CAS 106243-16-7 | N-Cyclohexyl-4-(1H-imidazol-5-yl)-1-piperidinecarbothioamide | CAS Number 106243-16-7

Title	Journal
Involvement of the histamine H4 receptor in clozapine-induced hematopoietic toxicity: Vulnerability under granulocytic differentiation of HL-60 cells.	Toxicology and applied pharmacology 20160901
Histamine at low concentrations aggravates rat liver BRL-3A cell injury induced by hypoxia/reoxygenation through histamine H2 receptor in vitro.	Toxicology in vitro : an international journal published in association with BIBRA 20130201
Proxyfan acts as a neutral antagonist of histamine H3 receptors in the feeding-related hypothalamic ventromedial nucleus.	British journal of pharmacology 20121101
Histamine H4 receptor antagonists as potent modulators of mammalian vestibular primary neuron excitability.	British journal of pharmacology 20121001
Ophthalmic antihistamines and H1-H4 receptors.	Current opinion in allergy and clinical immunology 20121001
Role of L-carnosine in the control of blood glucose, blood pressure, thermogenesis, and lipolysis by autonomic nerves in rats: involvement of the circadian clock and histamine.	Amino acids 20120701
A bioinformatics search for selective histamine h4 receptor antagonists through structure-based virtual screening strategies.	Chemical biology & drug design 20120501
Effects of neonatal methamphetamine and thioperamide exposure on spatial memory retention and circadian activity later in life.	Behavioural brain research 20120421
Histamine reverses a memory deficit induced in rats by early postnatal maternal deprivation.	Neurobiology of learning and memory 20120101
Ligand based design of novel histamine H₄ receptor antagonists; fragment optimization and analysis of binding kinetics.	Bioorganic & medicinal chemistry letters 20120101
In vivo receptor occupancy assay of histamine H₃ receptor antagonist in rats using non-radiolabeled tracer.	Journal of pharmacological and toxicological methods 20120101
Anti-stress effects of carnosine on restraint-evoked immunocompromise in mice through spleen lymphocyte number maintenance.	PloS one 20120101
Unusual effects of nicotine as a psychostimulant on ambulatory activity in mice.	ISRN pharmacology 20120101
Histamine is a modulator of metamorphic competence in Strongylocentrotus purpuratus (Echinodermata: Echinoidea).	BMC developmental biology 20120101
Desipramine inhibits histamine H1 receptor-induced Ca2+ signaling in rat hypothalamic cells.	PloS one 20120101
Histamine neurons in the tuberomamillary nucleus: a whole center or distinct subpopulations?	Frontiers in systems neuroscience 20120101
Histamine h3 receptor: a novel therapeutic target in alcohol dependence?	Frontiers in systems neuroscience 20120101
Identification and characterization of ZEL-H16 as a novel agonist of the histamine H3 receptor.	PloS one 20120101
The mediation of the central histaminergic system in the pressor effect of intracerebroventricularly injected melittin, a phospholipase A2 activator, in normotensive rats.	Prostaglandins, leukotrienes, and essential fatty acids 20120101
Searching for the Multi-Target-Directed Ligands against Alzheimer's disease: discovery of quinoxaline-based hybrid compounds with AChE, H₃R and BACE 1 inhibitory activities.	Bioorganic & medicinal chemistry 20111201
The role of cortical and hypothalamic histamine-3 receptors in the modulation of central histamine neurotransmission: an in vivo electrophysiology and microdialysis study.	The European journal of neuroscience 20111201
The hydrophobic amino acids in putative helix 8 in carboxy-terminus of histamine H(3) receptor are involved in receptor-G-protein coupling.	Cellular signalling 20111101
Differential modulation of excitatory and inhibitory striatal synaptic transmission by histamine.	The Journal of neuroscience : the official journal of the Society for Neuroscience 20111026
Differential effects of histamine H(3) receptor inverse agonist thioperamide, given alone or in combination with the N-methyl-d-aspartate receptor antagonist dizocilpine, on reconsolidation and consolidation of a contextual fear memory in mice.	Neuroscience 20111013
Histamine facilitates consolidation of fear extinction.	The international journal of neuropsychopharmacology 20111001
In vivo electrochemical evidence for simultaneous 5-HT and histamine release in the rat substantia nigra pars reticulata following medial forebrain bundle stimulation.	Journal of neurochemistry 20110901
Role of the second and third extracellular loops of the histamine H(4) receptor in receptor activation.	Naunyn-Schmiedeberg's archives of pharmacology 20110901
Ontogenetic serotoninergic lesioning alters histaminergic activity in rats in adulthood.	Neurotoxicity research 20110801
Thioperamide, an H₃ receptor antagonist prevents [³H]glucose uptake in brain of adult rats lesioned as neonates with 5,7-dihydroxytryptamine.	Neurotoxicity research 20110701
Involvement of histaminergic receptor mechanisms in the stimulation of NT-3 synthesis in astrocytes.	Neuropharmacology 20110601
Prepulse inhibition of the startle reflex and response to antipsychotic treatments in two outbred mouse strains in comparison to the inbred DBA/2 mouse.	Psychopharmacology 20110601
Memory facilitating effects of agomelatine in the novel object recognition memory paradigm in the rat.	Pharmacology, biochemistry, and behavior 20110601
Histaminergic regulation of seasonal metabolic rhythms in Siberian hamsters.	Physiology & behavior 20110601
Regulation of ERK2 phosphorylation by histamine in splenocytes.	Immunopharmacology and immunotoxicology 20110601
The histamine H3 receptor: from discovery to clinical trials with pitolisant.	British journal of pharmacology 20110601
Effects of histamine H3 receptors on chemical hyperalgesia in diabetic rats.	Neuropharmacology 20110501
N-Alkenyl and cycloalkyl carbamates as dual acting histamine H3 and H4 receptor ligands.	Bioorganic & medicinal chemistry 20110501
Agonist-biased signaling at the histamine H4 receptor: JNJ7777120 recruits β-arrestin without activating G proteins.	Molecular pharmacology 20110401
Newer molecules in the treatment of schizophrenia: A clinical update.	Indian journal of pharmacology 20110401
Triazole ligands reveal distinct molecular features that induce histamine H4 receptor affinity and subtly govern H4/H3 subtype selectivity.	Journal of medicinal chemistry 20110324
Antidiabetic properties of the histamine H3 receptor protean agonist proxyfan.	Endocrinology 20110301
Skin application of urea-containing cream affected cutaneous arterial sympathetic nerve activity, blood flow, and water evaporation.	Skin research and technology : official journal of International Society for Bioengineering and the Skin (ISBS) [and] International Society for Digital Imaging of Skin (ISDIS) [and] International Society for Skin Imaging (ISSI) 20110201
Guinea pig ileum motility stimulation elicited by N-formyl-Met-Leu-Phe (fMLF) involves neurotransmitters and prostanoids.	Peptides 20110201
[Roles of histamine in the exacerbated allergic dermatitis].	Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20110201
Histamine H3 receptor as a drug discovery target.	Journal of medicinal chemistry 20110113
H3 receptors and pain modulation: peripheral, spinal, and brain interactions.	The Journal of pharmacology and experimental therapeutics 20110101
Effects of antihistamines on innate immune responses to severe bacterial infection in mice.	International archives of allergy and immunology 20110101
Histaminergic mechanisms for modulation of memory systems.	Neural plasticity 20110101
Inverse agonism and its therapeutic significance.	Indian journal of pharmacology 20110101
Thioperamide induces CD4 CD25 Foxp3 regulatory T lymphocytes in the lung mucosa of allergic mice through its action on dendritic cells.	Journal of asthma and allergy 20110101
Kv4.2 mediates histamine modulation of preoptic neuron activity and body temperature.	PloS one 20110101
Biological Significance of GPCR Heteromerization in the Neuro-Endocrine System.	Frontiers in endocrinology 20110101
Histamine 3 receptor activation mediates inhibition of acid secretion during Helicobacter-induced gastritis.	World journal of gastrointestinal pathophysiology 20101215
Microinjection of histamine into the dentate gyrus produces antinociception in the formalin test in rats.	Pharmacology, biochemistry, and behavior 20101201
Comparison of the pharmacological properties of human and rat histamine H(3)-receptors.	Biochemical pharmacology 20101101
Structural basis of drug binding to CYP46A1, an enzyme that controls cholesterol turnover in the brain.	The Journal of biological chemistry 20101008
Validation and pharmacological characterisation of MK-801-induced locomotor hyperactivity in BALB/C mice as an assay for detection of novel antipsychotics.	Psychopharmacology 20101001
Histamine H(3) receptor modulates nociception in a rat model of cholestasis.	Pharmacology, biochemistry, and behavior 20100901
Environmental stressors and neurobiological features of marine teleosts: histamine receptors as targets.	Critical reviews in toxicology 20100801
Effect of anserine ingestion on hyperglycemia and the autonomic nerves in rats and humans.	Nutritional neuroscience 20100801
Effect of combined treatment of thioperamide with some antiepileptic drugs on methionine-sulfoximine induced convulsions in mice.	Indian journal of experimental biology 20100801
Histamine H3 receptor activation potentiates peripheral opioid-mediated antinociception: substance P role in peripheral inflammation in mice.	European journal of pharmacology 20100725
Effect of anserine ingestion on the hyperglycemia and autonomic nerves in rats and humans.	Nutritional neuroscience 20100601
Effects of sympathetic histamine on vasomotor responses of blood vessels in rabbit ear to electrical stimulation.	Neuroscience bulletin 20100601
Investigation of the bioactive conformation of histamine H3 receptor antagonists by the cyclopropylic strain-based conformational restriction strategy.	Journal of medicinal chemistry 20100513
Molecular determinants of ligand binding to H4R species variants.	Molecular pharmacology 20100501
Impact of the DRY motif and the missing 'ionic lock' on constitutive activity and G-protein coupling of the human histamine H4 receptor.	The Journal of pharmacology and experimental therapeutics 20100501
Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists.	Bioorganic & medicinal chemistry letters 20100415
Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.	Journal of medicinal chemistry 20100325
Modulation of histamine H(3) receptor function by monovalent ions.	Neuroscience letters 20100319
Neuropharmacology of vestibular system disorders.	Current neuropharmacology 20100301
Modeling G protein-coupled receptors for structure-based drug discovery using low-frequency normal modes for refinement of homology models: application to H3 antagonists.	Proteins 20100201
Synthesis and structural and pharmacological properties of cyclopropane-based conformationally restricted analogs of 4-methylhistamine as histamine H3/H4 receptor ligands.	Bioorganic & medicinal chemistry 20100201
Involvement of the histaminergic system in cytidine 5'-diphosphocholine-induced reversal of critical haemorrhagic hypotension in rats.	Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20100201
Effects of anserine on the renal sympathetic nerve activity and blood pressure in urethane-anesthetized rats.	Physiological research 20100101
Oral L-histidine exerts antihypertensive effects via central histamine H3 receptors and decreases nitric oxide content in the rostral ventrolateral medulla in spontaneously hypertensive rats.	Clinical and experimental pharmacology & physiology 20100101
Contribution of mast cells to the oedema induced by Bothrops moojeni snake venom and a pharmacological assessment of the inflammatory mediators involved.	Toxicon : official journal of the International Society on Toxinology 20100101
Pretreatment with l-histidine produces a shift from methamphetamine-induced stereotypical biting to persistent locomotion in mice.	Pharmacology, biochemistry, and behavior 20100101
R-(-)-alpha-methylhistamine, a histamine H3 receptor agonist, induces endothelium-dependent vasodilation in rat mesenteric resistance arteries.	Biological & pharmaceutical bulletin 20100101
Different role of cAMP dependent protein kinase and CaMKII in H3 receptor regulation of histamine synthesis and release.	Neuroscience 20091215
The effects of thioperamide on extracellular levels of glutamate and GABA in the rat prefrontal cortex.	Psychopharmacology 20091201
Histamine H3 and H4 receptor affinity of branched 3-(1H-imidazol-4-yl)propyl N-alkylcarbamates.	Bioorganic & medicinal chemistry letters 20091201
Heterocyclic replacement of the central phenyl core of diamine-based histamine H3 receptor antagonists.	European journal of medicinal chemistry 20091101
Interactions of histamine H1-receptor agonists and antagonists with the human histamine H4-receptor.	Molecular pharmacology 20091101
Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H4 receptor agonists.	Journal of medicinal chemistry 20091022
2,4-Diaminopyrimidines as histamine H4 receptor ligands--Scaffold optimization and pharmacological characterization.	Bioorganic & medicinal chemistry 20091015
Diamine-based human histamine H3 receptor antagonists: (4-aminobutyn-1-yl)benzylamines.	European journal of medicinal chemistry 20091001
Effects of the H(3) antagonist, thioperamide, on behavioral alterations induced by systemic MK-801 administration in rats.	Psychopharmacology 20090901
Enhanced morphine-induced antinociception in histamine H3 receptor gene knockout mice.	Neuropharmacology 20090901
Anxiolytic-like profiles of histamine H3 receptor agonists in animal models of anxiety: a comparative study with antidepressants and benzodiazepine anxiolytic.	Psychopharmacology 20090801
Development of a selective and potent radioactive ligand for histamine H(3) receptors: A compound potentially useful for receptor occupancy studies.	Bioorganic & medicinal chemistry letters 20090801
JNJ-10181457, a selective non-imidazole histamine H(3) receptor antagonist, normalizes acetylcholine neurotransmission and has efficacy in translational rat models of cognition.	Neuropharmacology 20090601
Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studies.	Bioorganic & medicinal chemistry 20090601
Heterogeneity of histaminergic neurons in the tuberomammillary nucleus of the rat.	The European journal of neuroscience 20090601
N(G)-acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.	Journal of medicinal chemistry 20090423
Non-imidazole histamine H3 ligands, part IV: SAR of 1-[2-thiazol-5-yl-(2-aminoethyl)]-4-n-propylpiperazine derivatives.	European journal of medicinal chemistry 20090401
Characterization of histamine-induced relaxation in pre-contracted rat aorta.	Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20090401
Histaminergic activity in a rodent model of Parkinson's disease.	Neurotoxicity research 20090401
Effects of the H3 receptor inverse agonist thioperamide on cocaine-induced locomotion in mice: role of the histaminergic system and potential pharmacokinetic interactions.	Psychopharmacology 20090301
The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.	Behavioural pharmacology 20090301
High constitutive activity and a G-protein-independent high-affinity state of the human histamine H(4)-receptor.	Biochemistry 20090217
Autonomic and cardiovascular effects of central neuromedin U in rats.	Physiology & behavior 20090216
Possible role of the histaminergic system in autonomic and cardiovascular responses to neuropeptide Y.	Neuropeptides 20090201
H3 receptor antagonists reverse delay-dependent deficits in novel object discrimination by enhancing retrieval.	Psychopharmacology 20090101
Modification of the picryl chloride-induced allergic dermatitis model in mouse ear lobes by 12-O-tetradecanoylphorbol 13-acetate, and analysis of the role of histamine in the modified model.	International archives of allergy and immunology 20090101
L-histidine enhances learning in stressed zebrafish.	Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20090101
Cytokine responses of intraepithelial lymphocytes are regulated by histamine H(2) receptor.	Journal of gastroenterology 20090101
A novel flow cytometric high throughput assay for a systematic study on molecular mechanisms underlying T cell receptor-mediated integrin activation.	PloS one 20090101
Alpha2 adrenoceptors modulate histamine release from sympathetic nerves in the guinea pig vas deferens.	Neuropharmacology 20090101
H4 histamine receptors mediate cell cycle arrest in growth factor-induced murine and human hematopoietic progenitor cells.	PloS one 20090101
Modulatory effects of histamine on cat carotid body chemoreception.	Respiratory physiology & neurobiology 20081231
Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach.	Journal of medicinal chemistry 20081225
Role of histamine in short- and long-term effects of methamphetamine on the developing mouse brain.	Journal of neurochemistry 20081101
Biphasic effects of orexin-A on autonomic nerve activity and lipolysis.	Neuroscience letters 20081024
Effect of thioperamide on oxidative stress markers in middle cerebral artery occlusion model of focal cerebral ischemia in rats.	Human & experimental toxicology 20081001
The alkaloid conessine and analogues as potent histamine H3 receptor antagonists.	Journal of medicinal chemistry 20080911
Electrophysiology-based analysis of human histamine H(4) receptor pharmacology using GIRK channel coupling in Xenopus oocytes.	European journal of pharmacology 20080904
Localization and function of histamine H3 receptor in the nasal mucosa.	Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20080901
Alleviation of ischemia-induced brain edema by activation of the central histaminergic system in rats.	Journal of pharmacological sciences 20080901
Regulation of sympathetic nerve activity by L-carnosine in mammalian white adipose tissue.	Neuroscience letters 20080815
Discovery of novel human histamine H4 receptor ligands by large-scale structure-based virtual screening.	Journal of medicinal chemistry 20080612
Correlation between ex vivo receptor occupancy and wake-promoting activity of selective H3 receptor antagonists.	The Journal of pharmacology and experimental therapeutics 20080601
Blocking histamine H(1) improves learning and mnemonic dysfunction in mice with social isolation plus repeated methamphetamine injection.	Journal of pharmacological sciences 20080601
Zebrafish: An in vivo model for the study of neurological diseases.	Neuropsychiatric disease and treatment 20080601
Narcolepsy: current treatment options and future approaches.	Neuropsychiatric disease and treatment 20080601
Interactions between histamine H3 and dopamine D2 receptors and the implications for striatal function.	Neuropharmacology 20080516
Fragment based design of new H4 receptor-ligands with anti-inflammatory properties in vivo.	Journal of medicinal chemistry 20080424
Histamine action on vertebrate GABAA receptors: direct channel gating and potentiation of GABA responses.	The Journal of biological chemistry 20080418
Role of histamine in brain protection in surgical brain injury in mice.	Brain research 20080418
Effects of oolong tea on renal sympathetic nerve activity and spontaneous hypertension in rats.	Metabolism: clinical and experimental 20080401
Ontogenetic noradrenergic lesion alters histaminergic activity in adult rats.	Neurotoxicity research 20080401
Specific cerebral heat shock proteins and histamine receptor cross-talking mechanisms promote distinct lead-dependent neurotoxic responses in teleosts.	Toxicology and applied pharmacology 20080301
Comparative effects of olanzapine and ziprasidone on hypophagia induced by enhanced histamine neurotransmission in the rat.	Behavioural pharmacology 20080301
Carnosine protects against Abeta42-induced neurotoxicity in differentiated rat PC12 cells.	Cellular and molecular neurobiology 20080201
Effects of central histamine receptors blockade on GABA(A) agonist-induced food intake in broiler cockerels.	Pakistan journal of biological sciences : PJBS 20080201
Antigen inhalation induces mast cells and eosinophils infiltration in the guinea pig esophageal epithelium involving histamine-mediated pathway.	Life sciences 20080130
Distinctive role of central histamine H3 receptor in various orexigenic pathways.	European journal of pharmacology 20080128
CSF histamine levels in rats reflect the central histamine neurotransmission.	Neuroscience letters 20080117
Modulation of hippocampal theta oscillation by histamine H3 receptors.	The Journal of pharmacology and experimental therapeutics 20080101
Mast cell-derived histamine mediates cystitis pain.	PloS one 20080101
Histamine H(3) receptor ligands modulate L-dopa-evoked behavioral responses and L-dopa derived extracellular dopamine in dopamine-denervated rat striatum.	Neurotoxicity research 20080101
Antagonist affinity measurements at the Gi-coupled human histamine H3 receptor expressed in CHO cells.	BMC pharmacology 20080101
Histamine-induced itch and its relationship with pain.	Molecular pain 20080101
The possible involvement of hyperpolarizing mechanisms in histamine-induced relaxation of the rat portal vein.	Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi 20080101
Histamine in Macaca mulatto monkey cardiac sympathetic nerve system: a morphological and functional assessment.	Autonomic neuroscience : basic & clinical 20071230
Functional expression of H4 histamine receptor in human natural killer cells, monocytes, and dendritic cells.	Journal of immunology (Baltimore, Md. : 1950) 20071201
The role of carcinine in signaling at the Drosophila photoreceptor synapse.	PLoS genetics 20071201
Activation of peripheral and spinal histamine H3 receptors inhibits formalin-induced inflammation and nociception, respectively.	Pharmacology, biochemistry, and behavior 20071101
Reduced histamine levels and H3 receptor antagonist-induced histamine release in the amygdala of Apoe-/- mice.	Journal of neurochemistry 20071001
The Akt/GSK-3beta axis as a new signaling pathway of the histamine H(3) receptor.	Journal of neurochemistry 20071001
Histamine improves antigen uptake and cross-presentation by dendritic cells.	Journal of immunology (Baltimore, Md. : 1950) 20070915
Interaction of nicotinic and histamine H(3) systems in the radial-arm maze repeated acquisition task.	European journal of pharmacology 20070813
Betahistine in the treatment of Ménière's disease.	Neuropsychiatric disease and treatment 20070801
Histaminergic ligands improve vestibular compensation in the cat: behavioural, neurochemical and molecular evidence.	European journal of pharmacology 20070730
Blockade of brain histamine metabolism alters methamphetamine-induced expression pattern of stereotypy in mice via histamine H1 receptors.	Neuroscience 20070713
Histamine H4 receptor agonists have more activities than H4 agonism in antigen-specific human T-cell responses.	Immunology 20070601
Interaction of calcitonin gene-related peptide, nitric oxide and histamine release in neurogenic blood flow and afferent activation in the rat cranial dura mater.	Cephalalgia : an international journal of headache 20070601
H3 histamine receptor agonist inhibits biliary growth of BDL rats by downregulation of the cAMP-dependent PKA/ERK1/2/ELK-1 pathway.	Laboratory investigation; a journal of technical methods and pathology 20070501
Histaminergic H1 receptors mediate L-histidine-induced anxiety in elevated plus-maze test in mice.	Behavioural pharmacology 20070501
Identification of zebrafish histamine H1, H2 and H3 receptors and effects of histaminergic ligands on behavior.	Biochemical pharmacology 20070415
The brain H3-receptor as a novel therapeutic target for vigilance and sleep-wake disorders.	Biochemical pharmacology 20070415
Auditory stimulation affects renal sympathetic nerve activity and blood pressure in rats.	Neuroscience letters 20070412
Thioperamide reduces intracellular calcium in mouse brain synaptosomes.	European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20070401
Influence of the H3/H4 receptor antagonist, thioperamide on regional haemodynamics in rats with trinitrobenzene sulfonic acid-induced colitis.	Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20070401
Thioperamide delays vestibular compensation in goldfish.	Neuroscience letters 20070326
Sex- and histamine-dependent long-term cognitive effects of methamphetamine exposure.	Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20070301
Carnosine protects against NMDA-induced neurotoxicity in differentiated rat PC12 cells through carnosine-histidine-histamine pathway and H(1)/H(3) receptors.	Biochemical pharmacology 20070301
Histamine affects STAT6 phosphorylation via its effects on IL-4 secretion: role of H1 receptors in the regulation of IL-4 production.	International immunopharmacology 20070301
Suppression of inflammatory cell recruitment by histamine receptor stimulation in ischemic rat brains.	European journal of pharmacology 20070227
Involvement of the histaminergic system in renal sympathetic and cardiovascular responses to leptin and ghrelin.	Neuroscience letters 20070208
In vitro pharmacology at human histamine H3 receptors and brain access of non-imidazole alkylpiperidine derivatives.	Pharmacological research 20070201
Modification of formalin-induced nociception by different histamine receptor agonists and antagonists.	European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20070115
Role of apolipoprotein E in anxiety.	Neural plasticity 20070101
Role of histamine H3 and H4 receptors in mechanical hyperalgesia following peripheral nerve injury.	Neuroimmunomodulation 20070101
Histamine H3 receptor agonist- and antagonist-evoked vacuous chewing movements in 6-OHDA-lesioned rats occurs in an absence of change in microdialysate dopamine levels.	European journal of pharmacology 20061215
Feeding differences in pubertal and aged golden hamsters (Mesocricetus auratus) are related to specific cerebral expression pattern of histamine subtype 3 receptor.	Behavioral neuroscience 20061201
Expression of histamine receptors and effect of histamine in the rat carotid body chemoafferent pathway.	The European journal of neuroscience 20061201
Mechanism of imipramine-induced seizures in amygdala-kindled rats.	Epilepsy research 20061101
Renoprotective effects of l-carnosine on ischemia/reperfusion-induced renal injury in rats.	The Journal of pharmacology and experimental therapeutics 20061101
Dose-different effects of orexin-A on the renal sympathetic nerve and blood pressure in urethane-anesthetized rats.	Experimental biology and medicine (Maywood, N.J.) 20061101
A comparison of protective effects between L-histidine and hypothermia against ischemia-induced neuronal damage in gerbil hippocampus.	European journal of pharmacology 20060928
Stereochemical diversity-oriented conformational restriction strategy. Development of potent histamine H3 and/or H4 receptor antagonists with an imidazolylcyclopropane structure.	Journal of medicinal chemistry 20060907
Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway.	Neuropharmacology 20060901
Suppression of ischemia/reperfusion liver injury by histamine H4 receptor stimulation in rats.	European journal of pharmacology 20060821
Homologous down-regulation of histamine H3 receptors in rat striatal slices.	Synapse (New York, N.Y.) 20060801
Antipsychotic-like profile of thioperamide, a selective H3-receptor antagonist in mice.	Fundamental & clinical pharmacology 20060801
Evidence for histamine as a neurotransmitter in the cardiac sympathetic nervous system.	American journal of physiology. Heart and circulatory physiology 20060701
Histamine enhances inhibitory avoidance memory consolidation through a H2 receptor-dependent mechanism.	Neurobiology of learning and memory 20060701
Impaired drinking response in histamine H3 receptor knockout mice following dehydration or angiotensin-II challenge.	Pharmacology, biochemistry, and behavior 20060701
Increasing synaptic noradrenaline, serotonin and histamine enhances in vivo binding of phosphodiesterase-4 inhibitor (R)-[11C]rolipram in rat brain, lung and heart.	Life sciences 20060620
Changes in the histaminergic system during vestibular compensation in the cat.	The Journal of physiology 20060615
The effect of histamine on field-stimulated contractions of the guinea-pig prostate.	Naunyn-Schmiedeberg's archives of pharmacology 20060601
Histamine-induced enhancement of vasopressin and oxytocin secretion in rat neurohypophyseal tissue cultures.	Regulatory peptides 20060515
Olfactory stimulation with scent of lavender oil affects autonomic neurotransmission and blood pressure in rats.	Neuroscience letters 20060501
Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.	British journal of pharmacology 20060401
Effects of the H3-receptor inverse agonist thioperamide on the psychomotor effects induced by acutely and repeatedly given cocaine in C57BL/6J mice.	Pharmacology, biochemistry, and behavior 20060401
Effects of histamine H(3) antagonists and donepezil on learning and mnemonic deficits induced by pentylenetetrazol kindling in weanling mice.	Neuropharmacology 20060301
Role of H1 receptors in histamine-mediated up-regulation of STAT4 phosphorylation.	International immunopharmacology 20060301
Histamine protects against NMDA-induced necrosis in cultured cortical neurons through H receptor/cyclic AMP/protein kinase A and H receptor/GABA release pathways.	Journal of neurochemistry 20060301
Histamine increases sickle erythrocyte adherence to endothelium.	British journal of haematology 20060201
[The effect of central histamine H3 receptor on breathing activity of asthmatic guinea pigs].	Zhongguo ying yong sheng li xue za zhi = Zhongguo yingyong shenglixue zazhi = Chinese journal of applied physiology 20060201
Histaminergic neurons protect the developing hippocampus from kainic acid-induced neuronal damage in an organotypic coculture system.	The Journal of neuroscience : the official journal of the Society for Neuroscience 20060125
The hallucinogenic herb Salvia divinorum and its active ingredient salvinorin A inhibit enteric cholinergic transmission in the guinea-pig ileum.	Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20060101
Histamine receptors influence blood-spinal cord barrier permeability, edema formation, and spinal cord blood flow following trauma to the rat spinal cord.	Acta neurochirurgica. Supplement 20060101
Aversive memory reactivation engages in the amygdala only some neurotransmitters involved in consolidation.	Learning & memory (Cold Spring Harbor, N.Y.) 20060101
Reduction in brain infarction by augmentation of central histaminergic activity in rats.	Brain research 20051220
Histamine (H3) receptors modulate the excitatory amino acid receptor response of the vestibular afferents.	Brain research 20051207
Effects of intraduodenal injection of Lactobacillus johnsonii La1 on renal sympathetic nerve activity and blood pressure in urethane-anesthetized rats.	Neuroscience letters 20051202
Mechanisms of histamine-induced relaxation in bovine small adrenal cortical arteries.	American journal of physiology. Endocrinology and metabolism 20051201
Sleep disturbances, psychiatric disorders, and psychotropic drugs.	Dialogues in clinical neuroscience 20051201
Some environmental contaminants influence motor and feeding behaviors in the ornate wrasse (Thalassoma pavo) via distinct cerebral histamine receptor subtypes.	Environmental health perspectives 20051101
The histaminergic signaling system exerts a neuroprotective role against neurodegenerative-induced processes in the hamster.	The Journal of pharmacology and experimental therapeutics 20051001
Modulation of spontaneous alternation performance of mice treated with thioperamide and tacrine in a cross maze task.	Fundamental & clinical pharmacology 20051001
Effect of thioperamide on modified forced swimming test-induced oxidative stress in mice.	Basic & clinical pharmacology & toxicology 20051001
Olfactory stimulation with scent of lavender oil affects autonomic nerves, lipolysis and appetite in rats.	Neuroscience letters 20050701
Involvement of histamine H1 and H2 receptors in the regulation of STAT-1 phosphorylation: inverse agonism exhibited by the receptor antagonists.	International immunopharmacology 20050701
Histamine excites noradrenergic neurons in locus coeruleus in rats.	Neuropharmacology 20050701
Histamine-3 receptor antagonists reduce superoxide anion generation and lipid peroxidation in rat brain homogenates.	The Journal of pharmacy and pharmacology 20050601
Generation of cell lines for drug discovery through random activation of gene expression: application to the human histamine H3 receptor.	Assay and drug development technologies 20050601
Lack of cataleptogenic potentiation with non-imidazole H3 receptor antagonists reveals potential drug-drug interactions between imidazole-based H3 receptor antagonists and antipsychotic drugs.	Brain research 20050531
The H3 antagonist thioperamide reveals conditioned preference for a context associated with an inactive small dose of cocaine in C57BL/6J mice.	Behavioural brain research 20050507
Effects of histamine H3 receptor antagonists in two models of spatial learning.	Behavioural brain research 20050430
Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H3 receptor antagonist.	The Journal of pharmacology and experimental therapeutics 20050401
4-phenoxypiperidines: potent, conformationally restricted, non-imidazole histamine H3 antagonists.	Journal of medicinal chemistry 20050324
Effect of combined histamine H1 and H3 receptor blockade on cutaneous microvascular permeability elicited by compound 48/80.	Life sciences 20050304
Histamine receptors that influence blockage of the normal human nasal airway.	British journal of pharmacology 20050301
Assessment of pharmacology and potential anti-obesity properties of H3 receptor antagonists/inverse agonists.	Expert opinion on investigational drugs 20050301
Dose-dependent effects of L-carnosine on the renal sympathetic nerve and blood pressure in urethane-anesthetized rats.	American journal of physiology. Regulatory, integrative and comparative physiology 20050201
A biochemical and pharmacological examination of Rhamphiophis oxyrhynchus (Rufous beaked snake) venom.	Toxicon : official journal of the International Society on Toxinology 20050201
Role of capsaicin-sensitive nerves and histamine H1, H2, and H3 receptors in the gastroprotective effect of histamine against stress ulcers in rats.	European journal of pharmacology 20050131
4-(2-[2-(2(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and related 2-aminoethylbenzofuran H3 receptor antagonists potently enhance cognition and attention.	Journal of medicinal chemistry 20050113
2-(4-alkylpiperazin-1-yl)quinolines as a new class of imidazole-free histamine H3 receptor antagonists.	Journal of medicinal chemistry 20050113
Histaminergic modulation of excitatory synaptic transmission in the rat basolateral amygdala.	Neuroscience 20050101
Histamine-induced cyclic AMP formation in the chick hypothalamus: interaction with vasoactive intestinal peptide.	Pharmacological reports : PR 20050101
[Participation of cyclic nucleotides and phospholipidis in signal transduction of histamin receptor H3 of the gastric mucosa parietal cells in rats with experimental ulcer].	Ukrains'kyi biokhimichnyi zhurnal (1999 ) 20050101
Role of histaminergic neurons in development of epileptic seizures in EL mice.	Brain research. Molecular brain research 20041206
Unusual functional properties of homo- and heteromultimeric histamine-gated chloride channels of Drosophila melanogaster: spontaneous currents and dual gating by GABA and histamine.	Neuroscience letters 20041130
Pharmacological effects of carcinine on histaminergic neurons in the brain.	British journal of pharmacology 20041101
Medicinal chemical and pharmacological aspects of imidazole-containing histamine H3 receptor antagonists.	Mini reviews in medicinal chemistry 20041101
Role of the histamine system in nefopam-induced antinociception in mice.	European journal of pharmacology 20041025
Histamine H3 receptors inhibit serotonin release in substantia nigra pars reticulata.	The Journal of neuroscience : the official journal of the Society for Neuroscience 20041006
Intranigral injection of the H3 agonist immepip and systemic apomorphine elicit ipsilateral turning behaviour in naive rats, but reduce contralateral turning in hemiparkinsonian rats.	Behavioural brain research 20041005
The in vitro and in vivo pharmacological activity of Boiga dendrophila (mangrove catsnake) venom.	Autonomic & autacoid pharmacology 20041001
Histamine H3 antagonist thioperamide dose-dependently enhances memory consolidation and reverses amnesia induced by dizocilpine or scopolamine in a one-trial inhibitory avoidance task in mice.	Behavioural brain research 20040923
Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist.	Biochemical pharmacology 20040901
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.	Journal of neurochemistry 20040901
Enhancement of prepulse inhibition of startle in mice by the H3 receptor antagonists thioperamide and ciproxifan.	Behavioural brain research 20040812
Liver-expressed chemokine/CC chemokine ligand 16 attracts eosinophils by interacting with histamine H4 receptor.	Journal of immunology (Baltimore, Md. : 1950) 20040801
Histamine H3 receptor activation inhibits dopamine D1 receptor-induced cAMP accumulation in rat striatal slices.	Neuroscience letters 20040708
Critical role of L-selectin and histamine H4 receptor in zymosan-induced neutrophil recruitment from the bone marrow: comparison with carrageenan.	The Journal of pharmacology and experimental therapeutics 20040701
Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain.	Journal of medicinal chemistry 20040603
Central H3R activation by thioperamide does not affect energy balance.	Pharmacology, biochemistry, and behavior 20040601
1-alkyl-4-acylpiperazines as a new class of imidazole-free histamine H(3) receptor antagonists.	Journal of medicinal chemistry 20040520
4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists.	Journal of medicinal chemistry 20040506
Involvement of histamine H4 and H1 receptors in scratching induced by histamine receptor agonists in Balb C mice.	British journal of pharmacology 20040501
Histamine H4 receptor mediates eosinophil chemotaxis with cell shape change and adhesion molecule upregulation.	British journal of pharmacology 20040501
Intracerebroventricular administration of histamine H3 receptor antagonists decreases seizures in rat models of epilepsia.	Methods and findings in experimental and clinical pharmacology 20040501
Histamine h3 receptor antagonists potentiate methamphetamine self-administration and methamphetamine-induced accumbal dopamine release.	Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040401
Inhibitory effect of iodophenpropit, a selective histamine H3 antagonist, on amygdaloid kindled seizures.	Brain research bulletin 20040315
Pruritus-associated response mediated by cutaneous histamine H3 receptors.	Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20040301
Thioperamide-elicited increase of histamine release from basolateral amygdala of freely moving rats and its therapeutic implications.	Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20040301
Role of histamine H3 receptors during ischemia/reperfusion in isolated rat hearts.	Journal of cardiovascular pharmacology 20040301
Plasticity of histamine H3 receptor expression and binding in the vestibular nuclei after labyrinthectomy in rat.	BMC neuroscience 20040101
Critical role of histamine H4 receptor in leukotriene B4 production and mast cell-dependent neutrophil recruitment induced by zymosan in vivo.	The Journal of pharmacology and experimental therapeutics 20031201
Role of histamine receptors in the regulation of edema and circulation postburn.	Burns : journal of the International Society for Burn Injuries 20031201
Histamine induces cytoskeletal changes in human eosinophils via the H(4) receptor.	British journal of pharmacology 20031101
Possible role of L-carnosine in the regulation of blood glucose through controlling autonomic nerves.	Experimental biology and medicine (Maywood, N.J.) 20031101
Generation and characterization of highly constitutive active histamine H3 receptors.	The Journal of pharmacology and experimental therapeutics 20031001
Aminergic control of high-frequency (approximately 200 Hz) network oscillations in the hippocampus of the behaving rat.	Neuroscience letters 20030911
The first potent and selective non-imidazole human histamine H4 receptor antagonists.	Journal of medicinal chemistry 20030911
Central endogenous histamine modulates sympathetic outflow through H3 receptors in the conscious rabbit.	British journal of pharmacology 20030701
Identification of a dual histamine H1/H3 receptor ligand based on the H1 antagonist chlorpheniramine.	Bioorganic & medicinal chemistry letters 20030616
Antinociceptive mechanisms of orally administered decursinol in the mouse.	Life sciences 20030613
Activation of spinal histamine H3 receptors inhibits mechanical nociception.	European journal of pharmacology 20030606
Two novel and selective nonimidazole H3 receptor antagonists A-304121 and A-317920: II. In vivo behavioral and neurophysiological characterization.	The Journal of pharmacology and experimental therapeutics 20030601
Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects.	The Journal of pharmacology and experimental therapeutics 20030601
Histamine H4 receptor mediates chemotaxis and calcium mobilization of mast cells.	The Journal of pharmacology and experimental therapeutics 20030601
H3 receptor blockade by thioperamide enhances cognition in rats without inducing locomotor sensitization.	Psychopharmacology 20030601
Cyclopropane-based conformational restriction of histamine. (1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a highly selective agonist for the histamine H3 receptor, having a cis-cyclopropane structure.	Journal of medicinal chemistry 20030508
Regulation by prostaglandin E2 and histamine of angiogenesis in inflammatory granulation tissue.	Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20030501
Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds.	Journal of medicinal chemistry 20030410
Histamine inhibits lipopolysaccharide-induced tumor necrosis factor-alpha production in an intercellular adhesion molecule-1- and B7.1-dependent manner.	The Journal of pharmacology and experimental therapeutics 20030201
Histaminergic modulation of the intact respiratory network of adult mice.	Pflugers Archiv : European journal of physiology 20030201
Histamine-induced chloride secretion is mediated via H2-receptors in the pig proximal colon.	Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20030201
Neuroimmune interactions in guinea pig stomach and small intestine.	American journal of physiology. Gastrointestinal and liver physiology 20030101
Functional identification of epithelial and smooth muscle histamine-dependent relaxing mechanisms in the bovine trachea, but not in bronchi.	Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20030101
Replacement of imidazole by a piperidine moiety differentially affects the potency of histamine H3-receptor antagonists.	Naunyn-Schmiedeberg's archives of pharmacology 20030101
High-frequency oscillation in the hippocampus of the behaving rat and its modulation by the histaminergic system.	Hippocampus 20030101
Contribution of the histaminergic receptor subtypes to histamine-induced cerebellar granular neurotoxicity.	Polish journal of pharmacology 20030101
Targeted disruption of H3 receptors results in changes in brain histamine tone leading to an obese phenotype.	The Journal of clinical investigation 20021215
Novel human histamine H(3) receptor antagonists.	Bioorganic & medicinal chemistry letters 20021118
Coordination of histamine H3 receptor antagonists with human adrenal cytochrome P450 enzymes.	Pharmacology 20021101
Activation of the extraneuronal monoamine transporter (EMT) from rat expressed in 293 cells.	British journal of pharmacology 20021101
Endogenous central histamine-induced reversal of critical haemorrhagic hypotension in rats--studies with histamine N-methyltransferase inhibitor SKF 91488.	Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20021101
Characteristics of recombinantly expressed rat and human histamine H3 receptors.	European journal of pharmacology 20021018
Histamine H3 receptor activation inhibits neurogenic sympathetic vasoconstriction in porcine nasal mucosa.	European journal of pharmacology 20021011
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.	The Journal of pharmacology and experimental therapeutics 20021001
Behavioral characterization of mice lacking histamine H(3) receptors.	Molecular pharmacology 20020801
Different role of the histamine H3-receptor in vagal-, betanechol-, pentagastrin-induced gastric acid secretion in anaesthetized rats.	Scandinavian journal of gastroenterology 20020701
Betahistine dihydrochloride interaction with the histaminergic system in the cat: neurochemical and molecular mechanisms.	European journal of pharmacology 20020620
Effects of N-alpha-methyl-histamine on human H(2) receptors expressed in CHO cells.	Gut 20020601
Histamine H(2) -like receptors in chick cerebral cortex: effects on cyclic AMP synthesis and characterization by [(3) H]tiotidine binding.	Journal of neurochemistry 20020601
Modulation of the discriminative stimulus effects of cocaine and methamphetamine by the histaminergic system.	Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology 20020601
Differential in vivo effects of H3 receptor ligands in a new mouse dipsogenia model.	Pharmacology, biochemistry, and behavior 20020601
Rodent antinociception following acute treatment with different histamine receptor agonists and antagonists.	Pharmacology, biochemistry, and behavior 20020601
Experimental anxiety induced by histaminergics in mast cell-deficient and congenitally normal mice.	Pharmacology, biochemistry, and behavior 20020501
Role of histamine H3 receptors in control of mouse intestinal motility in vivo and in vitro: comparison with alpha2-adrenoceptors.	Digestive diseases and sciences 20020501
Endogenous histamine in the medial septum-diagonal band complex increases the release of acetylcholine from the hippocampus: a dual-probe microdialysis study in the freely moving rat.	The European journal of neuroscience 20020501
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.	The Journal of biological chemistry 20020419
Putative effect of Helicobacter pylori and gastritis on gastric acid secretion in cat.	American journal of physiology. Gastrointestinal and liver physiology 20020401
Effects of histidine, a precursor of histamine, on pentylenetetrazole-induced seizures in rats.	Acta pharmacologica Sinica 20020401
Contractile response of horse deep dorsal penile vein to histamine.	International journal of impotence research 20020401
Evidence for activation of histamine H3 autoreceptors during handling stress in the prefrontal cortex of the rat.	Synapse (New York, N.Y.) 20020315
Histamine excites GABAergic cells in the rat substantia nigra and ventral tegmental area in vitro.	Neuroscience letters 20020308
Hypothalamic histamine neurons activate lipolysis in rat adipose tissue.	Experimental biology and medicine (Maywood, N.J.) 20020301
Histamine regulation of interleukin-18-initiating cytokine cascade is associated with down-regulation of intercellular adhesion molecule-1 expression in human peripheral blood mononuclear cells.	The Journal of pharmacology and experimental therapeutics 20020101
Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.	Molecular pharmacology 20020101
Mouse light/dark box test reveals anxiogenic-like effects by activation of histamine H1 receptors.	Pharmacology, biochemistry, and behavior 20020101
Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.	British journal of pharmacology 20020101
Histamine H3-receptor blockade in the rat nucleus basalis magnocellularis improves place recognition memory.	Psychopharmacology 20020101
Characterisation of the calcium responses to histamine in capsaicin-sensitive and capsaicin-insensitive sensory neurones.	Neuroscience 20020101
Muscarinic, adenosine A(2) and histamine H(3) receptor modulation of haloperidol-induced c-fos expression in the striatum and nucleus accumbens.	Neuroscience 20020101
Influence of SKF 91488, histamine N-methyltransferase inhibitor, on the central cardiovascular regulation during controlled, stepwise hemorrhagic hypotension in rats.	Polish journal of pharmacology 20020101
Identification of a histamine H4 receptor on human eosinophils--role in eosinophil chemotaxis.	Journal of receptor and signal transduction research 20020101
Constitutive activity of histamine h(3) receptors stably expressed in SK-N-MC cells: display of agonism and inverse agonism by H(3) antagonists.	The Journal of pharmacology and experimental therapeutics 20011201
Enhancement by histamine of vascular endothelial growth factor production in granulation tissue via H(2) receptors.	British journal of pharmacology 20011201
Histamine H3 receptor activation inhibits glutamate release from rat striatal synaptosomes.	Neuropharmacology 20011201
Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?	European journal of pharmacology 20011116
Effect of L-carnosine on the hyperglycemia caused by intracranial injection of 2-deoxy-D-glucose in rats.	Neuroscience letters 20011102
Histamine H1 receptors mediate the anorectic action of the pancreatic hormone amylin.	American journal of physiology. Regulatory, integrative and comparative physiology 20011101
Histamine H3 receptor-mediated impairment of contextual fear conditioning and in-vivo inhibition of cholinergic transmission in the rat basolateral amygdala.	The European journal of neuroscience 20011101
Histamine H1 receptor-mediated inhibition of potassium-evoked release of 5-hydroxytryptamine from mouse forebrains.	Behavioural brain research 20011015
Histamine H(3)-receptor antagonism improves memory retention and reverses the cognitive deficit induced by scopolamine in a two-trial place recognition task.	Behavioural brain research 20011015
Involvement of central histamine in amygdaloid kindled seizures in rats.	Behavioural brain research 20011015
Comparison of human, mouse, rat, and guinea pig histamine H4 receptors reveals substantial pharmacological species variation.	The Journal of pharmacology and experimental therapeutics 20011001
Inhibitory effect of histamine on axonal transport in cultured mouse dorsal root ganglion neurons.	Neuroscience research 20011001
Regulation of IL-13 production by histamine in cloned murine T helper type 2 cells.	International immunopharmacology 20011001
Regional differences in functional receptor distribution and calcium mobilization in the intact human lens.	Investigative ophthalmology & visual science 20010901
Histaminergic modulation of GABAergic transmission in rat ventromedial hypothalamic neurones.	The Journal of physiology 20010801
Effects of histamine H3-receptor ligands on brain monoamine oxidase in various mammalian species.	Brain research 20010706
Disturbance of the prejunctional modulation of cholinergic neurotransmission during chronic granulomatous inflammation of the mouse ileum.	British journal of pharmacology 20010701
Novel histaprodifen analogues as potent histamine H1-receptor agonists in the pithed and in the anaesthetized rat.	Naunyn-Schmiedeberg's archives of pharmacology 20010701
[Identification and characterization of histamine H4 receptor].	Nihon yakurigaku zasshi. Folia pharmacologica Japonica 20010701
The H3 receptor is involved in cholecystokinin inhibition of food intake in rats.	Life sciences 20010615
Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists.	European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20010601
Development of a pharmacophore model for histamine H3 receptor antagonists, using the newly developed molecular modeling program SLATE.	Journal of medicinal chemistry 20010524
Activation of histamine H3 receptors inhibits renal noradrenergic neurotransmission in anesthetized dogs.	American journal of physiology. Regulatory, integrative and comparative physiology 20010501
Histamine H(3) receptor-mediated inhibition of depolarization-induced, dopamine D(1) receptor-dependent release of [(3)H]-gamma-aminobutryic acid from rat striatal slices.	British journal of pharmacology 20010501
[Role of central histamine in amygdaloid kindled seizures].	Nihon yakurigaku zasshi. Folia pharmacologica Japonica 20010501
Genomic organization and characterization of splice variants of the human histamine H3 receptor.	The Biochemical journal 20010415
Different antagonist binding properties of human and rat histamine H3 receptors.	Bioorganic & medicinal chemistry letters 20010409
Cognitive enhancing properties of thioperamide infused into the nucleus basalis magnocellularis of the rat.	Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20010401
Histamine and selective H3-receptor ligands: a possible role in the mechanism and management of epilepsy.	Pharmacology, biochemistry, and behavior 20010401
Role of central histaminergic system in lorazepam withdrawal syndrome in rats.	Pharmacology, biochemistry, and behavior 20010401
Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow.	Molecular pharmacology 20010301
Cloning, expression, and pharmacological characterization of a novel human histamine receptor.	Molecular pharmacology 20010301
Cloning and characterization of a novel human histamine receptor.	The Journal of pharmacology and experimental therapeutics 20010301
Histamine H1 and H2 receptor antagonists accelerate skin barrier repair and prevent epidermal hyperplasia induced by barrier disruption in a dry environment.	The Journal of investigative dermatology 20010201
H3 receptor-mediated inhibition of intestinal acetylcholine release: pharmacological characterization of signal transduction pathways.	Naunyn-Schmiedeberg's archives of pharmacology 20010201
The rat H3 receptor: gene organization and multiple isoforms.	Biochemical and biophysical research communications 20010112
Histamine H(3) receptors depress synaptic transmission in the corticostriatal pathway.	Neuropharmacology 20010101
Cortical acetylcholine release elicited by stimulation of histamine H1 receptors in the nucleus basalis magnocellularis: a dual-probe microdialysis study in the freely moving rat.	The European journal of neuroscience 20010101
Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain.	British journal of pharmacology 20001201
Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes.	The Journal of biological chemistry 20001124
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.	Journal of neurochemistry 20000801
Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles.	The Journal of pharmacology and experimental therapeutics 20000601
Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.	Behavioural brain research 19991001
Therapeutic doses of theophylline exert proconvulsant effects in developing mice.	Brain & development 19970901
Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.	Naunyn-Schmiedeberg's archives of pharmacology 19970201
Effect of adenosine and histamine receptor stimulation on canine histamine release to pentagastrin.	Digestion 19970101
Thioperamide, the selective histamine H3 receptor antagonist, attenuates stimulant-induced locomotor activity in the mouse.	European journal of pharmacology 19940701
Modulation of the intracellular and H3-histamine receptors and chemically-induced seizures in mice.	Agents and actions 19940601
Identification of two H3-histamine receptor subtypes.	Molecular pharmacology 19901101

Role of L-carnosine in the control of blood glucose, blood pressure, thermogenesis, and lipolysis by autonomic nerves in rats: involvement of the circadian clock and histamine.

Amino acids 20120701

A bioinformatics search for selective histamine h4 receptor antagonists through structure-based virtual screening strategies.

Chemical biology & drug design 20120501

Effects of neonatal methamphetamine and thioperamide exposure on spatial memory retention and circadian activity later in life.

Behavioural brain research 20120421

Histamine reverses a memory deficit induced in rats by early postnatal maternal deprivation.

Neurobiology of learning and memory 20120101

Ligand based design of novel histamine H₄ receptor antagonists; fragment optimization and analysis of binding kinetics.

Bioorganic & medicinal chemistry letters 20120101

In vivo receptor occupancy assay of histamine H₃ receptor antagonist in rats using non-radiolabeled tracer.

Journal of pharmacological and toxicological methods 20120101

Anti-stress effects of carnosine on restraint-evoked immunocompromise in mice through spleen lymphocyte number maintenance.

PloS one 20120101

Unusual effects of nicotine as a psychostimulant on ambulatory activity in mice.

ISRN pharmacology 20120101

Histamine is a modulator of metamorphic competence in Strongylocentrotus purpuratus (Echinodermata: Echinoidea).

BMC developmental biology 20120101

Desipramine inhibits histamine H1 receptor-induced Ca2+ signaling in rat hypothalamic cells.

PloS one 20120101

Histamine neurons in the tuberomamillary nucleus: a whole center or distinct subpopulations?

Frontiers in systems neuroscience 20120101

Histamine h3 receptor: a novel therapeutic target in alcohol dependence?

Frontiers in systems neuroscience 20120101

Identification and characterization of ZEL-H16 as a novel agonist of the histamine H3 receptor.

PloS one 20120101

The mediation of the central histaminergic system in the pressor effect of intracerebroventricularly injected melittin, a phospholipase A2 activator, in normotensive rats.

Prostaglandins, leukotrienes, and essential fatty acids 20120101

Searching for the Multi-Target-Directed Ligands against Alzheimer's disease: discovery of quinoxaline-based hybrid compounds with AChE, H₃R and BACE 1 inhibitory activities.

Bioorganic & medicinal chemistry 20111201

The role of cortical and hypothalamic histamine-3 receptors in the modulation of central histamine neurotransmission: an in vivo electrophysiology and microdialysis study.

The European journal of neuroscience 20111201

The hydrophobic amino acids in putative helix 8 in carboxy-terminus of histamine H(3) receptor are involved in receptor-G-protein coupling.

Cellular signalling 20111101

Differential modulation of excitatory and inhibitory striatal synaptic transmission by histamine.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20111026

Differential effects of histamine H(3) receptor inverse agonist thioperamide, given alone or in combination with the N-methyl-d-aspartate receptor antagonist dizocilpine, on reconsolidation and consolidation of a contextual fear memory in mice.

Neuroscience 20111013

Histamine facilitates consolidation of fear extinction.

The international journal of neuropsychopharmacology 20111001

In vivo electrochemical evidence for simultaneous 5-HT and histamine release in the rat substantia nigra pars reticulata following medial forebrain bundle stimulation.

Journal of neurochemistry 20110901

Role of the second and third extracellular loops of the histamine H(4) receptor in receptor activation.

Naunyn-Schmiedeberg's archives of pharmacology 20110901

Ontogenetic serotoninergic lesioning alters histaminergic activity in rats in adulthood.

Neurotoxicity research 20110801

Thioperamide, an H₃ receptor antagonist prevents [³H]glucose uptake in brain of adult rats lesioned as neonates with 5,7-dihydroxytryptamine.

Neurotoxicity research 20110701

Involvement of histaminergic receptor mechanisms in the stimulation of NT-3 synthesis in astrocytes.

Neuropharmacology 20110601

Prepulse inhibition of the startle reflex and response to antipsychotic treatments in two outbred mouse strains in comparison to the inbred DBA/2 mouse.

Psychopharmacology 20110601

Memory facilitating effects of agomelatine in the novel object recognition memory paradigm in the rat.

Pharmacology, biochemistry, and behavior 20110601

Histaminergic regulation of seasonal metabolic rhythms in Siberian hamsters.

Physiology & behavior 20110601

Regulation of ERK2 phosphorylation by histamine in splenocytes.

Immunopharmacology and immunotoxicology 20110601

The histamine H3 receptor: from discovery to clinical trials with pitolisant.

British journal of pharmacology 20110601

Effects of histamine H3 receptors on chemical hyperalgesia in diabetic rats.

Neuropharmacology 20110501

N-Alkenyl and cycloalkyl carbamates as dual acting histamine H3 and H4 receptor ligands.

Bioorganic & medicinal chemistry 20110501

Agonist-biased signaling at the histamine H4 receptor: JNJ7777120 recruits β-arrestin without activating G proteins.

Molecular pharmacology 20110401

Newer molecules in the treatment of schizophrenia: A clinical update.

Indian journal of pharmacology 20110401

Triazole ligands reveal distinct molecular features that induce histamine H4 receptor affinity and subtly govern H4/H3 subtype selectivity.

Journal of medicinal chemistry 20110324

Antidiabetic properties of the histamine H3 receptor protean agonist proxyfan.

Endocrinology 20110301

Skin application of urea-containing cream affected cutaneous arterial sympathetic nerve activity, blood flow, and water evaporation.

Skin research and technology : official journal of International Society for Bioengineering and the Skin (ISBS) [and] International Society for Digital Imaging of Skin (ISDIS) [and] International Society for Skin Imaging (ISSI) 20110201

Guinea pig ileum motility stimulation elicited by N-formyl-Met-Leu-Phe (fMLF) involves neurotransmitters and prostanoids.

Peptides 20110201

[Roles of histamine in the exacerbated allergic dermatitis].

Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20110201

Histamine H3 receptor as a drug discovery target.

Journal of medicinal chemistry 20110113

H3 receptors and pain modulation: peripheral, spinal, and brain interactions.

The Journal of pharmacology and experimental therapeutics 20110101

Effects of antihistamines on innate immune responses to severe bacterial infection in mice.

International archives of allergy and immunology 20110101

Histaminergic mechanisms for modulation of memory systems.

Neural plasticity 20110101

Inverse agonism and its therapeutic significance.

Indian journal of pharmacology 20110101

Thioperamide induces CD4 CD25 Foxp3 regulatory T lymphocytes in the lung mucosa of allergic mice through its action on dendritic cells.

Journal of asthma and allergy 20110101

Kv4.2 mediates histamine modulation of preoptic neuron activity and body temperature.

PloS one 20110101

Biological Significance of GPCR Heteromerization in the Neuro-Endocrine System.

Frontiers in endocrinology 20110101

Histamine 3 receptor activation mediates inhibition of acid secretion during Helicobacter-induced gastritis.

World journal of gastrointestinal pathophysiology 20101215

Microinjection of histamine into the dentate gyrus produces antinociception in the formalin test in rats.

Pharmacology, biochemistry, and behavior 20101201

Comparison of the pharmacological properties of human and rat histamine H(3)-receptors.

Biochemical pharmacology 20101101

Structural basis of drug binding to CYP46A1, an enzyme that controls cholesterol turnover in the brain.

The Journal of biological chemistry 20101008

Validation and pharmacological characterisation of MK-801-induced locomotor hyperactivity in BALB/C mice as an assay for detection of novel antipsychotics.

Psychopharmacology 20101001

Histamine H(3) receptor modulates nociception in a rat model of cholestasis.

Pharmacology, biochemistry, and behavior 20100901

Environmental stressors and neurobiological features of marine teleosts: histamine receptors as targets.

Critical reviews in toxicology 20100801

Effect of anserine ingestion on hyperglycemia and the autonomic nerves in rats and humans.

Nutritional neuroscience 20100801

Effect of combined treatment of thioperamide with some antiepileptic drugs on methionine-sulfoximine induced convulsions in mice.

Indian journal of experimental biology 20100801

Histamine H3 receptor activation potentiates peripheral opioid-mediated antinociception: substance P role in peripheral inflammation in mice.

European journal of pharmacology 20100725

Effect of anserine ingestion on the hyperglycemia and autonomic nerves in rats and humans.

Nutritional neuroscience 20100601

Effects of sympathetic histamine on vasomotor responses of blood vessels in rabbit ear to electrical stimulation.

Neuroscience bulletin 20100601

Investigation of the bioactive conformation of histamine H3 receptor antagonists by the cyclopropylic strain-based conformational restriction strategy.

Journal of medicinal chemistry 20100513

Molecular determinants of ligand binding to H4R species variants.

Molecular pharmacology 20100501

Impact of the DRY motif and the missing 'ionic lock' on constitutive activity and G-protein coupling of the human histamine H4 receptor.

The Journal of pharmacology and experimental therapeutics 20100501

Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists.

Bioorganic & medicinal chemistry letters 20100415

Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.

Journal of medicinal chemistry 20100325

Modulation of histamine H(3) receptor function by monovalent ions.

Neuroscience letters 20100319

Neuropharmacology of vestibular system disorders.

Current neuropharmacology 20100301

Modeling G protein-coupled receptors for structure-based drug discovery using low-frequency normal modes for refinement of homology models: application to H3 antagonists.

Proteins 20100201

Synthesis and structural and pharmacological properties of cyclopropane-based conformationally restricted analogs of 4-methylhistamine as histamine H3/H4 receptor ligands.

Bioorganic & medicinal chemistry 20100201

Involvement of the histaminergic system in cytidine 5'-diphosphocholine-induced reversal of critical haemorrhagic hypotension in rats.

Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20100201

Effects of anserine on the renal sympathetic nerve activity and blood pressure in urethane-anesthetized rats.

Physiological research 20100101

Oral L-histidine exerts antihypertensive effects via central histamine H3 receptors and decreases nitric oxide content in the rostral ventrolateral medulla in spontaneously hypertensive rats.

Clinical and experimental pharmacology & physiology 20100101

Contribution of mast cells to the oedema induced by Bothrops moojeni snake venom and a pharmacological assessment of the inflammatory mediators involved.

Toxicon : official journal of the International Society on Toxinology 20100101

Pretreatment with l-histidine produces a shift from methamphetamine-induced stereotypical biting to persistent locomotion in mice.

Pharmacology, biochemistry, and behavior 20100101

R-(-)-alpha-methylhistamine, a histamine H3 receptor agonist, induces endothelium-dependent vasodilation in rat mesenteric resistance arteries.

Biological & pharmaceutical bulletin 20100101

Different role of cAMP dependent protein kinase and CaMKII in H3 receptor regulation of histamine synthesis and release.

Neuroscience 20091215

The effects of thioperamide on extracellular levels of glutamate and GABA in the rat prefrontal cortex.

Psychopharmacology 20091201

Histamine H3 and H4 receptor affinity of branched 3-(1H-imidazol-4-yl)propyl N-alkylcarbamates.

Bioorganic & medicinal chemistry letters 20091201

Heterocyclic replacement of the central phenyl core of diamine-based histamine H3 receptor antagonists.

European journal of medicinal chemistry 20091101

Interactions of histamine H1-receptor agonists and antagonists with the human histamine H4-receptor.

Molecular pharmacology 20091101

Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H4 receptor agonists.

Journal of medicinal chemistry 20091022

2,4-Diaminopyrimidines as histamine H4 receptor ligands--Scaffold optimization and pharmacological characterization.

Bioorganic & medicinal chemistry 20091015

Diamine-based human histamine H3 receptor antagonists: (4-aminobutyn-1-yl)benzylamines.

European journal of medicinal chemistry 20091001

Effects of the H(3) antagonist, thioperamide, on behavioral alterations induced by systemic MK-801 administration in rats.

Psychopharmacology 20090901

Enhanced morphine-induced antinociception in histamine H3 receptor gene knockout mice.

Neuropharmacology 20090901

Anxiolytic-like profiles of histamine H3 receptor agonists in animal models of anxiety: a comparative study with antidepressants and benzodiazepine anxiolytic.

Psychopharmacology 20090801

Development of a selective and potent radioactive ligand for histamine H(3) receptors: A compound potentially useful for receptor occupancy studies.

Bioorganic & medicinal chemistry letters 20090801

JNJ-10181457, a selective non-imidazole histamine H(3) receptor antagonist, normalizes acetylcholine neurotransmission and has efficacy in translational rat models of cognition.

Neuropharmacology 20090601

Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studies.

Bioorganic & medicinal chemistry 20090601

Heterogeneity of histaminergic neurons in the tuberomammillary nucleus of the rat.

The European journal of neuroscience 20090601

N(G)-acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.

Journal of medicinal chemistry 20090423

Non-imidazole histamine H3 ligands, part IV: SAR of 1-[2-thiazol-5-yl-(2-aminoethyl)]-4-n-propylpiperazine derivatives.

European journal of medicinal chemistry 20090401

Characterization of histamine-induced relaxation in pre-contracted rat aorta.

Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20090401

Histaminergic activity in a rodent model of Parkinson's disease.

Neurotoxicity research 20090401

Effects of the H3 receptor inverse agonist thioperamide on cocaine-induced locomotion in mice: role of the histaminergic system and potential pharmacokinetic interactions.

Psychopharmacology 20090301

The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.

Behavioural pharmacology 20090301

High constitutive activity and a G-protein-independent high-affinity state of the human histamine H(4)-receptor.

Biochemistry 20090217

Autonomic and cardiovascular effects of central neuromedin U in rats.

Physiology & behavior 20090216

Possible role of the histaminergic system in autonomic and cardiovascular responses to neuropeptide Y.

Neuropeptides 20090201

H3 receptor antagonists reverse delay-dependent deficits in novel object discrimination by enhancing retrieval.

Psychopharmacology 20090101

Modification of the picryl chloride-induced allergic dermatitis model in mouse ear lobes by 12-O-tetradecanoylphorbol 13-acetate, and analysis of the role of histamine in the modified model.

International archives of allergy and immunology 20090101

L-histidine enhances learning in stressed zebrafish.

Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20090101

Cytokine responses of intraepithelial lymphocytes are regulated by histamine H(2) receptor.

Journal of gastroenterology 20090101

A novel flow cytometric high throughput assay for a systematic study on molecular mechanisms underlying T cell receptor-mediated integrin activation.

PloS one 20090101

Alpha2 adrenoceptors modulate histamine release from sympathetic nerves in the guinea pig vas deferens.

Neuropharmacology 20090101

H4 histamine receptors mediate cell cycle arrest in growth factor-induced murine and human hematopoietic progenitor cells.

PloS one 20090101

Modulatory effects of histamine on cat carotid body chemoreception.

Respiratory physiology & neurobiology 20081231

Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach.

Journal of medicinal chemistry 20081225

Role of histamine in short- and long-term effects of methamphetamine on the developing mouse brain.

Journal of neurochemistry 20081101

Biphasic effects of orexin-A on autonomic nerve activity and lipolysis.

Neuroscience letters 20081024

Effect of thioperamide on oxidative stress markers in middle cerebral artery occlusion model of focal cerebral ischemia in rats.

Human & experimental toxicology 20081001

The alkaloid conessine and analogues as potent histamine H3 receptor antagonists.

Journal of medicinal chemistry 20080911

Electrophysiology-based analysis of human histamine H(4) receptor pharmacology using GIRK channel coupling in Xenopus oocytes.

European journal of pharmacology 20080904

Localization and function of histamine H3 receptor in the nasal mucosa.

Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20080901

Alleviation of ischemia-induced brain edema by activation of the central histaminergic system in rats.

Journal of pharmacological sciences 20080901

Regulation of sympathetic nerve activity by L-carnosine in mammalian white adipose tissue.

Neuroscience letters 20080815

Discovery of novel human histamine H4 receptor ligands by large-scale structure-based virtual screening.

Journal of medicinal chemistry 20080612

Correlation between ex vivo receptor occupancy and wake-promoting activity of selective H3 receptor antagonists.

The Journal of pharmacology and experimental therapeutics 20080601

Blocking histamine H(1) improves learning and mnemonic dysfunction in mice with social isolation plus repeated methamphetamine injection.

Journal of pharmacological sciences 20080601

Zebrafish: An in vivo model for the study of neurological diseases.

Neuropsychiatric disease and treatment 20080601

Narcolepsy: current treatment options and future approaches.

Neuropsychiatric disease and treatment 20080601

Interactions between histamine H3 and dopamine D2 receptors and the implications for striatal function.

Neuropharmacology 20080516

Fragment based design of new H4 receptor-ligands with anti-inflammatory properties in vivo.

Journal of medicinal chemistry 20080424

Histamine action on vertebrate GABAA receptors: direct channel gating and potentiation of GABA responses.

The Journal of biological chemistry 20080418

Role of histamine in brain protection in surgical brain injury in mice.

Brain research 20080418

Effects of oolong tea on renal sympathetic nerve activity and spontaneous hypertension in rats.

Metabolism: clinical and experimental 20080401

Ontogenetic noradrenergic lesion alters histaminergic activity in adult rats.

Neurotoxicity research 20080401

Specific cerebral heat shock proteins and histamine receptor cross-talking mechanisms promote distinct lead-dependent neurotoxic responses in teleosts.

Toxicology and applied pharmacology 20080301

Comparative effects of olanzapine and ziprasidone on hypophagia induced by enhanced histamine neurotransmission in the rat.

Behavioural pharmacology 20080301

Carnosine protects against Abeta42-induced neurotoxicity in differentiated rat PC12 cells.

Cellular and molecular neurobiology 20080201

Effects of central histamine receptors blockade on GABA(A) agonist-induced food intake in broiler cockerels.

Pakistan journal of biological sciences : PJBS 20080201

Antigen inhalation induces mast cells and eosinophils infiltration in the guinea pig esophageal epithelium involving histamine-mediated pathway.

Life sciences 20080130

Distinctive role of central histamine H3 receptor in various orexigenic pathways.

European journal of pharmacology 20080128

CSF histamine levels in rats reflect the central histamine neurotransmission.

Neuroscience letters 20080117

Modulation of hippocampal theta oscillation by histamine H3 receptors.

The Journal of pharmacology and experimental therapeutics 20080101

Mast cell-derived histamine mediates cystitis pain.

PloS one 20080101

Histamine H(3) receptor ligands modulate L-dopa-evoked behavioral responses and L-dopa derived extracellular dopamine in dopamine-denervated rat striatum.

Neurotoxicity research 20080101

Antagonist affinity measurements at the Gi-coupled human histamine H3 receptor expressed in CHO cells.

BMC pharmacology 20080101

Histamine-induced itch and its relationship with pain.

Molecular pain 20080101

The possible involvement of hyperpolarizing mechanisms in histamine-induced relaxation of the rat portal vein.

Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi 20080101

Histamine in Macaca mulatto monkey cardiac sympathetic nerve system: a morphological and functional assessment.

Autonomic neuroscience : basic & clinical 20071230

Functional expression of H4 histamine receptor in human natural killer cells, monocytes, and dendritic cells.

Journal of immunology (Baltimore, Md. : 1950) 20071201

The role of carcinine in signaling at the Drosophila photoreceptor synapse.

PLoS genetics 20071201

Activation of peripheral and spinal histamine H3 receptors inhibits formalin-induced inflammation and nociception, respectively.

Pharmacology, biochemistry, and behavior 20071101

Reduced histamine levels and H3 receptor antagonist-induced histamine release in the amygdala of Apoe-/- mice.

Journal of neurochemistry 20071001

The Akt/GSK-3beta axis as a new signaling pathway of the histamine H(3) receptor.

Journal of neurochemistry 20071001

Histamine improves antigen uptake and cross-presentation by dendritic cells.

Journal of immunology (Baltimore, Md. : 1950) 20070915

Interaction of nicotinic and histamine H(3) systems in the radial-arm maze repeated acquisition task.

European journal of pharmacology 20070813

Betahistine in the treatment of Ménière's disease.

Neuropsychiatric disease and treatment 20070801

Histaminergic ligands improve vestibular compensation in the cat: behavioural, neurochemical and molecular evidence.

European journal of pharmacology 20070730

Blockade of brain histamine metabolism alters methamphetamine-induced expression pattern of stereotypy in mice via histamine H1 receptors.

Neuroscience 20070713

Histamine H4 receptor agonists have more activities than H4 agonism in antigen-specific human T-cell responses.

Immunology 20070601

Interaction of calcitonin gene-related peptide, nitric oxide and histamine release in neurogenic blood flow and afferent activation in the rat cranial dura mater.

Cephalalgia : an international journal of headache 20070601

H3 histamine receptor agonist inhibits biliary growth of BDL rats by downregulation of the cAMP-dependent PKA/ERK1/2/ELK-1 pathway.

Laboratory investigation; a journal of technical methods and pathology 20070501

Histaminergic H1 receptors mediate L-histidine-induced anxiety in elevated plus-maze test in mice.

Behavioural pharmacology 20070501

Identification of zebrafish histamine H1, H2 and H3 receptors and effects of histaminergic ligands on behavior.

Biochemical pharmacology 20070415

The brain H3-receptor as a novel therapeutic target for vigilance and sleep-wake disorders.

Biochemical pharmacology 20070415

Auditory stimulation affects renal sympathetic nerve activity and blood pressure in rats.

Neuroscience letters 20070412

Thioperamide reduces intracellular calcium in mouse brain synaptosomes.

European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20070401

Influence of the H3/H4 receptor antagonist, thioperamide on regional haemodynamics in rats with trinitrobenzene sulfonic acid-induced colitis.

Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20070401

Thioperamide delays vestibular compensation in goldfish.

Neuroscience letters 20070326

Sex- and histamine-dependent long-term cognitive effects of methamphetamine exposure.

Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20070301

Carnosine protects against NMDA-induced neurotoxicity in differentiated rat PC12 cells through carnosine-histidine-histamine pathway and H(1)/H(3) receptors.

Biochemical pharmacology 20070301

Histamine affects STAT6 phosphorylation via its effects on IL-4 secretion: role of H1 receptors in the regulation of IL-4 production.

International immunopharmacology 20070301

Suppression of inflammatory cell recruitment by histamine receptor stimulation in ischemic rat brains.

European journal of pharmacology 20070227

Involvement of the histaminergic system in renal sympathetic and cardiovascular responses to leptin and ghrelin.

Neuroscience letters 20070208

In vitro pharmacology at human histamine H3 receptors and brain access of non-imidazole alkylpiperidine derivatives.

Pharmacological research 20070201

Modification of formalin-induced nociception by different histamine receptor agonists and antagonists.

European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20070115

Role of apolipoprotein E in anxiety.

Neural plasticity 20070101

Role of histamine H3 and H4 receptors in mechanical hyperalgesia following peripheral nerve injury.

Neuroimmunomodulation 20070101

Histamine H3 receptor agonist- and antagonist-evoked vacuous chewing movements in 6-OHDA-lesioned rats occurs in an absence of change in microdialysate dopamine levels.

European journal of pharmacology 20061215

Feeding differences in pubertal and aged golden hamsters (Mesocricetus auratus) are related to specific cerebral expression pattern of histamine subtype 3 receptor.

Behavioral neuroscience 20061201

Expression of histamine receptors and effect of histamine in the rat carotid body chemoafferent pathway.

The European journal of neuroscience 20061201

Mechanism of imipramine-induced seizures in amygdala-kindled rats.

Epilepsy research 20061101

Renoprotective effects of l-carnosine on ischemia/reperfusion-induced renal injury in rats.

The Journal of pharmacology and experimental therapeutics 20061101

Dose-different effects of orexin-A on the renal sympathetic nerve and blood pressure in urethane-anesthetized rats.

Experimental biology and medicine (Maywood, N.J.) 20061101

A comparison of protective effects between L-histidine and hypothermia against ischemia-induced neuronal damage in gerbil hippocampus.

European journal of pharmacology 20060928

Stereochemical diversity-oriented conformational restriction strategy. Development of potent histamine H3 and/or H4 receptor antagonists with an imidazolylcyclopropane structure.

Journal of medicinal chemistry 20060907

Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway.

Neuropharmacology 20060901

Suppression of ischemia/reperfusion liver injury by histamine H4 receptor stimulation in rats.

European journal of pharmacology 20060821

Homologous down-regulation of histamine H3 receptors in rat striatal slices.

Synapse (New York, N.Y.) 20060801

Antipsychotic-like profile of thioperamide, a selective H3-receptor antagonist in mice.

Fundamental & clinical pharmacology 20060801

Evidence for histamine as a neurotransmitter in the cardiac sympathetic nervous system.

American journal of physiology. Heart and circulatory physiology 20060701

Histamine enhances inhibitory avoidance memory consolidation through a H2 receptor-dependent mechanism.

Neurobiology of learning and memory 20060701

Impaired drinking response in histamine H3 receptor knockout mice following dehydration or angiotensin-II challenge.

Pharmacology, biochemistry, and behavior 20060701

Increasing synaptic noradrenaline, serotonin and histamine enhances in vivo binding of phosphodiesterase-4 inhibitor (R)-[11C]rolipram in rat brain, lung and heart.

Life sciences 20060620

Changes in the histaminergic system during vestibular compensation in the cat.

The Journal of physiology 20060615

The effect of histamine on field-stimulated contractions of the guinea-pig prostate.

Naunyn-Schmiedeberg's archives of pharmacology 20060601

Histamine-induced enhancement of vasopressin and oxytocin secretion in rat neurohypophyseal tissue cultures.

Regulatory peptides 20060515

Olfactory stimulation with scent of lavender oil affects autonomic neurotransmission and blood pressure in rats.

Neuroscience letters 20060501

Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.

British journal of pharmacology 20060401

Effects of the H3-receptor inverse agonist thioperamide on the psychomotor effects induced by acutely and repeatedly given cocaine in C57BL/6J mice.

Pharmacology, biochemistry, and behavior 20060401

Effects of histamine H(3) antagonists and donepezil on learning and mnemonic deficits induced by pentylenetetrazol kindling in weanling mice.

Neuropharmacology 20060301

Role of H1 receptors in histamine-mediated up-regulation of STAT4 phosphorylation.

International immunopharmacology 20060301

Histamine protects against NMDA-induced necrosis in cultured cortical neurons through H receptor/cyclic AMP/protein kinase A and H receptor/GABA release pathways.

Journal of neurochemistry 20060301

Histamine increases sickle erythrocyte adherence to endothelium.

British journal of haematology 20060201

[The effect of central histamine H3 receptor on breathing activity of asthmatic guinea pigs].

Zhongguo ying yong sheng li xue za zhi = Zhongguo yingyong shenglixue zazhi = Chinese journal of applied physiology 20060201

Histaminergic neurons protect the developing hippocampus from kainic acid-induced neuronal damage in an organotypic coculture system.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20060125

The hallucinogenic herb Salvia divinorum and its active ingredient salvinorin A inhibit enteric cholinergic transmission in the guinea-pig ileum.

Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20060101

Histamine receptors influence blood-spinal cord barrier permeability, edema formation, and spinal cord blood flow following trauma to the rat spinal cord.

Acta neurochirurgica. Supplement 20060101

Aversive memory reactivation engages in the amygdala only some neurotransmitters involved in consolidation.

Learning & memory (Cold Spring Harbor, N.Y.) 20060101

Reduction in brain infarction by augmentation of central histaminergic activity in rats.

Brain research 20051220

Histamine (H3) receptors modulate the excitatory amino acid receptor response of the vestibular afferents.

Brain research 20051207

Effects of intraduodenal injection of Lactobacillus johnsonii La1 on renal sympathetic nerve activity and blood pressure in urethane-anesthetized rats.

Neuroscience letters 20051202

Mechanisms of histamine-induced relaxation in bovine small adrenal cortical arteries.

American journal of physiology. Endocrinology and metabolism 20051201

Sleep disturbances, psychiatric disorders, and psychotropic drugs.

Dialogues in clinical neuroscience 20051201

Some environmental contaminants influence motor and feeding behaviors in the ornate wrasse (Thalassoma pavo) via distinct cerebral histamine receptor subtypes.

Environmental health perspectives 20051101

The histaminergic signaling system exerts a neuroprotective role against neurodegenerative-induced processes in the hamster.

The Journal of pharmacology and experimental therapeutics 20051001

Modulation of spontaneous alternation performance of mice treated with thioperamide and tacrine in a cross maze task.

Fundamental & clinical pharmacology 20051001

Effect of thioperamide on modified forced swimming test-induced oxidative stress in mice.

Basic & clinical pharmacology & toxicology 20051001

Olfactory stimulation with scent of lavender oil affects autonomic nerves, lipolysis and appetite in rats.

Neuroscience letters 20050701

Involvement of histamine H1 and H2 receptors in the regulation of STAT-1 phosphorylation: inverse agonism exhibited by the receptor antagonists.

International immunopharmacology 20050701

Histamine excites noradrenergic neurons in locus coeruleus in rats.

Neuropharmacology 20050701

Histamine-3 receptor antagonists reduce superoxide anion generation and lipid peroxidation in rat brain homogenates.

The Journal of pharmacy and pharmacology 20050601

Generation of cell lines for drug discovery through random activation of gene expression: application to the human histamine H3 receptor.

Assay and drug development technologies 20050601

Lack of cataleptogenic potentiation with non-imidazole H3 receptor antagonists reveals potential drug-drug interactions between imidazole-based H3 receptor antagonists and antipsychotic drugs.

Brain research 20050531

The H3 antagonist thioperamide reveals conditioned preference for a context associated with an inactive small dose of cocaine in C57BL/6J mice.

Behavioural brain research 20050507

Effects of histamine H3 receptor antagonists in two models of spatial learning.

Behavioural brain research 20050430

Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H3 receptor antagonist.

The Journal of pharmacology and experimental therapeutics 20050401

4-phenoxypiperidines: potent, conformationally restricted, non-imidazole histamine H3 antagonists.

Journal of medicinal chemistry 20050324

Effect of combined histamine H1 and H3 receptor blockade on cutaneous microvascular permeability elicited by compound 48/80.

Life sciences 20050304

Histamine receptors that influence blockage of the normal human nasal airway.

British journal of pharmacology 20050301

Assessment of pharmacology and potential anti-obesity properties of H3 receptor antagonists/inverse agonists.

Expert opinion on investigational drugs 20050301

Dose-dependent effects of L-carnosine on the renal sympathetic nerve and blood pressure in urethane-anesthetized rats.

American journal of physiology. Regulatory, integrative and comparative physiology 20050201

A biochemical and pharmacological examination of Rhamphiophis oxyrhynchus (Rufous beaked snake) venom.

Toxicon : official journal of the International Society on Toxinology 20050201

Role of capsaicin-sensitive nerves and histamine H1, H2, and H3 receptors in the gastroprotective effect of histamine against stress ulcers in rats.

European journal of pharmacology 20050131

4-(2-[2-(2(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and related 2-aminoethylbenzofuran H3 receptor antagonists potently enhance cognition and attention.

Journal of medicinal chemistry 20050113

2-(4-alkylpiperazin-1-yl)quinolines as a new class of imidazole-free histamine H3 receptor antagonists.

Journal of medicinal chemistry 20050113

Histaminergic modulation of excitatory synaptic transmission in the rat basolateral amygdala.

Neuroscience 20050101

Histamine-induced cyclic AMP formation in the chick hypothalamus: interaction with vasoactive intestinal peptide.

Pharmacological reports : PR 20050101

[Participation of cyclic nucleotides and phospholipidis in signal transduction of histamin receptor H3 of the gastric mucosa parietal cells in rats with experimental ulcer].

Ukrains'kyi biokhimichnyi zhurnal (1999 ) 20050101

Role of histaminergic neurons in development of epileptic seizures in EL mice.

Brain research. Molecular brain research 20041206

Unusual functional properties of homo- and heteromultimeric histamine-gated chloride channels of Drosophila melanogaster: spontaneous currents and dual gating by GABA and histamine.

Neuroscience letters 20041130

Pharmacological effects of carcinine on histaminergic neurons in the brain.

British journal of pharmacology 20041101

Medicinal chemical and pharmacological aspects of imidazole-containing histamine H3 receptor antagonists.

Mini reviews in medicinal chemistry 20041101

Role of the histamine system in nefopam-induced antinociception in mice.

European journal of pharmacology 20041025

Histamine H3 receptors inhibit serotonin release in substantia nigra pars reticulata.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20041006

Intranigral injection of the H3 agonist immepip and systemic apomorphine elicit ipsilateral turning behaviour in naive rats, but reduce contralateral turning in hemiparkinsonian rats.

Behavioural brain research 20041005

The in vitro and in vivo pharmacological activity of Boiga dendrophila (mangrove catsnake) venom.

Autonomic & autacoid pharmacology 20041001

Histamine H3 antagonist thioperamide dose-dependently enhances memory consolidation and reverses amnesia induced by dizocilpine or scopolamine in a one-trial inhibitory avoidance task in mice.

Behavioural brain research 20040923

Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist.

Biochemical pharmacology 20040901

Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.

Journal of neurochemistry 20040901

Enhancement of prepulse inhibition of startle in mice by the H3 receptor antagonists thioperamide and ciproxifan.

Behavioural brain research 20040812

Liver-expressed chemokine/CC chemokine ligand 16 attracts eosinophils by interacting with histamine H4 receptor.

Journal of immunology (Baltimore, Md. : 1950) 20040801

Histamine H3 receptor activation inhibits dopamine D1 receptor-induced cAMP accumulation in rat striatal slices.

Neuroscience letters 20040708

Critical role of L-selectin and histamine H4 receptor in zymosan-induced neutrophil recruitment from the bone marrow: comparison with carrageenan.

The Journal of pharmacology and experimental therapeutics 20040701

Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain.

Journal of medicinal chemistry 20040603

Central H3R activation by thioperamide does not affect energy balance.

Pharmacology, biochemistry, and behavior 20040601

1-alkyl-4-acylpiperazines as a new class of imidazole-free histamine H(3) receptor antagonists.

Journal of medicinal chemistry 20040520

4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists.

Journal of medicinal chemistry 20040506

Involvement of histamine H4 and H1 receptors in scratching induced by histamine receptor agonists in Balb C mice.

British journal of pharmacology 20040501

Histamine H4 receptor mediates eosinophil chemotaxis with cell shape change and adhesion molecule upregulation.

British journal of pharmacology 20040501

Intracerebroventricular administration of histamine H3 receptor antagonists decreases seizures in rat models of epilepsia.

Methods and findings in experimental and clinical pharmacology 20040501

Histamine h3 receptor antagonists potentiate methamphetamine self-administration and methamphetamine-induced accumbal dopamine release.

Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040401

Inhibitory effect of iodophenpropit, a selective histamine H3 antagonist, on amygdaloid kindled seizures.

Brain research bulletin 20040315

Pruritus-associated response mediated by cutaneous histamine H3 receptors.

Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20040301

Thioperamide-elicited increase of histamine release from basolateral amygdala of freely moving rats and its therapeutic implications.

Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20040301

Role of histamine H3 receptors during ischemia/reperfusion in isolated rat hearts.

Journal of cardiovascular pharmacology 20040301

Plasticity of histamine H3 receptor expression and binding in the vestibular nuclei after labyrinthectomy in rat.

BMC neuroscience 20040101

Critical role of histamine H4 receptor in leukotriene B4 production and mast cell-dependent neutrophil recruitment induced by zymosan in vivo.

The Journal of pharmacology and experimental therapeutics 20031201

Role of histamine receptors in the regulation of edema and circulation postburn.

Burns : journal of the International Society for Burn Injuries 20031201

Histamine induces cytoskeletal changes in human eosinophils via the H(4) receptor.

British journal of pharmacology 20031101

Possible role of L-carnosine in the regulation of blood glucose through controlling autonomic nerves.

Experimental biology and medicine (Maywood, N.J.) 20031101

Generation and characterization of highly constitutive active histamine H3 receptors.

The Journal of pharmacology and experimental therapeutics 20031001

Aminergic control of high-frequency (approximately 200 Hz) network oscillations in the hippocampus of the behaving rat.

Neuroscience letters 20030911

The first potent and selective non-imidazole human histamine H4 receptor antagonists.

Journal of medicinal chemistry 20030911

Central endogenous histamine modulates sympathetic outflow through H3 receptors in the conscious rabbit.

British journal of pharmacology 20030701

Identification of a dual histamine H1/H3 receptor ligand based on the H1 antagonist chlorpheniramine.

Bioorganic & medicinal chemistry letters 20030616

Antinociceptive mechanisms of orally administered decursinol in the mouse.

Life sciences 20030613

Activation of spinal histamine H3 receptors inhibits mechanical nociception.

European journal of pharmacology 20030606

Two novel and selective nonimidazole H3 receptor antagonists A-304121 and A-317920: II. In vivo behavioral and neurophysiological characterization.

The Journal of pharmacology and experimental therapeutics 20030601

Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects.

The Journal of pharmacology and experimental therapeutics 20030601

Histamine H4 receptor mediates chemotaxis and calcium mobilization of mast cells.

The Journal of pharmacology and experimental therapeutics 20030601

H3 receptor blockade by thioperamide enhances cognition in rats without inducing locomotor sensitization.

Psychopharmacology 20030601

Cyclopropane-based conformational restriction of histamine. (1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a highly selective agonist for the histamine H3 receptor, having a cis-cyclopropane structure.

Journal of medicinal chemistry 20030508

Regulation by prostaglandin E2 and histamine of angiogenesis in inflammatory granulation tissue.

Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20030501

Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds.

Journal of medicinal chemistry 20030410

Histamine inhibits lipopolysaccharide-induced tumor necrosis factor-alpha production in an intercellular adhesion molecule-1- and B7.1-dependent manner.

The Journal of pharmacology and experimental therapeutics 20030201

Histaminergic modulation of the intact respiratory network of adult mice.

Pflugers Archiv : European journal of physiology 20030201

Histamine-induced chloride secretion is mediated via H2-receptors in the pig proximal colon.

Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20030201

Neuroimmune interactions in guinea pig stomach and small intestine.

American journal of physiology. Gastrointestinal and liver physiology 20030101

Functional identification of epithelial and smooth muscle histamine-dependent relaxing mechanisms in the bovine trachea, but not in bronchi.

Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20030101

Replacement of imidazole by a piperidine moiety differentially affects the potency of histamine H3-receptor antagonists.

Naunyn-Schmiedeberg's archives of pharmacology 20030101

High-frequency oscillation in the hippocampus of the behaving rat and its modulation by the histaminergic system.

Hippocampus 20030101

Contribution of the histaminergic receptor subtypes to histamine-induced cerebellar granular neurotoxicity.

Polish journal of pharmacology 20030101

Targeted disruption of H3 receptors results in changes in brain histamine tone leading to an obese phenotype.

The Journal of clinical investigation 20021215

Novel human histamine H(3) receptor antagonists.

Bioorganic & medicinal chemistry letters 20021118

Coordination of histamine H3 receptor antagonists with human adrenal cytochrome P450 enzymes.

Pharmacology 20021101

Activation of the extraneuronal monoamine transporter (EMT) from rat expressed in 293 cells.

British journal of pharmacology 20021101

Endogenous central histamine-induced reversal of critical haemorrhagic hypotension in rats--studies with histamine N-methyltransferase inhibitor SKF 91488.

Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20021101

Characteristics of recombinantly expressed rat and human histamine H3 receptors.

European journal of pharmacology 20021018

Histamine H3 receptor activation inhibits neurogenic sympathetic vasoconstriction in porcine nasal mucosa.

European journal of pharmacology 20021011

Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.

The Journal of pharmacology and experimental therapeutics 20021001

Behavioral characterization of mice lacking histamine H(3) receptors.

Molecular pharmacology 20020801

Different role of the histamine H3-receptor in vagal-, betanechol-, pentagastrin-induced gastric acid secretion in anaesthetized rats.

Scandinavian journal of gastroenterology 20020701

Betahistine dihydrochloride interaction with the histaminergic system in the cat: neurochemical and molecular mechanisms.

European journal of pharmacology 20020620

Effects of N-alpha-methyl-histamine on human H(2) receptors expressed in CHO cells.

Gut 20020601

Histamine H(2) -like receptors in chick cerebral cortex: effects on cyclic AMP synthesis and characterization by [(3) H]tiotidine binding.

Journal of neurochemistry 20020601

Modulation of the discriminative stimulus effects of cocaine and methamphetamine by the histaminergic system.

Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology 20020601

Differential in vivo effects of H3 receptor ligands in a new mouse dipsogenia model.

Pharmacology, biochemistry, and behavior 20020601

Rodent antinociception following acute treatment with different histamine receptor agonists and antagonists.

Pharmacology, biochemistry, and behavior 20020601

Experimental anxiety induced by histaminergics in mast cell-deficient and congenitally normal mice.

Pharmacology, biochemistry, and behavior 20020501

Role of histamine H3 receptors in control of mouse intestinal motility in vivo and in vitro: comparison with alpha2-adrenoceptors.

Digestive diseases and sciences 20020501

Endogenous histamine in the medial septum-diagonal band complex increases the release of acetylcholine from the hippocampus: a dual-probe microdialysis study in the freely moving rat.

The European journal of neuroscience 20020501

Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.

The Journal of biological chemistry 20020419

Putative effect of Helicobacter pylori and gastritis on gastric acid secretion in cat.

American journal of physiology. Gastrointestinal and liver physiology 20020401

Effects of histidine, a precursor of histamine, on pentylenetetrazole-induced seizures in rats.

Acta pharmacologica Sinica 20020401

Contractile response of horse deep dorsal penile vein to histamine.

International journal of impotence research 20020401

Evidence for activation of histamine H3 autoreceptors during handling stress in the prefrontal cortex of the rat.

Synapse (New York, N.Y.) 20020315

Histamine excites GABAergic cells in the rat substantia nigra and ventral tegmental area in vitro.

Neuroscience letters 20020308

Hypothalamic histamine neurons activate lipolysis in rat adipose tissue.

Experimental biology and medicine (Maywood, N.J.) 20020301

Histamine regulation of interleukin-18-initiating cytokine cascade is associated with down-regulation of intercellular adhesion molecule-1 expression in human peripheral blood mononuclear cells.

The Journal of pharmacology and experimental therapeutics 20020101

Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.

Molecular pharmacology 20020101

Mouse light/dark box test reveals anxiogenic-like effects by activation of histamine H1 receptors.

Pharmacology, biochemistry, and behavior 20020101

Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

British journal of pharmacology 20020101

Histamine H3-receptor blockade in the rat nucleus basalis magnocellularis improves place recognition memory.

Psychopharmacology 20020101

Characterisation of the calcium responses to histamine in capsaicin-sensitive and capsaicin-insensitive sensory neurones.

Neuroscience 20020101

Muscarinic, adenosine A(2) and histamine H(3) receptor modulation of haloperidol-induced c-fos expression in the striatum and nucleus accumbens.

Neuroscience 20020101

Influence of SKF 91488, histamine N-methyltransferase inhibitor, on the central cardiovascular regulation during controlled, stepwise hemorrhagic hypotension in rats.

Polish journal of pharmacology 20020101

Identification of a histamine H4 receptor on human eosinophils--role in eosinophil chemotaxis.

Journal of receptor and signal transduction research 20020101

Constitutive activity of histamine h(3) receptors stably expressed in SK-N-MC cells: display of agonism and inverse agonism by H(3) antagonists.

The Journal of pharmacology and experimental therapeutics 20011201

Enhancement by histamine of vascular endothelial growth factor production in granulation tissue via H(2) receptors.

British journal of pharmacology 20011201

Histamine H3 receptor activation inhibits glutamate release from rat striatal synaptosomes.

Neuropharmacology 20011201

Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?

European journal of pharmacology 20011116

Effect of L-carnosine on the hyperglycemia caused by intracranial injection of 2-deoxy-D-glucose in rats.

Neuroscience letters 20011102

Histamine H1 receptors mediate the anorectic action of the pancreatic hormone amylin.

American journal of physiology. Regulatory, integrative and comparative physiology 20011101

Histamine H3 receptor-mediated impairment of contextual fear conditioning and in-vivo inhibition of cholinergic transmission in the rat basolateral amygdala.

The European journal of neuroscience 20011101

Histamine H1 receptor-mediated inhibition of potassium-evoked release of 5-hydroxytryptamine from mouse forebrains.

Behavioural brain research 20011015

Histamine H(3)-receptor antagonism improves memory retention and reverses the cognitive deficit induced by scopolamine in a two-trial place recognition task.

Behavioural brain research 20011015

Involvement of central histamine in amygdaloid kindled seizures in rats.

Behavioural brain research 20011015

Comparison of human, mouse, rat, and guinea pig histamine H4 receptors reveals substantial pharmacological species variation.

The Journal of pharmacology and experimental therapeutics 20011001

Inhibitory effect of histamine on axonal transport in cultured mouse dorsal root ganglion neurons.

Neuroscience research 20011001

Regulation of IL-13 production by histamine in cloned murine T helper type 2 cells.

International immunopharmacology 20011001

Regional differences in functional receptor distribution and calcium mobilization in the intact human lens.

Investigative ophthalmology & visual science 20010901

Histaminergic modulation of GABAergic transmission in rat ventromedial hypothalamic neurones.

The Journal of physiology 20010801

Effects of histamine H3-receptor ligands on brain monoamine oxidase in various mammalian species.

Brain research 20010706

Disturbance of the prejunctional modulation of cholinergic neurotransmission during chronic granulomatous inflammation of the mouse ileum.

British journal of pharmacology 20010701

Novel histaprodifen analogues as potent histamine H1-receptor agonists in the pithed and in the anaesthetized rat.

Naunyn-Schmiedeberg's archives of pharmacology 20010701

[Identification and characterization of histamine H4 receptor].

Nihon yakurigaku zasshi. Folia pharmacologica Japonica 20010701

The H3 receptor is involved in cholecystokinin inhibition of food intake in rats.

Life sciences 20010615

Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists.

European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20010601

Development of a pharmacophore model for histamine H3 receptor antagonists, using the newly developed molecular modeling program SLATE.

Journal of medicinal chemistry 20010524

Activation of histamine H3 receptors inhibits renal noradrenergic neurotransmission in anesthetized dogs.

American journal of physiology. Regulatory, integrative and comparative physiology 20010501

Histamine H(3) receptor-mediated inhibition of depolarization-induced, dopamine D(1) receptor-dependent release of [(3)H]-gamma-aminobutryic acid from rat striatal slices.

British journal of pharmacology 20010501

[Role of central histamine in amygdaloid kindled seizures].

Nihon yakurigaku zasshi. Folia pharmacologica Japonica 20010501

Genomic organization and characterization of splice variants of the human histamine H3 receptor.

The Biochemical journal 20010415

Different antagonist binding properties of human and rat histamine H3 receptors.

Bioorganic & medicinal chemistry letters 20010409

Cognitive enhancing properties of thioperamide infused into the nucleus basalis magnocellularis of the rat.

Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20010401

Histamine and selective H3-receptor ligands: a possible role in the mechanism and management of epilepsy.

Pharmacology, biochemistry, and behavior 20010401

Role of central histaminergic system in lorazepam withdrawal syndrome in rats.

Pharmacology, biochemistry, and behavior 20010401

Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow.

Molecular pharmacology 20010301

Cloning, expression, and pharmacological characterization of a novel human histamine receptor.

Molecular pharmacology 20010301

Cloning and characterization of a novel human histamine receptor.

The Journal of pharmacology and experimental therapeutics 20010301

Histamine H1 and H2 receptor antagonists accelerate skin barrier repair and prevent epidermal hyperplasia induced by barrier disruption in a dry environment.

The Journal of investigative dermatology 20010201

H3 receptor-mediated inhibition of intestinal acetylcholine release: pharmacological characterization of signal transduction pathways.

Naunyn-Schmiedeberg's archives of pharmacology 20010201

The rat H3 receptor: gene organization and multiple isoforms.

Biochemical and biophysical research communications 20010112

Histamine H(3) receptors depress synaptic transmission in the corticostriatal pathway.

Neuropharmacology 20010101

Cortical acetylcholine release elicited by stimulation of histamine H1 receptors in the nucleus basalis magnocellularis: a dual-probe microdialysis study in the freely moving rat.

The European journal of neuroscience 20010101

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain.

British journal of pharmacology 20001201

Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes.

The Journal of biological chemistry 20001124

Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.

Journal of neurochemistry 20000801

Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles.

The Journal of pharmacology and experimental therapeutics 20000601

Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.

Behavioural brain research 19991001

Therapeutic doses of theophylline exert proconvulsant effects in developing mice.

Brain & development 19970901

Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.

Naunyn-Schmiedeberg's archives of pharmacology 19970201

Effect of adenosine and histamine receptor stimulation on canine histamine release to pentagastrin.

Digestion 19970101

Thioperamide, the selective histamine H3 receptor antagonist, attenuates stimulant-induced locomotor activity in the mouse.

European journal of pharmacology 19940701

Modulation of the intracellular and H3-histamine receptors and chemically-induced seizures in mice.

Agents and actions 19940601

Identification of two H3-histamine receptor subtypes.

Molecular pharmacology 19901101

106243-16-7 | N-Cyclohexyl-4-(1H-imidazol-5-yl)-1-piperidinecarbothioamide

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