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100-76-5 | Quinuclidine

CAS No: 100-76-5 Catalog No: AG00006Q MDL No:MFCD00006690

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Title Journal
Excited-state proton transfer and ion pair formation in a Cinchona organocatalyst. Physical chemistry chemical physics : PCCP 20121005
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Scope of stereoselective Mn-mediated radical addition to chiral hydrazones and application in a formal synthesis of quinine. The Journal of organic chemistry 20120406
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Making SharePoint® Chemically Aware™. Journal of cheminformatics 20120101
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The role of neurokinin-1 receptor in the microenvironment of inflammation and cancer. TheScientificWorldJournal 20120101
Reactions of nitroxides XIII: Synthesis of the Morita-Baylis-Hillman adducts bearing a nitroxyl moiety using 4-acryloyloxy-2,2,6,6-tetramethylpiperidine-1-oxyl as a starting compound, and DABCO and quinuclidine as catalysts. Beilstein journal of organic chemistry 20120101
Stepwise effective molarities in porphyrin oligomer complexes: preorganization results in exceptionally strong chelate cooperativity. Journal of the American Chemical Society 20111228
Asymmetric hydrogenation on chirally modified Pt: origin of hydrogen in the N-H-O interaction between cinchonidine and ketone. Journal of the American Chemical Society 20111214
New spirocyclic Δ²-isoxazoline derivatives related to selective agonists of α7 neuronal nicotinic acetylcholine receptors. European journal of medicinal chemistry 20111201
Diastereodivergent asymmetric sulfa-Michael additions of α-branched enones using a single chiral organic catalyst. Journal of the American Chemical Society 20111109
Identification of the best-suited leaving group for the diastereoselective synthesis of glycidic amides from stabilised ammonium ylides and aldehydes. Organic & biomolecular chemistry 20111021
Designing the synthesis of catalytically active Ti-β by using various new templates in the presence of fluoride anion. Physical chemistry chemical physics : PCCP 20110928
Theoretical investigation on mechanism of asymmetric Michael addition of malononitrile to chalcones catalyzed by Cinchona alkaloid aluminium(III) complex. Organic & biomolecular chemistry 20110921
Effect of stereogenic centers on the self-sorting, depolymerization, and atropisomerization kinetics of porphyrin-based aggregates. Journal of the American Chemical Society 20110810
Two squalene synthase inhibitors, E5700 and ER-119884, interfere with cellular proliferation and induce ultrastructural and lipid profile alterations in a Candida tropicalis strain resistant to fluconazole, itraconazole, and amphotericin B. Journal of infection and chemotherapy : official journal of the Japan Society of Chemotherapy 20110801
Intermolecular radical addition to N-acylhydrazones as a stereocontrol strategy for alkaloid synthesis: formal synthesis of quinine. Organic & biomolecular chemistry 20110607
Discovery of novel quaternary ammonium derivatives of (3R)-quinuclidinyl carbamates as potent and long acting muscarinic antagonists. Bioorganic & medicinal chemistry letters 20110601
The hydroxyl functionality and a rigid proximal N are required for forming a novel non-covalent quinine-heme complex. Journal of inorganic biochemistry 20110301
Synthetic arylquinuclidine derivatives exhibit antifungal activity against Candida albicans, Candida tropicalis and Candida parapsilopsis. Annals of clinical microbiology and antimicrobials 20110101
Synthesis and in vitro evaluation of novel nortropane derivatives as potential radiotracers for muscarinic m(2) receptors. International journal of molecular imaging 20110101
Squalene synthase inhibitors: An update on the search for new antihyperlipidemic and antiatherosclerotic agents. Current medicinal chemistry 20110101
Antiproliferative, Ultrastructural, and Physiological Effects of Amiodarone on Promastigote and Amastigote Forms of Leishmania amazonensis. Molecular biology international 20110101
Structural analysis of prolyl oligopeptidases using molecular docking and dynamics: insights into conformational changes and ligand binding. PloS one 20110101
Antiangiogenic properties of substituted (Z)-(±)-2-(N-benzylindol-3-ylmethylene)quinuclidin-3-ol/one analogs and their derivatives. Bioorganic & medicinal chemistry letters 20101215
Surface plasmon resonance biosensor based fragment screening using acetylcholine binding protein identifies ligand efficiency hot spots (LE hot spots) by deconstruction of nicotinic acetylcholine receptor α7 ligands. Journal of medicinal chemistry 20101014
Unexpected enantioseparation of mandelic acids and their derivatives on 1,2,3-triazolo-linked quinine tert-butyl carbamate anion exchange-type chiral stationary phase. Journal of separation science 20100901
3-D-QSAR and docking studies on the neuronal choline transporter. Bioorganic & medicinal chemistry letters 20100815
Multiple species metabolism of PHA-568487, a selective alpha 7 nicotinic acetylcholine receptor agonist. Drug metabolism letters 20100801
Binary complexes of tertiary amines with phenylacetylene. Dispersion wins over electrostatics. Physical chemistry chemical physics : PCCP 20100621
Using the pyridine and quinuclidine scaffolds for superbases: a DFT study. The Journal of organic chemistry 20100416
Enantioselective synthesis of a chiral C(3)-symmetric bridgehead amine. Organic letters 20100416
Chiral recognition in cinchona alkaloid protonated dimers: mass spectrometry and UV photodissociation studies. The journal of physical chemistry. A 20100311
HPLC method for determination of fluorescence derivatives of cortisol, cortisone and their tetrahydro- and allo-tetrahydro-metabolites in biological fluids. Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20100201
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Cucurbit[7]uril host-guest complexes of cholines and phosphonium cholines in aqueous solution. Organic & biomolecular chemistry 20100107
Delineation of downstream signalling components during acrosome reaction mediated by heat solubilized human zona pellucida. Reproductive biology and endocrinology : RB&E 20100101
Generating a generation of proteasome inhibitors: from microbial fermentation to total synthesis of salinosporamide a (marizomib) and other salinosporamides. Marine drugs 20100101
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Host-guest complexes and pseudorotaxanes of cucurbit[7]uril with acetylcholinesterase inhibitors. The Journal of organic chemistry 20091106
Atmospheric heterogeneous stereochemistry. Journal of the American Chemical Society 20090930
Organocatalytic activity of cinchona alkaloids: which nitrogen is more nucleophilic? The Journal of organic chemistry 20090918
Tertiary amine and N-heterocyclic carbene coordinated haloalanes--synthesis, structure, and application. Chemistry (Weinheim an der Bergstrasse, Germany) 20090914
Influence of peripheral groups on the physical and chemical behavior of cinchona alkaloids. The journal of physical chemistry. B 20090827
Stereocontrolled synthesis and pharmacological evaluation of cis-2,6-diphenethyl-1-azabicyclo[2.2.2]octanes as lobelane analogues. The Journal of organic chemistry 20090821
Fluorinated quinine alkaloids: synthesis, X-ray structure analysis and antimalarial parasite chemotherapy. Chemistry (Weinheim an der Bergstrasse, Germany) 20090803
New, improved treatments for Chagas disease: from the R&D pipeline to the patients. PLoS neglected tropical diseases 20090701
Discovery of novel 1-azoniabicyclo[2.2.2]octane muscarinic acetylcholine receptor antagonists. Journal of medicinal chemistry 20090423
Structure and rheology of cationic molecular hydrogels of quinuclidine grafted bile salts. Influence of the ionic strength and counter-ion type. The journal of physical chemistry. B 20090409
1-Pyridine- and 1-quinuclidine-1-boraadamantane as models for derivatives of 1-borabicyclo[2.2.2]octane. Experimental and theoretical evaluation of the B-N fragment as a polar isosteric substitution for the C-C group in liquid crystal compounds. The Journal of organic chemistry 20090220
Fluorescence quenching of CdSe quantum dots by tertiary amines and their surface binding effect. Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20090101
Efficient N-arylation/dealkylation of electron deficient heteroaryl chlorides and bicyclic tertiary amines under microwave irradiation. Journal of combinatorial chemistry 20090101
Management of postoperative nausea and vomiting: focus on palonosetron. Therapeutics and clinical risk management 20090101
Sterol Biosynthesis Pathway as Target for Anti-trypanosomatid Drugs. Interdisciplinary perspectives on infectious diseases 20090101
The solubilisation of boar sperm membranes by different detergents - a microscopic, MALDI-TOF MS, (31)P NMR and PAGE study on membrane lysis, extraction efficiency, lipid and protein composition. Lipids in health and disease 20090101
High-frequency Broadband Modulations of Electroencephalographic Spectra. Frontiers in human neuroscience 20090101
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Use of molecular electrostatic potential for quantitative assessment of inductive effect. Physical chemistry chemical physics : PCCP 20081121
Polyepichlorhydrin membranes for alkaline fuel cells: sorption and conduction properties. The journal of physical chemistry. B 20081002
Interaction energies and dynamics of acid-base pairs isolated in cavitands. The Journal of organic chemistry 20080905
The crystal structure of halofantrine-ferriprotoporphyrin IX and the mechanism of action of arylmethanol antimalarials. Journal of inorganic biochemistry 20080801
Application of the PM6 method to modeling the solid state. Journal of molecular modeling 20080601
(R)-(-)-3-Hydroxy-quinuclidinium chloride. Acta crystallographica. Section E, Structure reports online 20080501
3-Chloro-quinuclidinium chloride. Acta crystallographica. Section E, Structure reports online 20080501
alpha7 nicotinic acetylcholine receptor agonist properties of tilorone and related tricyclic analogues. British journal of pharmacology 20080301
Quinuclidine complex with alpha-cyclodextrin: a diffusion and 13C NMR relaxation study. Magnetic resonance in chemistry : MRC 20080301
Synthetic efforts for stereo structure determination of cytotoxic marine natural product pericosines as metabolites of Periconia sp. from sea hare. International journal of molecular sciences 20080301
1-[(Diethyl-amino-carbon-yl)meth-yl]-2-[hydr-oxy(6-methoxy-quinolin-4-yl)meth-yl]-5-vinyl-1-azoniabicyclo-[2.2.2]octane chloride monohydrate. Acta crystallographica. Section E, Structure reports online 20080201
Huge deuterated effect on permittivity in a metal-organic framework. Chemistry (Weinheim an der Bergstrasse, Germany) 20080101
Mixed-ligand metal-organic frameworks with large pores: gas sorption properties and single-crystal-to-single-crystal transformation on guest exchange. Chemistry (Weinheim an der Bergstrasse, Germany) 20080101
Synthesis and characterization of new nitrogen-donor-stabilized N-silylphosphoranimine cations. Inorganic chemistry 20071112
Adducts of rhodium(II) tetraacetate with some nitrogenous organic ligands: application of natural abundance 15N and 13C CPMAS NMR spectroscopy. Solid state nuclear magnetic resonance 20071001
Role of guiding groups in cinchona-modified platinum for controlling the sense of enantiodifferentiation in the hydrogenation of ketones. Journal of the American Chemical Society 20070829
Metabolism, pharmacokinetics, and excretion of a nonpeptidic substance P receptor antagonist, ezlopitant, in normal healthy male volunteers: characterization of polar metabolites by chemical derivatization with dansyl chloride. Drug metabolism and disposition: the biological fate of chemicals 20070701
Molecular structures of free quinuclidine and its adducts with metal trihydrides, MH3 (M=B, Al or Ga), studied by gas-phase electron diffraction, X-ray diffraction and quantum chemical calculations. Dalton transactions (Cambridge, England : 2003) 20070507
Quinuclidines as selective agonists for alpha-7 nicotinic acetylcholine receptors. Bioorganic & medicinal chemistry letters 20070315
Investigation of the stability of the M-H-B bond in borane sigma complexes [M(CO)5(eta1-BH2R.L)] and [CpMn(CO)2(eta1-BH2R.L)] (M=Cr, W; L=tertiary amine or phosphine): substituent and Lewis base effects. Chemistry (Weinheim an der Bergstrasse, Germany) 20070101
Effectiveness of low-dose doxycycline (LDD) on clinical symptoms of Sjögren's syndrome: a randomized, double-blind, placebo controlled cross-over study. Journal of negative results in biomedicine 20070101
The nature of the chemical bond in linear three-body systems: from i3- to mixed chalcogen/halogen and trichalcogen moieties. Bioinorganic chemistry and applications 20070101
A synthetic mimic of protein inner space: buried polar interactions in a deep water-soluble host. Journal of the American Chemical Society 20061206
Synthetic studies on quinine: quinuclidine construction via a ketone enolate regio- and diastereoselective Pd-mediated allylic alkylation. Organic letters 20060831
Method for enantiomeric purity of a quinuclidine candidate drug by capillary electrophoresis. Journal of separation science 20060801
RP-HPLC method with fluorescence detection for determination of small quantities of triamcinolone in plasma in presence of endogenous steroids after derivatization with 9-anthroyl nitrile; pharmacokinetic studies. Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20060724
Antiproliferative activities of two novel quinuclidine inhibitors against Toxoplasma gondii tachyzoites in vitro. The Journal of antimicrobial chemotherapy 20060701
A generalized two-point H-bonding model for catalytic stereoselective hydrogenation of activated ketones on chirally modified platinum. Journal of the American Chemical Society 20060614
Pyridinium, imidazolium and quinuclidinium compounds: toxicity and antidotal effects against the nerve agents Tabun and Soman. Arhiv za higijenu rada i toksikologiju 20060601
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Zona pellucida from fertilised human oocytes induces a voltage-dependent calcium influx and the acrosome reaction in spermatozoa, but cannot be penetrated by sperm. BMC developmental biology 20060101
Structure and reactivity of trans-bis[2-(2-chloroethyl)pyridine]palladium chloride (1). A study on the elimination reaction of 1 and 2-(2-chloroethyl)pyridine induced by quinuclidine in acetonitrile. The Journal of organic chemistry 20051223
Rate-limiting proton-transfer in the sigma-adduct forming reactions of 1,3,5-trinitrobenzene and 4-nitrobenzofuroxan with substituted anilines in dimethyl sulfoxide. Organic & biomolecular chemistry 20051107
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Orientational isomers of alpha-cyclodextrin [2]semi-rotaxanes with asymmetric dicationic threads. Organic & biomolecular chemistry 20050421
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