is attenuated in depressed patients: effect of treatment or an endophenotype of depression? | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040901 |
| Inhibition of bladder activity by 5-hydroxytryptamine1 serotonin receptor agonists in cats with chronic spinal cord injury. | The Journal of pharmacology and experimental therapeutics 20040901 |
| A positron emission tomography study of the 5-HT1A receptor in schizophrenia and during clozapine treatment. | Journal of psychopharmacology (Oxford, England) 20040901 |
| A 5-HT7 heteroreceptor-mediated inhibition of [3H]serotonin release in raphe nuclei slices of the rat: evidence for a serotonergic-glutamatergic interaction. | Neurochemical research 20040801 |
| Studies toward the discovery of the next generation of antidepressants. 3. Dual 5-HT1A and serotonin transporter affinity within a class of N-aryloxyethylindolylalkylamines. | Journal of medicinal chemistry 20040715 |
| WAY100635 and female rat lordosis behavior. | Brain research 20040709 |
| Toward brain imaging of serotonin 5-HT1A autoreceptor internalization. | NeuroImage 20040701 |
| Failure of repeated electroconvulsive shock treatment on 5-HT4-receptor-mediated depolarization due to protein kinase A system in young rat hippocampal CA1 neurons. | Journal of pharmacological sciences 20040701 |
| Perospirone, a novel atypical antipsychotic drug, potentiates fluoxetine-induced increases in dopamine levels via multireceptor actions in the rat medial prefrontal cortex. | Neuroscience letters 20040624 |
| Aripiprazole, a novel antipsychotic drug, preferentially increases dopamine release in the prefrontal cortex and hippocampus in rat brain. | European journal of pharmacology 20040616 |
| Acute treatment with the antidepressant fluoxetine internalizes 5-HT1A autoreceptors and reduces the in vivo binding of the PET radioligand [18F]MPPF in the nucleus raphe dorsalis of rat. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20040609 |
| Role of spinal 5-HT(1A) receptors in morphine analgesia and tolerance in rats. | European journal of pain (London, England) 20040601 |
| 5-HT1A receptor activation before acute stress counteracted the induced long-term behavioral effects. | Annals of the New York Academy of Sciences 20040601 |
| Blockade of supraspinal 5-HT1A receptors potentiates the inhibitory effect of venlafaxine on wind-up activity in mononeuropathic rats. | Brain research 20040522 |
| Dissociation of rewarding and dopamine transporter-mediated properties of amphetamine. | Proceedings of the National Academy of Sciences of the United States of America 20040518 |
| Effects of the 5-HT1A receptor ligands flesinoxan and WAY 100635 given systemically or microinjected into the laterodorsal tegmental nucleus on REM sleep in the rat. | Behavioural brain research 20040505 |
| Occupancy of agonist drugs at the 5-HT1A receptor. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040501 |
| Anticonvulsant action of hippocampal dopamine and serotonin is independently mediated by D and 5-HT receptors. | Journal of neurochemistry 20040501 |
| Mirtazapine increases dopamine release in prefrontal cortex by 5-HT1A receptor activation. | Brain research bulletin 20040430 |
| Limbic reductions of 5-HT1A receptor binding in human temporal lobe epilepsy. | Neurology 20040427 |
| Brain serotonin 1A receptor binding in bulimia nervosa. | Biological psychiatry 20040415 |
| Pharmacological studies of 8-OH-DPAT-induced pupillary dilation in anesthetized rats. | European journal of pharmacology 20040412 |
| Effects of nociceptin on the exploratory behavior of mice in the hole-board test. | European journal of pharmacology 20040405 |
| Aripiprazole (OPC-14597) fully substitutes for the 5-HT1A receptor agonist LY293284 in the drug discrimination assay in rats. | Psychopharmacology 20040401 |
| Effects of acute and chronic buspirone on impulsive choice and efflux of 5-HT and dopamine in hippocampus, nucleus accumbens and prefrontal cortex. | Psychopharmacology 20040401 |
| Persistent reduction in brain serotonin1A receptor binding in recovered depressed men measured by positron emission tomography with [11C]WAY-100635. | Molecular psychiatry 20040401 |
| Effect of combined administration of 5-HT1A or 5-HT1B/1D receptor antagonists and antidepressants in the forced swimming test. | European journal of pharmacology 20040308 |
| Decreased 5-HT1A receptor binding in amygdala of schizophrenia. | Biological psychiatry 20040301 |
| 5-Hydroxytryptamine 1B receptors mediate presynaptic inhibition of monosynaptic IPSC in the rat dorsolateral septal nucleus. | Neuroscience research 20040301 |
| Chronic fluoxetine-induced desensitization of 5-HT1A and 5-HT1B autoreceptors: regional differences and effects of WAY-100635. | European journal of pharmacology 20040213 |
| Further characterization of the 5-HT1 receptors mediating cardiac sympatho-inhibition in pithed rats: pharmacological correlation with the 5-HT1B and 5-HT1D subtypes. | Naunyn-Schmiedeberg's archives of pharmacology 20040201 |
| Differential autoreceptor control of extracellular 5-HT in guinea pig and rat: species and regional differences. | Psychopharmacology 20040201 |
| Involvement of 5-HT1A receptors in behavioural effects of the cannabinoid receptor agonist CP 55,940 in male rats. | Behavioural pharmacology 20040201 |
| 5-HT1A-mediated promotion of mitogen-activated T and B cell survival and proliferation is associated with increased translocation of NF-kappaB to the nucleus. | Brain, behavior, and immunity 20040101 |
| OS-EM and FBP reconstructions at low count rates: effect on 3D PET studies of [11C] WAY-100635. | NeuroImage 20040101 |
| The pyridinyl-6 position of WAY-100635 as a site for radiofluorination--effect on 5-HT1A receptor radioligand behavior in vivo. | Molecular imaging and biology : MIB : the official publication of the Academy of Molecular Imaging 20040101 |
| Endogenous 5-HT inhibits firing activity of hippocampal CA1 pyramidal neurons during conditioned fear stress-induced freezing behavior through stimulating 5-HT1A receptors. | Hippocampus 20040101 |
| The hypotensive effect of BMY 7378 involves central 5-HT1A receptor stimulation in the adult but not in the young rat. | Archives of medical research 20040101 |
| Direct activation by dopamine of recombinant human 5-HT1A receptors: comparison with human 5-HT2C and 5-HT3 receptors. | Synapse (New York, N.Y.) 20031215 |
| Anxiolytic-like effects of the selective 5-HT1A receptor antagonist WAY 100635 in non-human primates. | European journal of pharmacology 20031215 |
| 5-HT7 receptors increase the excitability of rat hippocampal CA1 pyramidal neurons. | Brain research 20031212 |
| SSR181507, a dopamine D(2) receptor antagonist and 5-HT(1A) receptor agonist. I: Neurochemical and electrophysiological profile. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20031201 |
| Mice lacking the serotonin transporter exhibit 5-HT(1A) receptor-mediated abnormalities in tests for anxiety-like behavior. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20031201 |
| Sensitization of adenylate cyclase by short-term activation of 5-HT1A receptors. | Cellular signalling 20031201 |
| The serotonergic system may be involved in the sleep-inducing action of oleamide in rats. | Naunyn-Schmiedeberg's archives of pharmacology 20031201 |
| Determination of volume of distribution using likelihood estimation in graphical analysis: elimination of estimation bias. | Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20031201 |
| 5-HT2C receptors inhibit and 5-HT1A receptors activate the generation of spike-wave discharges in a genetic rat model of absence epilepsy. | Experimental neurology 20031201 |
| LABORAS: Initial pharmacological validation of a system allowing continuous monitoring of laboratory rodent behaviour. | Journal of neuroscience methods 20031130 |
| Lack of effect of a single dose of hydrocortisone on serotonin(1A) receptors in recovered depressed patients measured by positron emission tomography with [11C]WAY-100635. | Biological psychiatry 20031101 |
| The serotonin system and spiritual experiences. | The American journal of psychiatry 20031101 |
| The 5-HT1A receptor agonist MKC-242 reverses isolation rearing-induced deficits of prepulse inhibition in mice. | Psychopharmacology 20031001 |
| 5-Hydroxytryptamine 1A receptors inhibit cold-induced sympathetically mediated cutaneous vasoconstriction in rabbits. | The Journal of physiology 20031001 |
| Pharmacological profile of the 5-HT-induced inhibition of cardioaccelerator sympathetic outflow in pithed rats: correlation with 5-HT1 and putative 5-ht5A/5B receptors. | British journal of pharmacology 20031001 |
| Sex hormone-dependent desensitization of 5-HT1A autoreceptors in knockout mice deficient in the 5-HT transporter. | The European journal of neuroscience 20031001 |
| Orienting and defensive behaviors elicited by superior colliculus stimulation in rats: effects of 5-HT depletion, uptake inhibition, and direct midbrain or frontal cortex application. | Behavioural brain research 20030915 |
| The 5-HT 1A receptor antagonist WAY 100635 improves rats performance in different models of amnesia evaluated by the object recognition task. | Brain research 20030905 |
| Cerebrospinal fluid monoamine and metabolite concentrations and aggression in rats. | Hormones and behavior 20030901 |
| Suppression of the micturition reflex in urethane-anesthetized rats by intracerebroventricular injection of WAY100635, a 5-HT(1A) receptor antagonist. | Brain research 20030808 |
| Flibanserin, a potential antidepressant drug, lowers 5-HT and raises dopamine and noradrenaline in the rat prefrontal cortex dialysate: role of 5-HT(1A) receptors. | British journal of pharmacology 20030801 |
| Responses to serotonin (5HT) in isolated corpus cavernosum penis of rabbit. | International journal of impotence research 20030801 |
| Activation of post-synaptic 5-HT(1A) receptors in the dorsal hippocampus prevents learned helplessness development. | Brain research 20030718 |
| Synthesis of a [6-pyridinyl-18F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT1A receptor imaging with PET. | Bioorganic & medicinal chemistry 20030703 |
| Effects of chronic paroxetine treatment on dialysate serotonin in 5-HT1B receptor knockout mice. | Journal of neurochemistry 20030701 |
| Do different mechanisms underlie two anxiogenic effects of systemic nicotine? | Behavioural pharmacology 20030701 |
| Involvement of presynaptic 5-HT(1A) and benzodiazepine receptors in the anticonflict activity of 5-HT(1A) receptor antagonists. | European journal of pharmacology 20030613 |
| The novel analgesic and high-efficacy 5-HT1A receptor agonist, F 13640 induces c-Fos protein expression in spinal cord dorsal horn neurons. | Brain research 20030606 |
| A 5-HT1A agonist and a 5-HT2c antagonist reduce social interaction deficit induced by multiple ethanol withdrawals in rats. | Psychopharmacology 20030601 |
| Mutation in a protein kinase C phosphorylation site of the 5-HT1A receptor preferentially attenuates Ca2+ responses to partial as opposed to higher-efficacy 5-HT1A agonists. | Neuropharmacology 20030601 |
| Effect of different 5-HT1A receptor antagonists in combination with paroxetine on expression of the immediate-early gene Arc in rat brain. | Neuropharmacology 20030601 |
| Use of Arc expression as a molecular marker of increased postsynaptic 5-HT function after SSRI/5-HT1A receptor antagonist co-administration. | Journal of neurochemistry 20030601 |
| Administration of the 5-hydroxytryptamine(1A) receptor antagonist WAY100635 suppresses acute experimental allergic encephalomyelitis in Lewis rats. | Neuroscience letters 20030515 |
| Effects of 8-OH-DPAT and WAY-100635 on performance on a time-constrained progressive-ratio schedule. | Psychopharmacology 20030501 |
| 5-HT1A agonists: alcohol drinking in rats and squirrel monkeys. | Psychopharmacology 20030501 |
| A comparison of the effects of loxapine with ziprasidone and thioridazine on the release of dopamine and acetylcholine in the prefrontal cortex and nucleus accumbens. | Psychopharmacology 20030501 |
| WAY-100635, an antagonist of 5-HT(1A) receptor, causes malformations of the CNS in ascidian embryos. | Development genes and evolution 20030501 |
| Adaptive changes in the reactivity of 5-HT1A and 5-HT2 receptors induced in rat frontal cortex by repeated imipramine and citalopram. | Naunyn-Schmiedeberg's archives of pharmacology 20030501 |
| Serotonin upregulates the activity of phagocytosis through 5-HT1A receptors. | British journal of pharmacology 20030501 |
| Profound, non-opioid analgesia produced by the high-efficacy 5-HT(1A) agonist F 13640 in the formalin model of tonic nociceptive pain. | Pharmacology 20030401 |
| Reversal of visual attention dysfunction after AMPA lesions of the nucleus basalis magnocellularis (NBM) by the cholinesterase inhibitor donepezil and by a 5-HT1A receptor antagonist WAY 100635. | Psychopharmacology 20030401 |
| Positron emission tomographic analysis of dose-dependent NAD-299 binding to 5-hydroxytryptamine-1A receptors in the human brain. | Psychopharmacology 20030401 |
| Ambient temperature influences core body temperature response in rat lines bred for differences in sensitivity to 8-hydroxy-dipropylaminotetralin. | The Journal of pharmacology and experimental therapeutics 20030401 |
| Alpha2-adrenoreceptor activation inhibits LTP and LTD in the basolateral amygdala: involvement of Gi/o-protein-mediated modulation of Ca2+-channels and inwardly rectifying K+-channels in LTD. | The European journal of neuroscience 20030401 |
| Noradrenergic and serotonergic blockade inhibits BDNF mRNA activation following exercise and antidepressant. | Pharmacology, biochemistry, and behavior 20030401 |
| Pharmacological characterization of MP349, a novel 5-HT1A-receptor antagonist with anxiolytic-like activity, in mice and rats. | The Journal of pharmacy and pharmacology 20030401 |
| Occupancy of 5-HT1A receptors by clozapine in the primate brain: a PET study. | Psychopharmacology 20030301 |
| Age differences in the sensitivity to clomipramine in an animal model of obsessive-compulsive disorder. | Psychopharmacology 20030301 |
| 5-hydroxytryptamine 1A receptor activation protects against N-methyl-D-aspartate-induced apoptotic cell death in striatal and mesencephalic cultures. | The Journal of pharmacology and experimental therapeutics 20030301 |
| Tremor in Parkinson's disease and serotonergic dysfunction: an 11C-WAY 100635 PET study. | Neurology 20030225 |
| Discriminative stimulus properties of 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane [(+/-)DOI] in C57BL/6J mice. | Psychopharmacology 20030201 |
| Inhibitory effect of hippocampal 5-HT1A receptors on human explicit memory. | The American journal of psychiatry 20030201 |
| Selective 5-HT1A antagonists WAY 100635 and NAD-299 attenuate the impairment of passive avoidance caused by scopolamine in the rat. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20030201 |
| Activation of 5-HT(1A) autoreceptors enhances the inhibitory effect of galanin on hippocampal 5-HT release in vivo. | Neuropharmacology 20030201 |
| The 5-HT1A receptor agonist MKC-242 increases the exploratory activity of mice in the elevated plus-maze. | European journal of pharmacology 20030101 |
| Differential regulation of corticosteroid receptors by monoamine neurotransmitters and antidepressant drugs in primary hippocampal culture. | Neuroscience 20030101 |
| An in vitro assay for predicting successful imaging radiotracers. | Molecular imaging and biology : MIB : the official publication of the Academy of Molecular Imaging 20030101 |
| Molecular dynamics simulations of the ligand-induced chemical information transfer in the 5-HT(1A) receptor. | Journal of chemical information and computer sciences 20030101 |
| In vivo drug action of tandospirone at 5-HT1A receptor examined using positron emission tomography and neuroendocrine response. | Psychopharmacology 20021201 |
| Antagonism by WAY-100635 of the effects of 8-OH-DPAT on performance on a free-operant timing schedule in intact and 5-HT-depleted rats. | Behavioural pharmacology 20021201 |
| Comparison of the effects of antidepressants on norepinephrine and serotonin concentrations in the rat frontal cortex: an in-vivo microdialysis study. | Journal of psychopharmacology (Oxford, England) 20021201 |
| Effect of 5-HT1A receptor-mediated serotonin augmentation on Fos immunoreactivity in rat brain. | European journal of pharmacology 20021129 |
| Evidence that NAN-190-induced hypotension involves vascular alpha1-adrenoceptor antagonism in the rat. | European journal of pharmacology 20021122 |
| Effects of sex, age, and aggressive traits in man on brain serotonin 5-HT1A receptor binding potential measured by PET using [C-11]WAY-100635. | Brain research 20021108 |
| Modulation of reflexly evoked vagal bradycardias by central 5-HT1A receptors in anaesthetized rabbits. | British journal of pharmacology 20021101 |
| 5-HT1A receptor-mediated autoinhibition does not function at physiological firing rates: evidence from in vitro electrophysiological studies in the rat dorsal raphe nucleus. | Neuropharmacology 20021101 |
| 5-HT1A receptor activation and anti-cataleptic effects: high-efficacy agonists maximally inhibit haloperidol-induced catalepsy. | European journal of pharmacology 20021025 |
| 5-HT1A receptor-mediated regulation of mitogen-activated protein kinase phosphorylation in rat brain. | European journal of pharmacology 20021004 |
| Effects of sigma(1) receptor ligand MS-377 on D(2) antagonists-induced behaviors. | Pharmacology, biochemistry, and behavior 20021001 |
| Mechanisms of nicotine actions on dorsal raphe serotoninergic neurons. | European journal of pharmacology 20020927 |
| Antibody capture assay reveals bell-shaped concentration-response isotherms for h5-HT(1A) receptor-mediated Galpha(i3) activation: conformational selection by high-efficacy agonists, and relationship to trafficking of receptor signaling. | Molecular pharmacology 20020901 |
| Effects of long-term acetyl-L-carnitine administration in rats: I. increased dopamine output in mesocorticolimbic areas and protection toward acute stress exposure. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020901 |
| Evaluation of EMD 128 130 occupancy of the 5-HT1A and the D2 receptor: a human PET study with [11C]WAY-100635 and [11C]raclopride. | Journal of psychopharmacology (Oxford, England) 20020901 |
| Repeated administration of milnacipran induces rapid desensitization of somatodendritic 5-HT1A autoreceptors but not postsynaptic 5-HT1A receptors. | Journal of psychopharmacology (Oxford, England) 20020901 |
| The selective serotonin(1A)-receptor antagonist WAY 100635 blocks behavioral stimulating effects of cocaine but not ventral striatal dopamine increase. | Behavioural brain research 20020821 |
| The role of 5-HT(1A) receptors in control of lower urinary tract function in cats. | Brain research 20020816 |
| Cocaine increases serotonergic activity in the hippocampus and nucleus accumbens in vivo: 5-HT1a-receptor antagonism blocks behavioral but potentiates serotonergic activation. | Synapse (New York, N.Y.) 20020801 |
| Postsynaptic 5-HT(1A) receptors mediate an increase in locomotor activity in the monoamine-depleted rat. | Psychopharmacology 20020801 |
| Influence of forced swimming-induced stress on the anxiolytic-like effect of 5HT(1A) agents in mice. | Psychopharmacology 20020701 |
| Aging alters in a region-specific manner serotonin transporter sites and 5-HT(1A) receptor-G protein interactions in hamster brain. | Neuropharmacology 20020701 |
| 5-HT(1A) and 5-HT(2A) receptors minimally contribute to clozapine-induced acetylcholine release in rat medial prefrontal cortex. | Brain research 20020607 |
| 5-Hydroxytryptamine1A receptor occupancy by novel full antagonist 2-[4-[4-(7-chloro-2,3-dihydro-1,4-benzdioxyn-5-yl)-1-piperazinyl]butyl]-1,2-benzisothiazol-3-(2H)-one-1,1-dioxide: a[11C][O-methyl-3H]-N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridinyl)cyclohexanecarboxamide trihydrochloride (WAY-100635) positron emission tomography study in humans. | The Journal of pharmacology and experimental therapeutics 20020601 |
| Involvement of 5-HT1A receptors in homeostatic and stress-induced adaptive regulations of paradoxical sleep: studies in 5-HT1A knock-out mice. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20020601 |
| Brain serotonin 5-HT(1A) receptor binding in schizophrenia measured by positron emission tomography and [11C]WAY-100635. | Archives of general psychiatry 20020601 |
| Effect of chronic fluoxetine and WAY-100635 treatment on serotonergic neurotransmission in the frontal cortex. | Journal of psychopharmacology (Oxford, England) 20020601 |
| Evidence that the hypotensive effect of WAY 100635, a 5-HT1A receptor antagonist, is related to vascular alpha 1-adrenoceptor blockade in the adult rat. | Autonomic & autacoid pharmacology 20020601 |
| Extended action of MKC-242, a selective 5-HT(1A) receptor agonist, on light-induced Per gene expression in the suprachiasmatic nucleus in mice. | Journal of neuroscience research 20020515 |
| Behavioural and biochemical studies of citalopram and WAY 100635 in rat chronic mild stress model. | Pharmacology, biochemistry, and behavior 20020501 |
| Enhanced detection of receptor constitutive activity in the presence of regulators of G protein signaling: applications to the detection and analysis of inverse agonists and low-efficacy partial agonists. | Molecular pharmacology 20020501 |
| Synthesis, biological and autoradiographic evaluation of a novel Tc-99m radioligand derived from WAY 100635 with high affinity for the 5-HT(1A) receptor and the alpha1-adrenergic receptor. | Nuclear medicine and biology 20020501 |
| Synthesis and biological evaluation of technetium(III) mixed-ligand complexes with high affinity for the cerebral 5-HT(1A) receptor and the alpha1-adrenergic receptor. | Nuclear medicine and biology 20020501 |
| Modulation by 5-hT2A receptors of aggressive behavior in isolated mice. | Japanese journal of pharmacology 20020501 |
| Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
| 5-HT1A agonist/antagonist modification of cocaine stimulant effects: implications for cocaine mechanisms. | Behavioural brain research 20020415 |
| Tandospirone potentiates the fluoxetine-induced increases in extracellular dopamine via 5-HT(1A) receptors in the rat medial frontal cortex. | Neurochemistry international 20020401 |
| A database of [(11)C]WAY-100635 binding to 5-HT(1A) receptors in normal male volunteers: normative data and relationship to methodological, demographic, physiological, and behavioral variables. | NeuroImage 20020301 |
| The PET radioligand [carbonyl-(11)C]desmethyl-WAY-100635 binds to 5-HT(1A) receptors and provides a higher radioactive signal than [carbonyl-(11)C]WAY-100635 in the human brain. | Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20020301 |
| Anxiolytic-like effect of way-100635 microinfusions into the median (but not dorsal) raphe nucleus in mice exposed to the plus-maze: influence of prior test experience. | Brain research 20020222 |
| Effects of intra-hippocampal infusion of WAY-100635 on plus-maze behavior in mice. Influence of site of injection and prior test experience. | Brain research 20020208 |
| Increased REM sleep after intra-dorsal raphe nucleus injection of flesinoxan or 8-OHDPAT: prevention with WAY 100635. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20020201 |
| Electroencephalographic activation by fluoxetine in rats: role of 5-HT(1A) receptors and enhancement of concurrent acetylcholinesterase inhibitor treatment. | Neuropharmacology 20020201 |
| Improvement in the selectivity and metabolic stability of the serotonin 5-HT(1A) ligand, S 15535: a series of cis- and trans-2-(arylcycloalkylamine) 1-indanols. | Journal of medicinal chemistry 20020103 |
| Renal sympathoinhibition mediated by 5-HT(1A) receptors in the RVLM during severe hemorrhage in rats. | American journal of physiology. Regulatory, integrative and comparative physiology 20020101 |
| 5-HT7 receptors modulate synchronized network activity in rat hippocampus. | Neuropharmacology 20020101 |
| A competitive interaction model predicts the effect of WAY-100,635 on the time course of R-(+)-8-hydroxy-2-(di-n-propylamino)tetralin-induced hypothermia. | The Journal of pharmacology and experimental therapeutics 20020101 |
| 5-HT(1B) receptor knockout mice show no adaptive changes in 5-HT(1A) receptor function as measured telemetrically on body temperature and heart rate responses. | Brain research bulletin 20020101 |
| Effect of endogenous serotonin on the binding of the 5-hT1A PET ligand 18F-MPPF in the rat hippocampus: kinetic beta measurements combined with microdialysis. | Journal of neurochemistry 20020101 |
| Serotonergic modulation of respiratory motoneurons and interneurons in brainstem slices of perinatal rats. | Neuroscience 20020101 |
| Nad-299 antagonises 5-HT-stimulated and spiperone-inhibited [35S]GTPgammaS binding in cloned 5-HT1A receptors. | Journal of receptor and signal transduction research 20020101 |
| Serotonin (1A) receptor ligands act on norepinephrine neuron firing through excitatory amino acid and GABA(A) receptors: a microiontophoretic study in the rat locus coeruleus. | Synapse (New York, N.Y.) 20011215 |
| Effects of aging on 5-HT(1A) receptors and their functional response to 5-HT(1a) agonist in the living brain: PET study with [carbonyl-(11)C]WAY-100635 in conscious monkeys. | Synapse (New York, N.Y.) 20011215 |
| Functional and pharmacological characterization of the modulatory role of serotonin on the firing activity of locus coeruleus norepinephrine neurons. | Brain research 20011213 |
| Involvement of benzodiazepine binding sites in an antiaggressive effect by 5-HT(1A) receptor activation in isolated mice. | European journal of pharmacology 20011207 |
| Effects of the selective norepinephrine reuptake inhibitor reboxetine on norepinephrine and serotonin transmission in the rat hippocampus. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20011201 |
| Effects of standardized extracts of St. John's wort on the single-unit activity of serotonergic dorsal Raphe neurons in awake cats: comparisons with fluoxetine and sertraline. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20011201 |
| Anxiety-like effects induced by acute fluoxetine, sertraline or m-CPP treatment are reversed by pretreatment with the 5-HT2C receptor antagonist SB-242084 but not the 5-HT1A receptor antagonist WAY-100635. | The international journal of neuropsychopharmacology 20011201 |
| 5-HT receptor subtypes involved in the spinal antinociceptive effect of acetaminophen in rats. | European journal of pharmacology 20011130 |
| Cocaine and serotonin: a role for the 5-HT(1A) receptor site in the mediation of cocaine stimulant effects. | Behavioural brain research 20011129 |
| Serotonin 5-HT1A agonist improves motor complications in rodent and primate parkinsonian models. | Neurology 20011127 |
| Agonist-induced internalization of serotonin-1a receptors in the dorsal raphe nucleus (autoreceptors) but not hippocampus (heteroreceptors). | The Journal of neuroscience : the official journal of the Society for Neuroscience 20011101 |
| Effects of endogenous neurotransmitters on the in vivo binding of dopamine and 5-HT radiotracers in mice. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20011101 |
| The role of central 5-HT(1A) receptors in the control of B-fibre cardiac and bronchoconstrictor vagal preganglionic neurones in anaesthetized cats. | The Journal of physiology 20011101 |
| Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices. | Journal of neurochemistry 20011101 |
| 5-hydroxytryptamine (5-HT)1A autoreceptor adaptive changes in substance P (neurokinin 1) receptor knock-out mice mimic antidepressant-induced desensitization. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20011015 |
| Efficacy of antipsychotic agents at human 5-HT(1A) receptors determined by [3H]WAY100,635 binding affinity ratios: relationship to efficacy for G-protein activation. | European journal of pharmacology 20011005 |
| Protective effects of 5-HT1A receptor agonists against emotional changes produced by stress stimuli are related to their neuroendocrine effects. | British journal of pharmacology 20011001 |
| The role of 5-HT1B receptors in the regulation of serotonin cell firing and release in the rat brain. | Journal of neurochemistry 20011001 |
| Nicotine stimulation of dorsal raphe neurons: effects on laterodorsal and pedunculopontine neurons. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20011001 |
| Stimulation of 5-HT(1A) receptors in the dorsal raphe ameliorates the impairment of spatial learning caused by intrahippocampal 7-chloro-kynurenic acid in naive and pretrained rats. | Psychopharmacology 20011001 |
| Rectal antinociceptive properties of alverine citrate are linked to antagonism at the 5-HT1A receptor subtype. | The Journal of pharmacy and pharmacology 20011001 |
| Changes in rat cerebral blood volume due to modulation of the 5-HT(1A) receptor measured with susceptibility enhanced contrast MRI. | Brain research 20010921 |
| Genetic regulation of extracellular serotonin by 5-hydroxytryptamine(1A) and 5-hydroxytryptamine(1B) autoreceptors in different brain regions of the mouse. | The Journal of pharmacology and experimental therapeutics 20010901 |
| Regional patterns of compensation following genetic deletion of either 5-hydroxytryptamine(1A) or 5-hydroxytryptamine(1B) receptor in the mouse. | The Journal of pharmacology and experimental therapeutics 20010901 |
| Functional alteration of brain dopaminergic system in isolated aggressive mice. | Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology 20010901 |
| Inhibitory effects of tandospirone, a 5-HT1A agonist, on medial vestibular nucleus neurons responding to lateral roll tilt stimulation in rats. | Brain research 20010810 |
| Effect of 5-HT on binding of [(11)C] WAY 100635 to 5-HT(IA) receptors in rat brain, assessed using in vivo microdialysis nd PET after fenfluramine. | Synapse (New York, N.Y.) 20010801 |
| Inverse relationship between serotonin 5-HT(1A) receptor binding and anxiety: a [(11)C]WAY-100635 PET investigation in healthy volunteers. | The American journal of psychiatry 20010801 |
| In vivo evaluation of 4-[123I]iodo-N-[2[4-(6-trifluoromethyl-2-pyridinyl)-1-piperazinyl]ethyl]benzamide, a potential SPECT radioligand for the 5-HT1A receptor. | Nuclear medicine and biology 20010801 |
| DOI, a 5-HT2A/2C receptor agonist, attenuates clozapine-induced cortical dopamine release. | Brain research 20010713 |
| Agonist properties of pindolol at h5-HT1A receptors coupled to mitogen-activated protein kinase. | European journal of pharmacology 20010713 |
| Serotonin 5-HT1A receptor imaging in the human brain with positron-emission tomography: coordination and the standardization and dissemination of methodology. | Journal of clinical pharmacology 20010701 |
| SB-272183, a selective 5-HT(1A), 5-HT(1B) and 5-HT(1D) receptor antagonist in native tissue. | British journal of pharmacology 20010701 |
| Researching the antidepressant actions of Hypericum perforatum (St. John's wort) in animals and man. | Pharmacopsychiatry 20010701 |
| Interaction between 5-HT(1A) and 5-HT(1B) receptors: effects of 8-OH-DPAT-induced hypothermia in 5-HT(1B) receptor knockout mice. | European journal of pharmacology 20010615 |
| In the formalin model of tonic nociceptive pain, 8-OH-DPAT produces 5-HT1A receptor-mediated, behaviorally specific analgesia. | European journal of pharmacology 20010608 |
| WAY-100635, a specific 5-HT1A antagonist, can increase the responsiveness of the mammalian circadian pacemaker to photic stimuli. | Neuroscience letters 20010601 |
| Effects of selective 5-HT1A receptor antagonists on regional serotonin synthesis in the rat brain: an autoradiographic study with alpha-[14C]methyl-L-tryptophan. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20010601 |
| Different tonic regulation of neuronal activity in the rat dorsal raphe and medial prefrontal cortex via 5-HT(1A) receptors. | Neuroscience letters 20010525 |
| 5-HT1A receptor activation and antidepressant-like effects: F 13714 has high efficacy and marked antidepressant potential. | European journal of pharmacology 20010525 |
| In vivo binding properties of [carbonyl-11C]WAY-100635: effect of endogenous serotonin. | Synapse (New York, N.Y.) 20010501 |
| Serotonin 5-HT1A receptor binding potential declines with age as measured by [11C]WAY-100635 and PET. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010501 |
| Effects of WAY100635, a selective 5-HT1A-receptor antagonist on the micturition-reflex pathway in the rat. | American journal of physiology. Regulatory, integrative and comparative physiology 20010501 |
| Biochemical, electrophysiological and neurohormonal studies with B-20991, a selective 5-HT1A receptor agonist. | Pharmacology 20010501 |
| The differential effects of intravenously administered 8-OH-DPAT on operant food intake in satiated and food-deprived pigs are mediated by central 5-HT(1A) receptors. | Physiology & behavior 20010501 |
| Differential effect of serotonin 5-HT(1A) receptor antagonists on the secretion of corticotropin and prolactin. | Neuroendocrinology 20010501 |
| 1,2,5-Thiadiazole derivatives are potent and selective ligands at human 5-HT1A receptors. | Bioorganic & medicinal chemistry letters 20010423 |
| Activation of 5-HT(1B/1D) receptors in the mesolimbic dopamine system increases dopamine release from the nucleus accumbens: a microdialysis study. | European journal of pharmacology 20010420 |
| Role of 5-HT(1A) and 5-HT(1B) receptors in the mediation of behavior in the forced swim test in mice. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010401 |
| Sympathoinhibition from ventrolateral periaqueductal gray mediated by 5-HT(1A) receptors in the RVLM. | American journal of physiology. Regulatory, integrative and comparative physiology 20010401 |
| Stress-induced hyperthermia in the 5-HT(1A) receptor knockout mouse is normal. | Biological psychiatry 20010401 |
| Involvement of 5-HT1A and 5-HT1B receptors for citalopram-induced hypothermia in the rat. | Psychopharmacology 20010401 |
| Gender-specific aging effects on the serotonin 1A receptor. | Brain research 20010323 |
| Differential occupancy of somatodendritic and postsynaptic 5HT(1A) receptors by pindolol: a dose-occupancy study with [11C]WAY 100635 and positron emission tomography in humans. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010301 |
| Modifications of the serotonergic system in mice lacking serotonin transporters: an in vivo electrophysiological study. | The Journal of pharmacology and experimental therapeutics 20010301 |
| Potentiation of the antinociceptive effect of clomipramine by a 5-ht(1A) antagonist in neuropathic pain in rats. | British journal of pharmacology 20010301 |
| Activation of 5-HT(1A) but not 5-HT(1B) receptors attenuates an increase in extracellular dopamine derived from exogenously administered L-DOPA in the striatum with nigrostriatal denervation. | Journal of neurochemistry 20010301 |
| 5-HT(2A) and D(2) receptor blockade increases cortical DA release via 5-HT(1A) receptor activation: a possible mechanism of atypical antipsychotic-induced cortical dopamine release. | Journal of neurochemistry 20010301 |
| Multiple 5-HT(1) autoreceptor subtypes govern serotonin release in dorsal and median raphé nuclei. | Neuropharmacology 20010301 |
| Acute and chronic effects of citalopram on postsynaptic 5-hydroxytryptamine(1A) receptor-mediated feedback: a microdialysis study in the amygdala. | Journal of neurochemistry 20010301 |
| Short and efficient syntheses of analogues of WAY-100635: new and potent 5-HT1A receptor antagonists. | Bioorganic & medicinal chemistry 20010301 |
| Development of novel mixed-ligand oxotechnetium [SNS/S] complexes as potential 5-HT1A receptor imaging agents. | Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20010301 |
| Corticosterone selectively attenuates 8-OH-DPAT-mediated hypothermia in mice. | The international journal of neuropsychopharmacology 20010301 |
| Selective inhibition of amine oxidases differently potentiate the hypophagic effect of benzylamine in mice. | European journal of pharmacology 20010209 |
| Endogenous 5-HT tonically inhibits spontaneous firing activity of dorsal hippocampus CA1 pyramidal neurons through stimulation of 5-HT(1A) receptors in quiet awake rats: in vivo electrophysiological evidence. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010201 |
| Pharmacological characterisation of the decrease in 5-HT synthesis in the mouse brain evoked by the selective serotonin re-uptake inhibitor citalopram. | Naunyn-Schmiedeberg's archives of pharmacology 20010201 |
| Serotonergic modulation of retinal input to the mouse suprachiasmatic nucleus mediated by 5-HT1B and 5-HT7 receptors. | Journal of biological rhythms 20010201 |
| New halogenated [11C]WAY analogues, [11C]6FPWAY and [11C]6BPWAY--radiosynthesis and assessment as radioligands for the study of brain 5-HT1A receptors in living monkey. | Nuclear medicine and biology 20010201 |
| New 1-aryl-3-(4-arylpiperazin-1-yl)propane derivatives, with dual action at 5-HT1A serotonin receptors and serotonin transporter, as a new class of antidepressants. | Journal of medicinal chemistry 20010201 |
| Exhaustion of the coital reflex in spinal male rats is reversed by the serotonergic agonist 8-OH-DPAT. | Behavioural brain research 20010129 |
| Catalepsy induced by the 5-HT(1A) receptor antagonist WAY 100635 in rats pretreated with the selective serotonin reuptake inhibitor citalopram. | European journal of pharmacology 20010112 |
| Desensitization of 5-HT(1A) autoreceptors by a low chronic fluoxetine dose effect of the concurrent administration of WAY-100635. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010101 |
| Role of dorsal raphe neurons in paradoxical sleep generation in the cat: no evidence for a serotonergic mechanism. | The European journal of neuroscience 20010101 |
| Differential modulation by GTPgammaS of agonist and inverse agonist binding to h5-HT(1A) receptors revealed by [3H]-WAY100,635. | British journal of pharmacology 20010101 |
| Regulation of 5-HT(1A) receptor-stimulated [35S]-GtpgammaS binding as measured by quantitative autoradiography following chronic agonist administration. | British journal of pharmacology 20010101 |
| 5-HT(7) receptors activate the mitogen activated protein kinase extracellular signal related kinase in cultured rat hippocampal neurons. | Neuroscience 20010101 |
| Selectively bred male rat lines differ in naïve and experienced sexual behavior. | Physiology & behavior 20010101 |
| Involvement of somatodendritic 5-HT(1A) receptors in Delta(9)-tetrahydrocannabinol-induced hypothermia in the rat. | Pharmacology, biochemistry, and behavior 20010101 |
| The hypotensive effect of BMY 7378 is antagonized by a silent 5-HT(1A) receptor antagonist: comparison with 8-hydroxy-dipropylamino tetralin. | Archives of medical research 20010101 |
| Interactive effects of cholecystokinin-8S and various serotonin receptor agonists on the firing activity of neostriatal neuronesin rats. | Neuropeptides 20010101 |
| 5-HT1A receptor agonists buspirone and gepirone attenuate apomorphine-induced aggressive behaviour in adult male Wistar rats. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20001201 |
| Involvement of 5-hydroxytryptamine(1A) receptors in nicotine-induced tail tremor in rats. | European journal of pharmacology 20001110 |
| Effects of the serotonin 5-HT(2) antagonist, ritanserin, and the serotonin 5-HT(1A) antagonist, WAY 100635, on cocaine-seeking in rats. | Pharmacology, biochemistry, and behavior 20001001 |
| Neurobiological mechanisms by which nicotine mediates different types of anxiety. | European journal of pharmacology 20000330 |
| S 15535, a benzodioxopiperazine acting as presynaptic agonist and postsynaptic 5-HT1A receptor antagonist, prevents the impairment of spatial learning caused by intrahippocampal scopolamine. | British journal of pharmacology 19991101 |
| RU-24969 disrupts d-amphetamine self-administration and responding for conditioned reward via stimulation of 5-HT1B receptors. | Behavioural pharmacology 19990301 |
| The effects of 5-HT1A receptor agonists, 5-HT1A receptor antagonists and their interaction on the fear-potentiated startle response. | Psychopharmacology 19981001 |
| Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study. | European journal of pharmacology 19980821 |
| Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists. | Naunyn-Schmiedeberg's archives of pharmacology 19980301 |
| Anxiolytic effects of flesinoxan in the stress-induced hyperthermia paradigm in singly-housed mice are 5-HT1A receptor mediated. | European journal of pharmacology 19980126 |
| The pharmacological characterization of a novel selective 5-hydroxytryptamine1A receptor antagonist, NAD-299. | The Journal of pharmacology and experimental therapeutics 19971001 |
| Agonist activity of antimigraine drugs at recombinant human 5-HT1A receptors: potential implications for prophylactic and acute therapy. | Naunyn-Schmiedeberg's archives of pharmacology 19970601 |
| The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. | European journal of pharmacology 19970501 |
| Potentiation of fluoxetine-induced penile erections by combined blockade of 5-HT1A and 5-HT1B receptors. | European journal of pharmacology 19970305 |
| Pharmacological characterization of recombinant human 5-hydroxytryptamine1A receptors using a novel antagonist radioligand, [3H]WAY-100635. | Life sciences 19970101 |
| 5-HT1A receptors are not involved in clozapine's lack of cataleptogenic potential. | Neuropharmacology 19960101 |
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