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Home > Imidazoles > 102575-24-6
CAS No: 102575-24-6 Catalog No: AG0007T3 MDL No:
Title | Journal |
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Effects of lisdexamfetamine in a rat model of binge-eating. | Journal of psychopharmacology (Oxford, England) 20151201 |
Blockade of α2-adrenoceptors induces Arc gene expression in rat brain in a glutamate receptor-dependent manner: a combined qPCR, in situ hybridisation and immunocytochemistry study. | Neuropharmacology 20121101 |
Lateral septal area α1- and α2-adrenoceptors differently modulate baroreflex activity in unanaesthetized rats. | Experimental physiology 20120901 |
The α₁-, but not α₂-, adrenoceptor in the nucleus accumbens plays an inhibitory role upon the accumbal noradrenaline and dopamine efflux of freely moving rats. | European journal of pharmacology 20120805 |
α1 and α2-adrenoceptors in the medial amygdaloid nucleus modulate differently the cardiovascular responses to restraint stress in rats. | Pharmacological research 20120801 |
The predicted N-terminal signal sequence of the human α₂C-adrenoceptor does not act as a functional cleavable signal peptide. | European journal of pharmacology 20120605 |
The function of alpha-2-adrenoceptors in the rat locus coeruleus is preserved in the chronic constriction injury model of neuropathic pain. | Psychopharmacology 20120501 |
Moxonidine into the lateral parabrachial nucleus reduces renal and hormonal responses to cell dehydration. | Neuroscience 20120419 |
Inhibition of sodium appetite by lipopolysaccharide: involvement of alpha2-adrenoceptors. | American journal of physiology. Regulatory, integrative and comparative physiology 20110701 |
Bed nucleus of the stria terminalis α1- and α2-adrenoceptors differentially modulate the cardiovascular responses to exercise in rats. | Neuroscience 20110317 |
Selective enhancement of mesocortical dopaminergic transmission by noradrenergic drugs: therapeutic opportunities in schizophrenia. | The international journal of neuropsychopharmacology 20110201 |
Adrenergic receptors modulate motoneuron excitability, sensory synaptic transmission and muscle spasms after chronic spinal cord injury. | Journal of neurophysiology 20110101 |
Alpha-adrenoceptor agonistic activity of oxymetazoline and xylometazoline. | Fundamental & clinical pharmacology 20101201 |
α2-adrenergic drugs modulate the binding of [18F]fallypride to dopamine D2/3 receptors in striatum of living mouse. | Synapse (New York, N.Y.) 20100801 |
Investigation of the distribution and function of alpha-adrenoceptors in the sheep isolated internal anal sphincter. | British journal of pharmacology 20100801 |
Adrenergic mechanisms of the Kölliker-Fuse/A7 area on the control of water and sodium intake. | Neuroscience 20091201 |
Insular cortex alpha1-adrenoceptors modulate the parasympathetic component of the baroreflex in unanesthetized rats. | Brain research 20091027 |
Role of the bed nucleus of the stria terminalis in the cardiovascular responses to acute restraint stress in rats. | Stress (Amsterdam, Netherlands) 20090501 |
Modulation of inflammatory response via alpha2-adrenoceptor blockade in acute murine colitis. | Clinical and experimental immunology 20090501 |
Probable involvement of alpha(2C)-adrenoceptor subtype and endogenous opioid peptides in the peripheral antinociceptive effect induced by xylazine. | European journal of pharmacology 20090417 |
Guanidine and 2-aminoimidazoline aromatic derivatives as alpha2-adrenoceptor ligands: searching for structure-activity relationships. | Journal of medicinal chemistry 20090212 |
Activation of alpha(2)-adrenoceptors in the lateral hypothalamus reduces pilocarpine-induced salivation in rats. | Neuroscience letters 20090206 |
Alpha adrenergic modulation on effects of norepinephrine transporter inhibitor reboxetine in five-choice serial reaction time task. | Journal of biomedical science 20090101 |
Interplay among catecholamine systems: dopamine binds to alpha2-adrenergic receptors in birds and mammals. | The Journal of comparative neurology 20081210 |
Differential effects of neonatal norepinephrine lesions on immediate early gene expression in developing and adult rat brain. | Neuroscience 20081210 |
Novel synthesis and pharmacological evaluation as alpha2-adrenoceptor ligands of O-phenylisouronium salts. | Bioorganic & medicinal chemistry 20080901 |
Alpha2-adrenoreceptors profile modulation. 4. From antagonist to agonist behavior. | Journal of medicinal chemistry 20080724 |
Guanidine and 2-aminoimidazoline aromatic derivatives as alpha2-adrenoceptor antagonists. 2. Exploring alkyl linkers for new antidepressants. | Journal of medicinal chemistry 20080612 |
Dopamine binds to alpha(2)-adrenergic receptors in the song control system of zebra finches (Taeniopygia guttata). | Journal of chemical neuroanatomy 20080301 |
Alpha2-adrenergic receptors activate cyclic AMP-response element-binding protein through arachidonic acid metabolism and protein kinase A in a subtype-specific manner. | Journal of neurochemistry 20071101 |
Guanidine and 2-aminoimidazoline aromatic derivatives as alpha(2)-adrenoceptor antagonists, 1: toward new antidepressants with heteroatomic linkers. | Journal of medicinal chemistry 20070906 |
Changes in adrenoreceptors in the prefrontal cortex of subjects with dementia: evidence of compensatory changes. | Neuroscience 20070425 |
Adrenergic drugs modify the level of noradrenaline in the insular cortex and alter extinction of conditioned taste aversion in rats. | Behavioural brain research 20070312 |
Disruption of noradrenergic transmission and the behavioural response to a novel environment in NK1R-/- mice. | The European journal of neuroscience 20070201 |
Pharmacologic characterization of the cloned human trace amine-associated receptor1 (TAAR1) and evidence for species differences with the rat TAAR1. | The Journal of pharmacology and experimental therapeutics 20070101 |
Contribution of imidazoline receptors and alpha2-adrenoceptors in the rostral ventrolateral medulla to sympathetic baroreflex inhibition by systemic rilmenidine. | Journal of hypertension 20070101 |
mRNA expression and binding sites for alpha2-adrenergic receptor subtypes in muscle layers of the ileum and spiral colon of dairy cows. | American journal of veterinary research 20061101 |
Alpha2-adrenergic activation in the lateral parabrachial nucleus induces NaCl intake under conditions of systemic hyperosmolarity. | Neuroscience 20060929 |
Analysis of brain adrenergic receptors in dopamine-beta-hydroxylase knockout mice. | Brain research 20060913 |
Pharmacological characterization and autoradiographic distribution of alpha2-adrenoceptor antagonist [3H]RX 821002 binding sites in the chicken brain. | Neuroscience 20060811 |
Role of CNS alpha1-adrenoceptor activity in central fos responses to novelty. | Synapse (New York, N.Y.) 20060401 |
Ontogenesis of mRNA levels and binding sites of hepatic alpha-adrenoceptors in young cattle. | Domestic animal endocrinology 20060301 |
Norepinephrine transporter knockout-induced up-regulation of brain alpha2A/C-adrenergic receptors. | Journal of neurochemistry 20060201 |
Compensatory changes in the noradrenergic nervous system in the locus ceruleus and hippocampus of postmortem subjects with Alzheimer's disease and dementia with Lewy bodies. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20060111 |
Prenatal cocaine exposure alters alpha2 receptor expression in adolescent rats. | BMC neuroscience 20060101 |
Long-lasting effects of yohimbine on the ejaculatory function in male dogs. | Biomedical research (Tokyo, Japan) 20051001 |
Serotonergic influence on the potentiation of D-amphetamine and apomorphine-induced rotational behavior by the alpha2-adrenoceptor antagonist 2-methoxy idazoxan in hemiparkinsonian rats. | Journal of neural transmission (Vienna, Austria : 1996) 20050901 |
alpha-Adrenergic and muscarinic cholinergic receptors are not involved in the modulation of the parasympathetic baroreflex by the medial prefrontal cortex in rats. | Life sciences 20050812 |
A comparison of neurokinin 1 receptor knock-out (NK1-/-) and wildtype mice: exploratory behaviour and extracellular noradrenaline concentration in the cerebral cortex of anaesthetised subjects. | Neuropharmacology 20050401 |
Estimation of endogenous noradrenaline release in rat brain in vivo using [3H]RX 821002. | Synapse (New York, N.Y.) 20050201 |
Influence of neonatal short-term reduction in brainstem alpha2A-adrenergic receptors on receptor ontogenesis, acoustic startle reflex, and prepulse inhibition in rats. | Behavioral neuroscience 20041201 |
The alpha-2B adrenoceptor in the paraventricular thalamic nucleus is persistently upregulated by chronic psychosocial stress. | Cellular and molecular neurobiology 20041201 |
Treatment with alpha2-adrenoceptor antagonist, 2-methoxy idazoxan, protects 6-hydroxydopamine-induced Parkinsonian symptoms in rats: neurochemical and behavioral evidence. | Behavioural brain research 20041005 |
Clonidine increases caspase-3 mRNA level and DNA fragmentation in the developing rat brainstem. | Brain research. Developmental brain research 20040917 |
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice. | European journal of pharmacology 20040830 |
Effects of tramadol on alpha2-adrenergic receptors in the rat brain. | Brain research 20040806 |
Imidazoline2 (I2) receptor- and alpha2-adrenoceptor-mediated modulation of hypothalamic-pituitary-adrenal axis activity in control and acute restraint stressed rats. | Journal of psychopharmacology (Oxford, England) 20040301 |
Alpha-2 adrenergic receptor development in rat CNS: an autoradiographic study. | Neuroscience 20040101 |
Activation of alpha2-adrenergic receptors into the lateral parabrachial nucleus enhances NaCl intake in rats. | Neuroscience 20040101 |
Attenuation of alpha2A-adrenergic receptor expression in neonatal rat brain by RNA interference or antisense oligonucleotide reduced anxiety in adulthood. | Neuroscience 20040101 |
Androgen-induced norepinephrine release mediating guinea pig seminal vesicle smooth muscle proliferation: potential role of pre-synaptic alpha2-adrenoceptors. | The Prostate 20030915 |
Molecular mechanisms of ligand-receptor interactions in transmembrane domain V of the alpha2A-adrenoceptor. | British journal of pharmacology 20030901 |
Nandrolone treatment decreases the level of rat kidney alpha(1B)-adrenoceptors. | Naunyn-Schmiedeberg's archives of pharmacology 20030801 |
[3H]RX 821002 in human dorsolateral prefrontal cortex: no changes in postmortem tissue from subjects with schizophrenia. | Psychiatry research 20030715 |
Constitutive precoupling to G(i) and increased agonist potency in the alpha(2B)-adrenoceptor. | Biochemical and biophysical research communications 20030711 |
Mechanisms involved in the pressor response to noradrenaline injection into the cingulate cortex of unanesthetized rats. | Neuropharmacology 20030501 |
Stimulation of interleukin-12 production in mouse macrophages via activation of p38 mitogen-activated protein kinase by alpha2-adrenoceptor agonists. | European journal of pharmacology 20030425 |
Piribedil enhances frontocortical and hippocampal release of acetylcholine in freely moving rats by blockade of alpha 2A-adrenoceptors: a dialysis comparison to talipexole and quinelorane in the absence of acetylcholinesterase inhibitors. | The Journal of pharmacology and experimental therapeutics 20030401 |
Central alpha(2) adrenergic receptors and cholinergic-induced salivation in rats. | Brain research bulletin 20030130 |
Importance of imidazoline-preferring receptors in the cardiovascular actions of chronically administered moxonidine, rilmenidine and clonidine in conscious rabbits. | Journal of hypertension 20030101 |
Regional distribution of alpha(2C)-adrenoceptors in brain and spinal cord of control mice and transgenic mice overexpressing the alpha(2C)-subtype: an autoradiographic study with [(3)H]RX821002 and [(3)H]rauwolscine. | Neuroscience 20030101 |
Different roles for Gi and Go proteins in modulation of adenylyl cyclase type-2 activity. | Journal of neurochemistry 20021201 |
Biochemical and functional characterization of alpha-adrenergic receptors in the rabbit vagina. | Life sciences 20021101 |
Effects of medullary alpha2-adrenoceptor blockade in the rat. | European journal of pharmacology 20021025 |
Alpha(1)-adrenoceptor stimulation directly induces growth of vascular wall in vivo. | American journal of physiology. Heart and circulatory physiology 20021001 |
Enhanced stability of wild-type and constitutively active alpha(2A)-adrenoceptors by ligands with agonist, silent and inverse agonist properties. | Naunyn-Schmiedeberg's archives of pharmacology 20020801 |
Alcohol-induced c-Fos expression in the Edinger-Westphal nucleus: pharmacological and signal transduction mechanisms. | The Journal of pharmacology and experimental therapeutics 20020801 |
Different alpha-adrenoceptors mediate migration of vascular smooth muscle cells and adventitial fibroblasts in vitro. | American journal of physiology. Heart and circulatory physiology 20020601 |
Imidazoline(2) (I(2)) binding site- and alpha(2)-adrenoceptor-mediated modulation of central noradrenergic and HPA axis function in control rats and chronically stressed rats with adjuvant-induced arthritis. | Neuropharmacology 20020601 |
Inhibition of pilocarpine-induced salivation in rats by central noradrenaline. | Archives of oral biology 20020601 |
In vivo tonic modulation of the noradrenaline release in the rat cortex by locus coeruleus somatodendritic alpha(2)-adrenoceptors. | European journal of pharmacology 20020510 |
alpha(2B)-Adrenergic receptors activate MAPK and modulate proliferation of primary cultured proximal tubule cells. | American journal of physiology. Renal physiology 20020501 |
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
Seasonal changes in the densities of alpha(2) noradrenergic receptors are inversely related to changes in testosterone and the volumes of song control nuclei in male European starlings. | The Journal of comparative neurology 20020225 |
Mechanisms involved in the water intake-related pressor response in the rat. | Journal of hypertension 20020201 |
Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole. | Journal of medicinal chemistry 20020103 |
Testosterone dependence of salt-induced hypertension in Sabra rats and role of renal alpha(2)-adrenoceptor subtypes. | The Journal of pharmacology and experimental therapeutics 20020101 |
Interactions between cutaneous afferent inputs to a withdrawal reflex in the decerebrated rabbit and their control by descending and segmental systems. | Neuroscience 20020101 |
RX 821002 as a tool for physiological investigation of alpha(2)-adrenoceptors. | CNS drug reviews 20020101 |
In vitro and in vivo impairment of alpha2-adrenergic receptor-dependent antilipolysis by fatty acids in human adipose tissue. | Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme 20011201 |
Evidence for the involvement of central I1 imidazoline receptor in ethanol counteraction of clonidine hypotension in spontaneously hypertensive rats. | Journal of cardiovascular pharmacology 20010901 |
Rabbit alpha2-adrenoceptors: both platelets and adipocytes have alpha2A-pharmacology. | The Journal of pharmacology and experimental therapeutics 20010701 |
Chronic subordination stress in male tree shrews: replacement of testosterone affects behavior and central alpha(2)-adrenoceptors. | Physiology & behavior 20010601 |
The alpha 2 adrenoceptor antagonists RX 821002 and yohimbine delay-dependently impair choice accuracy in a delayed non-matching-to-position task in rats. | Psychopharmacology 20010601 |
Brain alpha(2)-adrenoceptors in monoamine-depleted rats: increased receptor density, G coupling proteins, receptor turnover and receptor mRNA. | British journal of pharmacology 20010401 |
Agonist trafficking of G(i/o)-mediated alpha(2A)-adrenoceptor responses in HEL 92.1.7 cells. | British journal of pharmacology 20010401 |
Alpha2A-adrenoceptor mediated tachypnea in awake goats. | Respiration physiology 20010401 |
Inverse agonist activity at the alpha(2A)-adrenergic receptor. | Molecular pharmacology 20010301 |
Receptor phosphorylation mediates estradiol reduction of alpha2-adrenoceptor coupling to G protein in the hypothalamus of female rats. | Endocrine 20010301 |
A robust GTP-induced shift in alpha(2)-adrenoceptor agonist affinity in tissue sections from rat brain. | Journal of neuroscience methods 20010215 |
Chronic treatment with desipramine facilitates its effect on extracellular noradrenaline in the rat hippocampus: studies on the role of presynaptic alpha2-adrenoceptors. | Naunyn-Schmiedeberg's archives of pharmacology 20010101 |
alpha2C adrenoceptors inhibit adenylyl cyclase in mouse striatum: potential activation by dopamine. | The Journal of pharmacology and experimental therapeutics 19990601 |
Modulation of agonist binding to recombinant human alpha2-adrenoceptors by sodium ions. | Biochimica et biophysica acta 19981119 |
The role of alpha2-adrenoceptor antagonism in the anti-cataleptic properties of the atypical neuroleptic agent, clozapine, in the rat. | British journal of pharmacology 19980801 |
Characterization of the allosteric interactions between antagonists and amiloride analogues at the human alpha2A-adrenergic receptor. | Molecular pharmacology 19980501 |
Buffers differentially alter the binding of [3H]rauwolscine and [3H]RX821002 to the alpha-2 adrenergic receptor subtypes. | The Journal of pharmacology and experimental therapeutics 19960901 |
A comparative study of the reversal by different alpha 2-adrenoceptor antagonists of the central sympatho-inhibitory effect of clonidine. | British journal of pharmacology 19960201 |
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors. | The Journal of pharmacology and experimental therapeutics 19941201 |
Further characterization of human alpha 2-adrenoceptor subtypes: [3H]RX821002 binding and definition of additional selective drugs. | European journal of pharmacology 19940124 |
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